Peringatan Keamanan

Oral, LD50 = 238 mg/kg (mouse); Oral, LD50 = 781 mg/kg (rabbit); Oral, LD50 = 245 mg/kg (rat); Oral, LD50 = 375 mg/kg (rat)

Phenylbutazone

DB00812

small molecule approved vet_approved

Deskripsi

A drug that has anti-inflammatory, antipyretic, and analgesic activities. It is especially effective in the treatment of ankylosing spondylitis. It also is useful in rheumatoid arthritis and Reiter's syndrome (investigational indication). Although phenylbutazone is effective in gouty arthritis, risk/benefit considerations indicate that this drug should not be employed for this disease. (From AMA Drug Evaluations Annual, 1994, p1822)

Struktur Molekul 2D

Berat 308.3743
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol.
  • 2. Take with food. Food reduces irritation.

Interaksi Obat

1703 Data
Aripiprazole The metabolism of Aripiprazole can be increased when combined with Phenylbutazone.
Aripiprazole lauroxil The metabolism of Aripiprazole lauroxil can be increased when combined with Phenylbutazone.
Midodrine The risk or severity of hypertension can be increased when Midodrine is combined with Phenylbutazone.
Isoetharine The risk or severity of hypertension can be increased when Isoetharine is combined with Phenylbutazone.
Zolmitriptan The risk or severity of hypertension can be increased when Zolmitriptan is combined with Phenylbutazone.
Norepinephrine The risk or severity of hypertension can be increased when Norepinephrine is combined with Phenylbutazone.
Phenylephrine The risk or severity of hypertension can be increased when Phenylephrine is combined with Phenylbutazone.
Phenylpropanolamine The risk or severity of hypertension can be increased when Phenylpropanolamine is combined with Phenylbutazone.
Droperidol The risk or severity of hypertension can be increased when Droperidol is combined with Phenylbutazone.
Doxapram The risk or severity of hypertension can be increased when Doxapram is combined with Phenylbutazone.
Atropine The risk or severity of hypertension can be increased when Atropine is combined with Phenylbutazone.
Linezolid The risk or severity of hypertension can be increased when Linezolid is combined with Phenylbutazone.
Metaraminol The risk or severity of hypertension can be increased when Metaraminol is combined with Phenylbutazone.
Furazolidone The risk or severity of hypertension can be increased when Furazolidone is combined with Phenylbutazone.
Thioridazine The risk or severity of hypertension can be increased when Thioridazine is combined with Phenylbutazone.
Nicergoline The risk or severity of hypertension can be increased when Nicergoline is combined with Phenylbutazone.
Methoxamine The risk or severity of hypertension can be increased when Methoxamine is combined with Phenylbutazone.
Isoflurane The risk or severity of hypertension can be increased when Isoflurane is combined with Phenylbutazone.
Propiomazine The risk or severity of hypertension can be increased when Propiomazine is combined with Phenylbutazone.
Minaprine The risk or severity of hypertension can be increased when Minaprine is combined with Phenylbutazone.
Orciprenaline The risk or severity of hypertension can be increased when Phenylbutazone is combined with Orciprenaline.
Phenmetrazine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Phenmetrazine.
Trifluoperazine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Trifluoperazine.
Pseudoephedrine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Pseudoephedrine.
Ritodrine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Ritodrine.
Flupentixol The risk or severity of hypertension can be increased when Phenylbutazone is combined with Flupentixol.
Remifentanil The risk or severity of hypertension can be increased when Phenylbutazone is combined with Remifentanil.
Bitolterol The risk or severity of hypertension can be increased when Phenylbutazone is combined with Bitolterol.
Oxymetazoline The risk or severity of hypertension can be increased when Phenylbutazone is combined with Oxymetazoline.
Diethylpropion The risk or severity of hypertension can be increased when Phenylbutazone is combined with Diethylpropion.
Naratriptan The risk or severity of hypertension can be increased when Phenylbutazone is combined with Naratriptan.
Frovatriptan The risk or severity of hypertension can be increased when Phenylbutazone is combined with Frovatriptan.
Isoprenaline The risk or severity of hypertension can be increased when Phenylbutazone is combined with Isoprenaline.
Arbutamine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Arbutamine.
Desflurane The risk or severity of hypertension can be increased when Phenylbutazone is combined with Desflurane.
Isocarboxazid The risk or severity of hypertension can be increased when Phenylbutazone is combined with Isocarboxazid.
Lisdexamfetamine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Lisdexamfetamine.
Fenoterol The risk or severity of hypertension can be increased when Phenylbutazone is combined with Fenoterol.
Pirbuterol The risk or severity of hypertension can be increased when Phenylbutazone is combined with Pirbuterol.
Ephedra sinica root The risk or severity of hypertension can be increased when Phenylbutazone is combined with Ephedra sinica root.
Ephedrine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Ephedrine.
Mephentermine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Mephentermine.
Procaterol The risk or severity of hypertension can be increased when Phenylbutazone is combined with Procaterol.
Methotrimeprazine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Methotrimeprazine.
Clenbuterol The risk or severity of hypertension can be increased when Phenylbutazone is combined with Clenbuterol.
Bambuterol The risk or severity of hypertension can be increased when Phenylbutazone is combined with Bambuterol.
MMDA The risk or severity of hypertension can be increased when Phenylbutazone is combined with MMDA.
Midomafetamine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Midomafetamine.
2,5-Dimethoxy-4-ethylamphetamine The risk or severity of hypertension can be increased when Phenylbutazone is combined with 2,5-Dimethoxy-4-ethylamphetamine.
4-Methoxyamphetamine The risk or severity of hypertension can be increased when Phenylbutazone is combined with 4-Methoxyamphetamine.
4-Bromo-2,5-dimethoxyamphetamine The risk or severity of hypertension can be increased when Phenylbutazone is combined with 4-Bromo-2,5-dimethoxyamphetamine.
Tenamfetamine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Tenamfetamine.
Chlorphentermine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Chlorphentermine.
Dextroamphetamine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Dextroamphetamine.
Phendimetrazine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Phendimetrazine.
Periciazine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Periciazine.
Acepromazine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Acepromazine.
Thioproperazine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Thioproperazine.
Epicaptopril The risk or severity of hypertension can be increased when Phenylbutazone is combined with Epicaptopril.
Clorgiline The risk or severity of hypertension can be increased when Phenylbutazone is combined with Clorgiline.
1-benzylimidazole The risk or severity of hypertension can be increased when Phenylbutazone is combined with 1-benzylimidazole.
Nialamide The risk or severity of hypertension can be increased when Phenylbutazone is combined with Nialamide.
Amibegron The risk or severity of hypertension can be increased when Phenylbutazone is combined with Amibegron.
Naluzotan The risk or severity of hypertension can be increased when Phenylbutazone is combined with Naluzotan.
Pizotifen The risk or severity of hypertension can be increased when Phenylbutazone is combined with Pizotifen.
Solabegron The risk or severity of hypertension can be increased when Phenylbutazone is combined with Solabegron.
Esmirtazapine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Esmirtazapine.
Nitrous oxide The risk or severity of hypertension can be increased when Phenylbutazone is combined with Nitrous oxide.
Xylometazoline The risk or severity of hypertension can be increased when Phenylbutazone is combined with Xylometazoline.
Dexmethylphenidate The risk or severity of hypertension can be increased when Phenylbutazone is combined with Dexmethylphenidate.
Isometheptene The risk or severity of hypertension can be increased when Phenylbutazone is combined with Isometheptene.
Levonordefrin The risk or severity of hypertension can be increased when Phenylbutazone is combined with Levonordefrin.
Naphazoline The risk or severity of hypertension can be increased when Phenylbutazone is combined with Naphazoline.
Tetryzoline The risk or severity of hypertension can be increased when Phenylbutazone is combined with Tetryzoline.
Cinitapride The risk or severity of hypertension can be increased when Phenylbutazone is combined with Cinitapride.
Tyramine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Tyramine.
Adrafinil The risk or severity of hypertension can be increased when Phenylbutazone is combined with Adrafinil.
Isoxsuprine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Isoxsuprine.
Ifenprodil The risk or severity of hypertension can be increased when Phenylbutazone is combined with Ifenprodil.
Hexoprenaline The risk or severity of hypertension can be increased when Phenylbutazone is combined with Hexoprenaline.
Etilefrine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Etilefrine.
Cirazoline The risk or severity of hypertension can be increased when Phenylbutazone is combined with Cirazoline.
Synephrine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Synephrine.
Hydracarbazine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Hydracarbazine.
Benmoxin The risk or severity of hypertension can be increased when Phenylbutazone is combined with Benmoxin.
Mebanazine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Mebanazine.
Octamoxin The risk or severity of hypertension can be increased when Phenylbutazone is combined with Octamoxin.
Pheniprazine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Pheniprazine.
Phenoxypropazine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Phenoxypropazine.
Pivhydrazine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Pivhydrazine.
Safrazine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Safrazine.
Caroxazone The risk or severity of hypertension can be increased when Phenylbutazone is combined with Caroxazone.
Doxofylline The risk or severity of hypertension can be increased when Phenylbutazone is combined with Doxofylline.
Iofetamine I-123 The risk or severity of hypertension can be increased when Phenylbutazone is combined with Iofetamine I-123.
Racepinephrine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Racepinephrine.
Amitraz The risk or severity of hypertension can be increased when Phenylbutazone is combined with Amitraz.
Medetomidine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Medetomidine.
Xylazine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Xylazine.
Atipamezole The risk or severity of hypertension can be increased when Phenylbutazone is combined with Atipamezole.
Ractopamine The risk or severity of hypertension can be increased when Phenylbutazone is combined with Ractopamine.

Target Protein

Prostaglandin G/H synthase 1 PTGS1
Prostaglandin G/H synthase 2 PTGS2
Prostacyclin synthase PTGIS

Referensi & Sumber

Synthesis reference: Dieter Rahtz, Henning Koch, Erich Gerhards, "Hydroxy phenylbutazone derivatives and their preparation." U.S. Patent US3968219, issued January, 1971.

Contoh Produk & Brand

Produk: 5 • International brands: 1
Produk
  • Alka Phenyl Tab
    Tablet • - • Oral • Canada • Approved
  • Alka Phenylbutazone Tab
    Tablet • - • Oral • Canada • Approved
  • Apo Phenylbutazone Tab 100mg
    Tablet • 100 mg • Oral • Canada • Generic • Approved
  • Novo-butazone Tab 100mg
    Tablet • 100 mg • Oral • Canada • Generic • Approved
  • Phenylone Plus Tab
    Tablet • - • Oral • Canada • Approved
International Brands
  • Azolid

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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