Peringatan Keamanan

LD50=760 mg/kg (Orally in rats). Signs of overdose include dilated and sluggish pupils, warm, dry skin, facial flushing, decreased secretions of the mouth, pharynx, nose, and bronchi, foul-smelling breath, elevated temperature, tachycardia, cardiac arrhythmias, decreased bowel sounds, urinary retention, delirium, disorientation, anxiety, hallucinations, illusions, confusion, incoherence, agitation, hyperactivity, ataxia, loss of memory, paranoia, combativeness, and seizures.

Biperiden

DB00810

small molecule approved investigational

Deskripsi

A muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteriosclerotic, idiopathic, and postencephalitic parkinsonism. It has also been used to alleviate extrapyramidal symptoms induced by phenothiazine derivatives and reserpine.

Struktur Molekul 2D

Berat 311.4611
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

87% bioavailability

Metabolisme

The metabolism of biperiden is not completely understood, but does involve hydroxylation.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol.
  • 2. Take with food.

Interaksi Obat

717 Data
Aclidinium The risk or severity of adverse effects can be increased when Biperiden is combined with Aclidinium.
Mianserin Mianserin may increase the anticholinergic activities of Biperiden.
Mirabegron The risk or severity of urinary retention can be increased when Biperiden is combined with Mirabegron.
Potassium chloride The risk or severity of gastrointestinal ulceration can be increased when Biperiden is combined with Potassium chloride.
Pramlintide The risk or severity of reduced gastrointestinal motility can be increased when Pramlintide is combined with Biperiden.
Secretin porcine The therapeutic efficacy of Secretin porcine can be decreased when used in combination with Biperiden.
Tiotropium The risk or severity of adverse effects can be increased when Biperiden is combined with Tiotropium.
Topiramate The risk or severity of hyperthermia and oligohydrosis can be increased when Biperiden is combined with Topiramate.
Umeclidinium The risk or severity of adverse effects can be increased when Biperiden is combined with Umeclidinium.
Methylphenidate The risk or severity of adverse effects can be increased when Methylphenidate is combined with Biperiden.
Dexmethylphenidate The risk or severity of adverse effects can be increased when Dexmethylphenidate is combined with Biperiden.
Metoclopramide The therapeutic efficacy of Biperiden can be decreased when used in combination with Metoclopramide.
Atomoxetine The metabolism of Atomoxetine can be decreased when combined with Biperiden.
Glycopyrronium The risk or severity of adverse effects can be increased when Biperiden is combined with Glycopyrronium.
Botulinum toxin type A The risk or severity of adverse effects can be increased when Biperiden is combined with Botulinum toxin type A.
Glucagon Biperiden may increase the gastrointestinal motility reducing activities of Glucagon.
Sulpiride Biperiden may increase the anticholinergic activities of Sulpiride.
Botulinum toxin type B The risk or severity of adverse effects can be increased when Biperiden is combined with Botulinum toxin type B.
Eluxadoline The risk or severity of constipation can be increased when Biperiden is combined with Eluxadoline.
Ramosetron The risk or severity of constipation can be increased when Biperiden is combined with Ramosetron.
Naltrexone The risk or severity of adverse effects can be increased when Biperiden is combined with Naltrexone.
Bezitramide The risk or severity of adverse effects can be increased when Biperiden is combined with Bezitramide.
Hydromorphone The risk or severity of adverse effects can be increased when Biperiden is combined with Hydromorphone.
Butorphanol The risk or severity of adverse effects can be increased when Biperiden is combined with Butorphanol.
Pentazocine The risk or severity of adverse effects can be increased when Biperiden is combined with Pentazocine.
Sufentanil The risk or severity of adverse effects can be increased when Biperiden is combined with Sufentanil.
Alfentanil The risk or severity of adverse effects can be increased when Biperiden is combined with Alfentanil.
Fentanyl The risk or severity of adverse effects can be increased when Biperiden is combined with Fentanyl.
Nalbuphine The risk or severity of adverse effects can be increased when Biperiden is combined with Nalbuphine.
Levorphanol The risk or severity of adverse effects can be increased when Biperiden is combined with Levorphanol.
Remifentanil The risk or severity of adverse effects can be increased when Biperiden is combined with Remifentanil.
Diphenoxylate The risk or severity of adverse effects can be increased when Biperiden is combined with Diphenoxylate.
Dezocine The risk or severity of adverse effects can be increased when Biperiden is combined with Dezocine.
Levacetylmethadol The risk or severity of adverse effects can be increased when Biperiden is combined with Levacetylmethadol.
Methadyl acetate The risk or severity of adverse effects can be increased when Biperiden is combined with Methadyl acetate.
Dihydroetorphine The risk or severity of adverse effects can be increased when Biperiden is combined with Dihydroetorphine.
Diamorphine The risk or severity of adverse effects can be increased when Biperiden is combined with Diamorphine.
Etorphine The risk or severity of adverse effects can be increased when Biperiden is combined with Etorphine.
Dextromoramide The risk or severity of adverse effects can be increased when Biperiden is combined with Dextromoramide.
Desomorphine The risk or severity of adverse effects can be increased when Biperiden is combined with Desomorphine.
Carfentanil The risk or severity of adverse effects can be increased when Biperiden is combined with Carfentanil.
Alphacetylmethadol The risk or severity of adverse effects can be increased when Biperiden is combined with Alphacetylmethadol.
Dihydromorphine The risk or severity of adverse effects can be increased when Biperiden is combined with Dihydromorphine.
Ketobemidone The risk or severity of adverse effects can be increased when Biperiden is combined with Ketobemidone.
DPDPE The risk or severity of adverse effects can be increased when Biperiden is combined with DPDPE.
Lofentanil The risk or severity of adverse effects can be increased when Biperiden is combined with Lofentanil.
Normethadone The risk or severity of adverse effects can be increased when Biperiden is combined with Normethadone.
Piritramide The risk or severity of adverse effects can be increased when Biperiden is combined with Piritramide.
Alphaprodine The risk or severity of adverse effects can be increased when Biperiden is combined with Alphaprodine.
Nicomorphine The risk or severity of adverse effects can be increased when Biperiden is combined with Nicomorphine.
Meptazinol The risk or severity of adverse effects can be increased when Biperiden is combined with Meptazinol.
Phenoperidine The risk or severity of adverse effects can be increased when Biperiden is combined with Phenoperidine.
Phenazocine The risk or severity of adverse effects can be increased when Biperiden is combined with Phenazocine.
Tilidine The risk or severity of adverse effects can be increased when Biperiden is combined with Tilidine.
Carfentanil, C-11 The risk or severity of adverse effects can be increased when Biperiden is combined with Carfentanil, C-11.
Codeine The risk or severity of adverse effects can be increased when Biperiden is combined with Codeine.
Methadone The risk or severity of adverse effects can be increased when Biperiden is combined with Methadone.
Meperidine The risk or severity of adverse effects can be increased when Biperiden is combined with Meperidine.
Oxycodone The risk or severity of adverse effects can be increased when Biperiden is combined with Oxycodone.
Dextropropoxyphene The risk or severity of adverse effects can be increased when Biperiden is combined with Dextropropoxyphene.
Buprenorphine The risk or severity of adverse effects can be increased when Biperiden is combined with Buprenorphine.
Hydrocodone The risk or severity of adverse effects can be increased when Biperiden is combined with Hydrocodone.
Oxymorphone The risk or severity of adverse effects can be increased when Biperiden is combined with Oxymorphone.
Ethylmorphine The risk or severity of adverse effects can be increased when Biperiden is combined with Ethylmorphine.
Dihydrocodeine The risk or severity of adverse effects can be increased when Biperiden is combined with Dihydrocodeine.
Tapentadol The risk or severity of urinary retention and constipation can be increased when Biperiden is combined with Tapentadol.
Opium The risk or severity of adverse effects can be increased when Biperiden is combined with Opium.
Benzhydrocodone The risk or severity of adverse effects can be increased when Biperiden is combined with Benzhydrocodone.
Morphine The risk or severity of adverse effects can be increased when Biperiden is combined with Morphine.
Naloxegol The risk or severity of adverse effects can be increased when Biperiden is combined with Naloxegol.
Mecamylamine The risk or severity of adverse effects can be increased when Mecamylamine is combined with Biperiden.
Tropicamide The risk or severity of adverse effects can be increased when Tropicamide is combined with Biperiden.
Amantadine The risk or severity of adverse effects can be increased when Biperiden is combined with Amantadine.
Cyclopentolate The risk or severity of adverse effects can be increased when Biperiden is combined with Cyclopentolate.
Pentolinium The risk or severity of adverse effects can be increased when Biperiden is combined with Pentolinium.
Trimethaphan The risk or severity of adverse effects can be increased when Biperiden is combined with Trimethaphan.
Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione The risk or severity of adverse effects can be increased when Biperiden is combined with Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione.
Agmatine The risk or severity of adverse effects can be increased when Biperiden is combined with Agmatine.
Homatropine The risk or severity of adverse effects can be increased when Biperiden is combined with Homatropine.
Batefenterol The risk or severity of adverse effects can be increased when Biperiden is combined with Batefenterol.
Chlorphenoxamine The risk or severity of adverse effects can be increased when Biperiden is combined with Chlorphenoxamine.
Quinidine The risk or severity of adverse effects can be increased when Biperiden is combined with Quinidine.
Cimetropium The risk or severity of adverse effects can be increased when Biperiden is combined with Cimetropium.
Methyclothiazide The serum concentration of Methyclothiazide can be increased when it is combined with Biperiden.
Chlorthalidone The serum concentration of Chlorthalidone can be increased when it is combined with Biperiden.
Bendroflumethiazide The serum concentration of Bendroflumethiazide can be increased when it is combined with Biperiden.
Metolazone The serum concentration of Metolazone can be increased when it is combined with Biperiden.
Benzthiazide The serum concentration of Benzthiazide can be increased when it is combined with Biperiden.
Hydroflumethiazide The serum concentration of Hydroflumethiazide can be increased when it is combined with Biperiden.
Indapamide The serum concentration of Indapamide can be increased when it is combined with Biperiden.
Chlorothiazide The serum concentration of Chlorothiazide can be increased when it is combined with Biperiden.
Hydrochlorothiazide The serum concentration of Hydrochlorothiazide can be increased when it is combined with Biperiden.
Trichlormethiazide The serum concentration of Trichlormethiazide can be increased when it is combined with Biperiden.
Polythiazide The serum concentration of Polythiazide can be increased when it is combined with Biperiden.
Quinethazone The serum concentration of Quinethazone can be increased when it is combined with Biperiden.
Cyclopenthiazide The serum concentration of Cyclopenthiazide can be increased when it is combined with Biperiden.
Epitizide The serum concentration of Epitizide can be increased when it is combined with Biperiden.
Ziprasidone The therapeutic efficacy of Biperiden can be decreased when used in combination with Ziprasidone.
Olanzapine The therapeutic efficacy of Biperiden can be decreased when used in combination with Olanzapine.
Clozapine The serum concentration of Clozapine can be increased when it is combined with Biperiden.

Target Protein

Muscarinic acetylcholine receptor M1 CHRM1

Referensi & Sumber

Synthesis reference: Peter Klein, "Method for the production of biperiden II." U.S. Patent US20040152899, issued August 05, 2004.
Artikel (PubMed)
  • PMID: 8420174
    Nishiyama K, Mizuno T, Sakuta M, Kurisaki H: Chronic dementia in Parkinson's disease treated by anticholinergic agents. Neuropsychological and neuroradiological examination. Adv Neurol. 1993;60:479-83.

Contoh Produk & Brand

Produk: 3 • International brands: 2
Produk
  • Akineton
    Tablet • 2 mg/1 • Oral • US • Approved
  • Akineton
    Tablet • 2 mg/1 • Oral • US • Approved
  • Akineton Tab 2mg
    Tablet • 2 mg • Oral • Canada • Approved
International Brands
  • Bilino — Winston
  • Ipsatol — Orion

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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