Peringatan Keamanan

LD50=808mg/kg (orally in mice)

Tetracycline

DB00759

small molecule approved vet_approved withdrawn

Deskripsi

Tetracycline is a broad spectrum polyketide antibiotic produced by the Streptomyces genus of Actinobacteria. It exerts a bacteriostatic effect on bacteria by binding reversible to the bacterial 30S ribosomal subunit and blocking incoming aminoacyl tRNA from binding to the ribosome acceptor site. It also binds to some extent to the bacterial 50S ribosomal subunit and may alter the cytoplasmic membrane causing intracellular components to leak from bacterial cells.

The FDA withdrew its approval for the use of all liquid oral drug products formulated for pediatric use containing tetracycline in a concentration greater than 25 mg/ml.L43942 Other formulations of tetracycline continue to be used.

Struktur Molekul 2D

Berat 444.4346
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 6-12 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Bioavailability is less than 40% when administered via intramuscular injection, 100% intravenously, and 60-80% orally (fasting adults). Food and/or milk reduce GI absorption of oral preparations of tetracycline by 50% or more.

Metabolisme

Not metabolized

Rute Eliminasi

They are concentrated by the liver in the bile and excreted in the urine and feces at high concentrations in a biologically active form.

Interaksi Makanan

3 Data
  • 1. Avoid milk and dairy products.
  • 2. Take on an empty stomach. Take at least 1 hour before or 2 hours after meals.
  • 3. Take with a full glass of water.

Interaksi Obat

1267 Data
Eliglustat The metabolism of Eliglustat can be decreased when combined with Tetracycline.
Ibrutinib The metabolism of Ibrutinib can be decreased when combined with Tetracycline.
Succinylcholine The therapeutic efficacy of Succinylcholine can be increased when used in combination with Tetracycline.
Metocurine iodide The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Tetracycline.
Gallamine triethiodide The therapeutic efficacy of Gallamine triethiodide can be increased when used in combination with Tetracycline.
Cisatracurium Tetracycline may increase the neuromuscular blocking activities of Cisatracurium.
Rocuronium The therapeutic efficacy of Rocuronium can be increased when used in combination with Tetracycline.
Atracurium besylate The therapeutic efficacy of Atracurium besylate can be increased when used in combination with Tetracycline.
Doxacurium The therapeutic efficacy of Doxacurium can be increased when used in combination with Tetracycline.
Mivacurium The therapeutic efficacy of Mivacurium can be increased when used in combination with Tetracycline.
Decamethonium The therapeutic efficacy of Decamethonium can be increased when used in combination with Tetracycline.
Metocurine The therapeutic efficacy of Metocurine can be increased when used in combination with Tetracycline.
Pancuronium The therapeutic efficacy of Pancuronium can be increased when used in combination with Tetracycline.
Pipecuronium The therapeutic efficacy of Pipecuronium can be increased when used in combination with Tetracycline.
Vecuronium The therapeutic efficacy of Vecuronium can be increased when used in combination with Tetracycline.
Rapacuronium The therapeutic efficacy of Rapacuronium can be increased when used in combination with Tetracycline.
Pyrantel The therapeutic efficacy of Pyrantel can be increased when used in combination with Tetracycline.
Neosaxitoxin The therapeutic efficacy of Neosaxitoxin can be increased when used in combination with Tetracycline.
Atracurium The therapeutic efficacy of Atracurium can be increased when used in combination with Tetracycline.
Gallamine The therapeutic efficacy of Gallamine can be increased when used in combination with Tetracycline.
Alcuronium The therapeutic efficacy of Alcuronium can be increased when used in combination with Tetracycline.
Tubocurarine The therapeutic efficacy of Tubocurarine can be increased when used in combination with Tetracycline.
Cilostazol The metabolism of Cilostazol can be decreased when combined with Tetracycline.
Colchicine The metabolism of Colchicine can be decreased when combined with Tetracycline.
Fentanyl Tetracycline may decrease the excretion rate of Fentanyl which could result in a higher serum level.
Iloperidone The metabolism of Iloperidone can be decreased when combined with Tetracycline.
Retapamulin The metabolism of Retapamulin can be decreased when combined with Tetracycline.
Tofacitinib The metabolism of Tofacitinib can be decreased when combined with Tetracycline.
Vardenafil The metabolism of Vardenafil can be decreased when combined with Tetracycline.
Eszopiclone The metabolism of Eszopiclone can be decreased when combined with Tetracycline.
Zopiclone The metabolism of Zopiclone can be decreased when combined with Tetracycline.
Lovastatin The metabolism of Lovastatin can be decreased when combined with Tetracycline.
Bismuth subsalicylate The serum concentration of Tetracycline can be decreased when it is combined with Bismuth subsalicylate.
Mecamylamine Tetracycline may increase the neuromuscular blocking activities of Mecamylamine.
Mipomersen Tetracycline may increase the hepatotoxic activities of Mipomersen.
Quinapril Quinapril can cause a decrease in the absorption of Tetracycline resulting in a reduced serum concentration and potentially a decrease in efficacy.
Sucralfate Sucralfate can cause a decrease in the absorption of Tetracycline resulting in a reduced serum concentration and potentially a decrease in efficacy.
Iron sucrose The serum concentration of Tetracycline can be decreased when it is combined with Iron sucrose.
Alfuzosin The metabolism of Alfuzosin can be decreased when combined with Tetracycline.
Flucloxacillin The therapeutic efficacy of Flucloxacillin can be decreased when used in combination with Tetracycline.
Piperacillin The therapeutic efficacy of Piperacillin can be decreased when used in combination with Tetracycline.
Ampicillin The therapeutic efficacy of Ampicillin can be decreased when used in combination with Tetracycline.
Phenoxymethylpenicillin The therapeutic efficacy of Phenoxymethylpenicillin can be decreased when used in combination with Tetracycline.
Dicloxacillin The therapeutic efficacy of Dicloxacillin can be decreased when used in combination with Tetracycline.
Carbenicillin The therapeutic efficacy of Carbenicillin can be decreased when used in combination with Tetracycline.
Nafcillin The therapeutic efficacy of Nafcillin can be decreased when used in combination with Tetracycline.
Oxacillin The therapeutic efficacy of Oxacillin can be decreased when used in combination with Tetracycline.
Hetacillin The therapeutic efficacy of Hetacillin can be decreased when used in combination with Tetracycline.
Benzylpenicilloyl polylysine The therapeutic efficacy of Benzylpenicilloyl polylysine can be decreased when used in combination with Tetracycline.
Mezlocillin The therapeutic efficacy of Mezlocillin can be decreased when used in combination with Tetracycline.
Cyclacillin The therapeutic efficacy of Cyclacillin can be decreased when used in combination with Tetracycline.
Benzylpenicillin The therapeutic efficacy of Benzylpenicillin can be decreased when used in combination with Tetracycline.
Amoxicillin The therapeutic efficacy of Amoxicillin can be decreased when used in combination with Tetracycline.
Azlocillin The therapeutic efficacy of Azlocillin can be decreased when used in combination with Tetracycline.
Cloxacillin The therapeutic efficacy of Cloxacillin can be decreased when used in combination with Tetracycline.
Amdinocillin The therapeutic efficacy of Amdinocillin can be decreased when used in combination with Tetracycline.
Bacampicillin The therapeutic efficacy of Bacampicillin can be decreased when used in combination with Tetracycline.
Meticillin The therapeutic efficacy of Meticillin can be decreased when used in combination with Tetracycline.
Pivampicillin The therapeutic efficacy of Pivampicillin can be decreased when used in combination with Tetracycline.
Pivmecillinam The therapeutic efficacy of Pivmecillinam can be decreased when used in combination with Tetracycline.
Ticarcillin The therapeutic efficacy of Ticarcillin can be decreased when used in combination with Tetracycline.
Azidocillin The therapeutic efficacy of Azidocillin can be decreased when used in combination with Tetracycline.
Carindacillin The therapeutic efficacy of Carindacillin can be decreased when used in combination with Tetracycline.
Procaine benzylpenicillin The therapeutic efficacy of Procaine benzylpenicillin can be decreased when used in combination with Tetracycline.
Sultamicillin The therapeutic efficacy of Sultamicillin can be decreased when used in combination with Tetracycline.
Temocillin The therapeutic efficacy of Temocillin can be decreased when used in combination with Tetracycline.
Epicillin The therapeutic efficacy of Epicillin can be decreased when used in combination with Tetracycline.
Pheneticillin The therapeutic efficacy of Pheneticillin can be decreased when used in combination with Tetracycline.
Carfecillin The therapeutic efficacy of Carfecillin can be decreased when used in combination with Tetracycline.
Propicillin The therapeutic efficacy of Propicillin can be decreased when used in combination with Tetracycline.
Clometocillin The therapeutic efficacy of Clometocillin can be decreased when used in combination with Tetracycline.
Sulbenicillin The therapeutic efficacy of Sulbenicillin can be decreased when used in combination with Tetracycline.
Penamecillin The therapeutic efficacy of Penamecillin can be decreased when used in combination with Tetracycline.
Talampicillin The therapeutic efficacy of Talampicillin can be decreased when used in combination with Tetracycline.
Aspoxicillin The therapeutic efficacy of Aspoxicillin can be decreased when used in combination with Tetracycline.
Metampicillin The therapeutic efficacy of Metampicillin can be decreased when used in combination with Tetracycline.
Alprazolam The metabolism of Alprazolam can be decreased when combined with Tetracycline.
Quinine The serum concentration of Quinine can be increased when it is combined with Tetracycline.
Quinidine The serum concentration of Quinidine can be increased when it is combined with Tetracycline.
Aspartame The excretion of Tetracycline can be decreased when combined with Aspartame.
Aminohippuric acid The excretion of Tetracycline can be decreased when combined with Aminohippuric acid.
Guanidine The excretion of Tetracycline can be decreased when combined with Guanidine.
Oxytetracycline The excretion of Tetracycline can be decreased when combined with Oxytetracycline.
Leucovorin The excretion of Tetracycline can be decreased when combined with Leucovorin.
Succinic acid The excretion of Succinic acid can be decreased when combined with Tetracycline.
Citrulline The excretion of Citrulline can be decreased when combined with Tetracycline.
Cefdinir The excretion of Cefdinir can be decreased when combined with Tetracycline.
Fluorescein The excretion of Fluorescein can be decreased when combined with Tetracycline.
Dinoprostone The excretion of Dinoprostone can be decreased when combined with Tetracycline.
Famotidine The excretion of Famotidine can be decreased when combined with Tetracycline.
Rosuvastatin The excretion of Rosuvastatin can be decreased when combined with Tetracycline.
Tazobactam The excretion of Tazobactam can be decreased when combined with Tetracycline.
Cyclic adenosine monophosphate The excretion of Cyclic adenosine monophosphate can be decreased when combined with Tetracycline.
Cholic Acid The excretion of Cholic Acid can be decreased when combined with Tetracycline.
Glutaric Acid The excretion of Glutaric Acid can be decreased when combined with Tetracycline.
Oxalic Acid The excretion of Oxalic Acid can be decreased when combined with Tetracycline.
Saxagliptin The excretion of Saxagliptin can be decreased when combined with Tetracycline.
Ellagic acid The excretion of Ellagic acid can be decreased when combined with Tetracycline.
Avibactam The excretion of Avibactam can be decreased when combined with Tetracycline.
Eluxadoline The excretion of Eluxadoline can be decreased when combined with Tetracycline.

Target Protein

30S ribosomal protein S7 rpsG
30S ribosomal protein S14 rpsN
30S ribosomal protein S3 rpsC
30S ribosomal protein S8 rpsH
30S ribosomal protein S19 rpsS
16S ribosomal RNA
Major prion protein PRNP
Multidrug translocase MdfA mdfA
Protein-arginine deiminase type-4 PADI4

Referensi & Sumber

Synthesis reference: Thomas F. McNamara, Nungavaram S. Ramamurthy, Lorne M. Golub, "Non-antibacterial tetracycline compositions possessing anti-collagenolytic properties and methods of preparing and using same." U.S. Patent US4704383, issued May, 1963.
Artikel (PubMed)
  • PMID: 20592239
    Griffin MO, Fricovsky E, Ceballos G, Villarreal F: Tetracyclines: a pleitropic family of compounds with promising therapeutic properties. Review of the literature. Am J Physiol Cell Physiol. 2010 Sep;299(3):C539-48. doi: 10.1152/ajpcell.00047.2010. Epub 2010 Jun 30.

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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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