Peringatan Keamanan

In overdosage, some patients exhibit insomnia, restlessness and anxiety, progressing in severe cases to agitation, mental confusion and incoherence. Hypotension, dizziness, weakness and drowsiness may occur, progressing in severe cases to extreme dizziness and shock. A few patients have displayed hypertension with severe headache and other symptoms. Rare instances have been reported in which hypertension was accompanied by twitching or myoclonic fibrillation of skeletal muscles with hyperpyrexia, sometimes progressing to generalized rigidity and coma.

Tranylcypromine

DB00752

small molecule approved investigational

Deskripsi

A propylamine formed from the cyclization of the side chain of amphetamine. This monoamine oxidase inhibitor is effective in the treatment of major depression, dysthymic disorder, and atypical depression. It also is useful in panic and phobic disorders (From AMA Drug Evaluations Annual, 1994, p311).

Tranylcypromine is a racemate comprising equal amounts of (1R,2S)- and (1S,2R)-2-phenylcyclopropan-1-amine with the chiral centers both located on the cylopropane ring. An irreversible monoamine oxidase inhibitor that is used as an antidepressant (INN tranylcypromine).

Struktur Molekul 2D

Berat 133.194
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 1.5-3.2 hours in patients with normal renal and hepatic function
Volume Distribusi 1.1-5.7 L/kg
Klirens (Clearance) -

Absorpsi

Interindividual variability in absorption. May be biphasic in some individuals. Peak plasma concentrations occur in one hour following oral administration with a secondary peak occurring within 2-3 hours. Biphasic absorption may represent different rates of absorption of the stereoisomers of the drug, though additional studies are required to confirm this.

Metabolisme

Hepatic.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

3 Data
  • 1. Avoid alcohol. Ingesting alcohol may increase the CNS depressant effects of tranylcypromine.
  • 2. Avoid St. John's Wort. Administering tranylcypromine with St. John's Wort may increase the risk of serotonin syndrome.
  • 3. Avoid tyramine-containing foods and supplements. Tyramine-containing foods and beverages can cause a sudden elevation in blood pressure or a hypertensive crisis. Foods that contain tyramine include aged cheese, ripe bananas, red wine, some alcoholic beverages (beer), cured food, pickled food, and fava beans.

Interaksi Obat

1514 Data
Risperidone Tranylcypromine may increase the hypotensive activities of Risperidone.
Cilostazol The serum concentration of Cilostazol can be increased when it is combined with Tranylcypromine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Tranylcypromine.
Dronabinol The serum concentration of Dronabinol can be increased when it is combined with Tranylcypromine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Tranylcypromine.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Tranylcypromine.
Magnesium sulfate The therapeutic efficacy of Tranylcypromine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Tranylcypromine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Tranylcypromine may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Tranylcypromine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Tranylcypromine.
Orphenadrine Tranylcypromine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Tranylcypromine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Tranylcypromine.
Pramipexole Tranylcypromine may increase the sedative activities of Pramipexole.
Rotigotine Tranylcypromine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Tranylcypromine.
Sodium oxybate Tranylcypromine may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Tranylcypromine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Thalidomide Tranylcypromine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Tranylcypromine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Yohimbine The therapeutic efficacy of Tranylcypromine can be increased when used in combination with Yohimbine.
Eliglustat The metabolism of Eliglustat can be decreased when combined with Tranylcypromine.
Ibrutinib The metabolism of Ibrutinib can be decreased when combined with Tranylcypromine.
Brexpiprazole The metabolism of Brexpiprazole can be decreased when combined with Tranylcypromine.
Desmopressin The risk or severity of hypertension can be increased when Desmopressin is combined with Tranylcypromine.
Icosapent The risk or severity of hypertension can be increased when Icosapent is combined with Tranylcypromine.
Mesalazine The risk or severity of hypertension can be increased when Mesalazine is combined with Tranylcypromine.
Tolmetin The risk or severity of hypertension can be increased when Tolmetin is combined with Tranylcypromine.
Fenoprofen The risk or severity of hypertension can be increased when Fenoprofen is combined with Tranylcypromine.
Sulindac The risk or severity of hypertension can be increased when Sulindac is combined with Tranylcypromine.
Sulfasalazine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Sulfasalazine.
Carprofen The risk or severity of hypertension can be increased when Tranylcypromine is combined with Carprofen.
Phenmetrazine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Phenmetrazine.
Diflunisal The risk or severity of hypertension can be increased when Tranylcypromine is combined with Diflunisal.
Meclofenamic acid The risk or severity of hypertension can be increased when Tranylcypromine is combined with Meclofenamic acid.
Oxaprozin The risk or severity of hypertension can be increased when Tranylcypromine is combined with Oxaprozin.
Balsalazide The risk or severity of hypertension can be increased when Tranylcypromine is combined with Balsalazide.
Ephedrine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Ephedrine.
Magnesium salicylate The risk or severity of hypertension can be increased when Tranylcypromine is combined with Magnesium salicylate.
Salsalate The risk or severity of hypertension can be increased when Tranylcypromine is combined with Salsalate.
Choline magnesium trisalicylate The risk or severity of hypertension can be increased when Tranylcypromine is combined with Choline magnesium trisalicylate.
Antrafenine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Antrafenine.
Tiaprofenic acid The risk or severity of hypertension can be increased when Tranylcypromine is combined with Tiaprofenic acid.
Epicaptopril The risk or severity of hypertension can be increased when Tranylcypromine is combined with Epicaptopril.
Taxifolin The risk or severity of hypertension can be increased when Tranylcypromine is combined with Taxifolin.
Oxyphenbutazone The risk or severity of hypertension can be increased when Tranylcypromine is combined with Oxyphenbutazone.
1-benzylimidazole The risk or severity of hypertension can be increased when Tranylcypromine is combined with 1-benzylimidazole.
Benoxaprofen The risk or severity of hypertension can be increased when Tranylcypromine is combined with Benoxaprofen.
Metamizole The risk or severity of hypertension can be increased when Tranylcypromine is combined with Metamizole.
Cimicoxib The risk or severity of hypertension can be increased when Tranylcypromine is combined with Cimicoxib.
Amibegron The risk or severity of hypertension can be increased when Tranylcypromine is combined with Amibegron.
Solabegron The risk or severity of hypertension can be increased when Tranylcypromine is combined with Solabegron.
Saralasin The risk or severity of hypertension can be increased when Tranylcypromine is combined with Saralasin.
Azapropazone The risk or severity of hypertension can be increased when Tranylcypromine is combined with Azapropazone.
Salicylamide The risk or severity of hypertension can be increased when Tranylcypromine is combined with Salicylamide.
Tyramine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Tyramine.
Adrafinil The risk or severity of hypertension can be increased when Tranylcypromine is combined with Adrafinil.
Kebuzone The risk or severity of hypertension can be increased when Tranylcypromine is combined with Kebuzone.
Isoxicam The risk or severity of hypertension can be increased when Tranylcypromine is combined with Isoxicam.
Indoprofen The risk or severity of hypertension can be increased when Tranylcypromine is combined with Indoprofen.
Ibuproxam The risk or severity of hypertension can be increased when Tranylcypromine is combined with Ibuproxam.
Floctafenine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Floctafenine.
Fenbufen The risk or severity of hypertension can be increased when Tranylcypromine is combined with Fenbufen.
Etofenamate The risk or severity of hypertension can be increased when Tranylcypromine is combined with Etofenamate.
Etilefrine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Etilefrine.
Epirizole The risk or severity of hypertension can be increased when Tranylcypromine is combined with Epirizole.
Benzydamine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Benzydamine.
Synephrine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Synephrine.
Moxisylyte The risk or severity of hypertension can be increased when Tranylcypromine is combined with Moxisylyte.
Dexketoprofen The risk or severity of hypertension can be increased when Tranylcypromine is combined with Dexketoprofen.
Droxicam The risk or severity of hypertension can be increased when Tranylcypromine is combined with Droxicam.
Firocoxib The risk or severity of hypertension can be increased when Tranylcypromine is combined with Firocoxib.
Clonixin The risk or severity of hypertension can be increased when Tranylcypromine is combined with Clonixin.
Morniflumate The risk or severity of hypertension can be increased when Tranylcypromine is combined with Morniflumate.
Talniflumate The risk or severity of hypertension can be increased when Tranylcypromine is combined with Talniflumate.
DL-Methylephedrine The risk or severity of hypertension can be increased when Tranylcypromine is combined with DL-Methylephedrine.
Amitraz The risk or severity of hypertension can be increased when Tranylcypromine is combined with Amitraz.
Robenacoxib The risk or severity of hypertension can be increased when Tranylcypromine is combined with Robenacoxib.
Tepoxalin The risk or severity of hypertension can be increased when Tranylcypromine is combined with Tepoxalin.
Atipamezole The risk or severity of hypertension can be increased when Tranylcypromine is combined with Atipamezole.
Flunixin The risk or severity of hypertension can be increased when Tranylcypromine is combined with Flunixin.
Ractopamine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Ractopamine.
Tulobuterol The risk or severity of hypertension can be increased when Tranylcypromine is combined with Tulobuterol.
Dopexamine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Dopexamine.
Idazoxan The risk or severity of hypertension can be increased when Tranylcypromine is combined with Idazoxan.
Ebselen The risk or severity of hypertension can be increased when Tranylcypromine is combined with Ebselen.
Higenamine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Higenamine.
Reproterol The risk or severity of hypertension can be increased when Tranylcypromine is combined with Reproterol.
Tinoridine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Tinoridine.
Tramazoline The risk or severity of hypertension can be increased when Tranylcypromine is combined with Tramazoline.
Alclofenac The risk or severity of hypertension can be increased when Tranylcypromine is combined with Alclofenac.
Fentiazac The risk or severity of hypertension can be increased when Tranylcypromine is combined with Fentiazac.
Suxibuzone The risk or severity of hypertension can be increased when Tranylcypromine is combined with Suxibuzone.
Octopamine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Octopamine.
Bumadizone The risk or severity of hypertension can be increased when Tranylcypromine is combined with Bumadizone.
Alminoprofen The risk or severity of hypertension can be increased when Tranylcypromine is combined with Alminoprofen.
Fenozolone The risk or severity of hypertension can be increased when Tranylcypromine is combined with Fenozolone.
Difenpiramide The risk or severity of hypertension can be increased when Tranylcypromine is combined with Difenpiramide.
Norfenefrine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Norfenefrine.

Target Protein

Amine oxidase [flavin-containing] B MAOB
Amine oxidase [flavin-containing] A MAOA

Referensi & Sumber

Artikel (PubMed)

Contoh Produk & Brand

Produk: 19 • International brands: 1
Produk
  • M-tranylcypromine
    Tablet • 10 mg • Oral • Canada • Approved
  • Parnate
    Tablet, film coated • 10 mg/1 • Oral • US • Approved
  • Parnate
    Tablet, film coated • 10 mg/1 • Oral • US • Approved
  • Parnate
    Tablet, film coated • 10 mg/1 • Oral • US • Approved
  • Parnate
    Tablet, film coated • 10 mg/1 • Oral • US • Approved
  • Parnate
    Tablet, film coated • 10 mg/1 • Oral • US • Approved
  • Parnate
    Tablet • 10 mg • Oral • Canada • Approved
  • Tranylcypromine
    Tablet • 10 mg/1 • Oral • US • Generic • Approved
Menampilkan 8 dari 19 produk.
International Brands
  • Jatrosom — Aristo Pharma

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