Carbinoxamine

DB00748

small molecule approved

Deskripsi

Carbinoxamine is a first generation antihistamine that competes with free histamine for binding at HA-receptor sites. This antagonizes the effects of histamine on HA-receptors, leading to a reduction of the negative symptoms brought on by histamine HA-receptor binding. The product label for carbinoxamine as an over the counter cough and cold medicine is being modified to state "do not use" in children under 4 years of age in order to prevent and reduce misuse, as many unapproved carbinoxamine-containing preparations contained inappropriate labeling, which promoted unapproved uses (including management of congestion, cough, the common cold, and the use in children under 2 years of age), which can potentially cause serious health risks.

Struktur Molekul 2D

Berat 290.788
Wujud liquid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 10 to 20 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol. Ingesting alcohol may increase drowsiness caused by carbinoxamine.
  • 2. Take on an empty stomach.

Interaksi Obat

959 Data
Ivabradine Ivabradine may increase the QTc-prolonging activities of Carbinoxamine.
Buprenorphine Carbinoxamine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Carbinoxamine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Carbinoxamine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Carbinoxamine.
Hydrocodone Carbinoxamine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Magnesium sulfate The therapeutic efficacy of Carbinoxamine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Carbinoxamine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Carbinoxamine may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Carbinoxamine.
Mirtazapine Carbinoxamine may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Carbinoxamine.
Orphenadrine Carbinoxamine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Carbinoxamine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Carbinoxamine.
Pramipexole Carbinoxamine may increase the sedative activities of Pramipexole.
Ropinirole Carbinoxamine may increase the sedative activities of Ropinirole.
Rotigotine Carbinoxamine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Carbinoxamine.
Sodium oxybate Carbinoxamine may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Carbinoxamine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Carbinoxamine.
Thalidomide Carbinoxamine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Carbinoxamine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Benzylpenicilloyl polylysine Carbinoxamine may decrease effectiveness of Benzylpenicilloyl polylysine as a diagnostic agent.
Betahistine The therapeutic efficacy of Betahistine can be decreased when used in combination with Carbinoxamine.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Carbinoxamine.
Ethanol Carbinoxamine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Carbinoxamine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Carbinoxamine.
Fluvoxamine The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Fluvoxamine.
Duloxetine The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Duloxetine.
Paroxetine The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Sibutramine.
Zimelidine The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Seproxetine.
Indalpine The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Alaproclate.
Nefazodone The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Nefazodone.
Amphetamine Amphetamine may decrease the sedative activities of Carbinoxamine.
Phentermine Phentermine may decrease the sedative activities of Carbinoxamine.
Benzphetamine Benzphetamine may decrease the sedative activities of Carbinoxamine.
Diethylpropion Diethylpropion may decrease the sedative activities of Carbinoxamine.
Lisdexamfetamine Lisdexamfetamine may decrease the sedative activities of Carbinoxamine.
Mephentermine Mephentermine may decrease the sedative activities of Carbinoxamine.
MMDA MMDA may decrease the sedative activities of Carbinoxamine.
Midomafetamine Midomafetamine may decrease the sedative activities of Carbinoxamine.
2,5-Dimethoxy-4-ethylamphetamine 2,5-Dimethoxy-4-ethylamphetamine may decrease the sedative activities of Carbinoxamine.
4-Bromo-2,5-dimethoxyamphetamine 4-Bromo-2,5-dimethoxyamphetamine may decrease the sedative activities of Carbinoxamine.
Tenamfetamine Tenamfetamine may decrease the sedative activities of Carbinoxamine.
Chlorphentermine Chlorphentermine may decrease the sedative activities of Carbinoxamine.
Methylenedioxyethamphetamine Methylenedioxyethamphetamine may decrease the sedative activities of Carbinoxamine.
Dextroamphetamine Dextroamphetamine may decrease the sedative activities of Carbinoxamine.
Metamfetamine Metamfetamine may decrease the sedative activities of Carbinoxamine.
Iofetamine I-123 Iofetamine I-123 may decrease the sedative activities of Carbinoxamine.
Ritobegron Ritobegron may decrease the sedative activities of Carbinoxamine.
Mephedrone Mephedrone may decrease the sedative activities of Carbinoxamine.
Methoxyphenamine Methoxyphenamine may decrease the sedative activities of Carbinoxamine.
Gepefrine Gepefrine may decrease the sedative activities of Carbinoxamine.
2,5-Dimethoxy-4-ethylthioamphetamine 2,5-Dimethoxy-4-ethylthioamphetamine may decrease the sedative activities of Carbinoxamine.
Phendimetrazine Phendimetrazine may decrease the sedative activities of Carbinoxamine.
Cyproheptadine The risk or severity of CNS depression can be increased when Cyproheptadine is combined with Carbinoxamine.
Amoxapine The risk or severity of CNS depression can be increased when Amoxapine is combined with Carbinoxamine.
Propiomazine The risk or severity of CNS depression can be increased when Carbinoxamine is combined with Propiomazine.
Maprotiline The risk or severity of CNS depression can be increased when Carbinoxamine is combined with Maprotiline.
Desipramine The risk or severity of CNS depression can be increased when Carbinoxamine is combined with Desipramine.
Pizotifen The risk or severity of CNS depression can be increased when Carbinoxamine is combined with Pizotifen.
Dosulepin The risk or severity of CNS depression can be increased when Carbinoxamine is combined with Dosulepin.
Amitriptyline The risk or severity of QTc prolongation can be increased when Amitriptyline is combined with Carbinoxamine.
Imipramine The risk or severity of QTc prolongation can be increased when Imipramine is combined with Carbinoxamine.
Zopiclone The risk or severity of adverse effects can be increased when Carbinoxamine is combined with Zopiclone.
Citalopram The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Citalopram.
Anagrelide The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Anagrelide.
Disopyramide The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Disopyramide.
Clemastine The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Clemastine.
Ibutilide The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Ibutilide.
Valproic acid The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Valproic acid.
Grepafloxacin The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Grepafloxacin.
Quinine The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Quinine.
Sotalol The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Sotalol.
Toremifene The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Toremifene.
Imatinib The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Imatinib.
Thioridazine The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Thioridazine.
Trovafloxacin The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Trovafloxacin.
Cocaine The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Cocaine.
Procainamide The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Procainamide.
Arsenic trioxide The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Arsenic trioxide.
Escitalopram The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Escitalopram.
Domperidone The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Domperidone.
Sparfloxacin The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Sparfloxacin.
Halofantrine The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Halofantrine.
Bepridil The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Bepridil.
Paliperidone The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Paliperidone.
Lithium cation The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Lithium cation.
Temafloxacin The risk or severity of QTc prolongation can be increased when Carbinoxamine is combined with Temafloxacin.

Target Protein

Histamine H1 receptor HRH1

Referensi & Sumber

Synthesis reference: Tilford. C.H. and Shelton, R.S.; U.S. Patent 2,606,195;August 5,1952; assigned to The Wm.S. Merrell Company. Swain, A.P.; U.S. Patent 2800,485; July 23,1957; assigned to McNeil Laboratories, Inc.
Artikel (PubMed)
  • PMID: 13211145
    BEALE HD, RAWLING FF, FIGLEY KD: Clistin maleate; a clinical appraisal of a new antihistaminic. J Allergy. 1954 Nov;25(6):521-4.

Contoh Produk & Brand

Produk: 28 • International brands: 6
Produk
  • Arbinoxa
    Solution • 0.8 mg/1mL • Oral • US • Generic • Approved
  • Arbinoxa
    Tablet • 4 mg/1 • Oral • US • Generic • Approved
  • Carbinoxamine Maleate
    Tablet • 4 mg/1 • Oral • US • Generic • Approved
  • Carbinoxamine Maleate
    Solution • 4 mg/5mL • Oral • US • Generic • Approved
  • Carbinoxamine Maleate
    Tablet • 4 mg/1 • Oral • US • Generic • Approved
  • Carbinoxamine Maleate
    Syrup • 4 mg/5mL • Oral • US • Generic • Approved
  • Carbinoxamine Maleate
    Tablet • 4 mg/1 • Oral • US • Generic • Approved
  • Carbinoxamine Maleate
    Tablet • 4 mg/1 • Oral • US • Generic • Approved
Menampilkan 8 dari 28 produk.
International Brands
  • Allergefon — SERP
  • Clistin
  • Histin — Kenyaku
  • Karbinal
  • Rotoxamine
  • Satinmin — Shou Chan

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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