Peringatan Keamanan

Overdosage may be associated with transient disturbances of vision and psychic alterations. The oral LD 50 is 3.6 g/kg, 3.1 g/kg and 3.8 g/kg in the mouse, rat, and rabbit respectively.

Thiabendazole

DB00730

small molecule approved vet_approved

Deskripsi

2-Substituted benzimidazole first introduced in 1962. It is active against a variety of nematodes and is the drug of choice for strongyloidiasis. It has CNS side effects and hepatototoxic potential. (From Smith and Reynard, Textbook of Pharmacology, 1992, p919)

Struktur Molekul 2D

Berat 201.248
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The half-life for thiabendazole in both normal and anephric patients is 1.2 hours (range 0.9 to 2 hours). The half-life for the 5-hydroxythiabendazole metabolite in both normal and anephric patients is 1.7 hours (range 1.4 to 2 hours).
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Rapidly absorbed and peak plasma concentration is reached within 1 to 2 hours after the oral administration of a suspension. Some systemic absorption may occur from topical preparations applied to the skin.

Metabolisme

Hepatic. Metabolized almost completely to the 5-hydroxy form which appears in the urine as glucuronide or sulfate conjugates.

Rute Eliminasi

It is metabolized almost completely to the 5-hydroxy form which appears in the urine as glucuronide or sulfate conjugates.

Interaksi Obat

972 Data
Deferasirox The serum concentration of Thiabendazole can be increased when it is combined with Deferasirox.
Peginterferon alfa-2b The serum concentration of Thiabendazole can be increased when it is combined with Peginterferon alfa-2b.
Leflunomide The serum concentration of Thiabendazole can be decreased when it is combined with Leflunomide.
Teriflunomide The serum concentration of Thiabendazole can be decreased when it is combined with Teriflunomide.
Caffeine The metabolism of Caffeine can be decreased when combined with Thiabendazole.
Theophylline The metabolism of Theophylline can be decreased when combined with Thiabendazole.
Dyphylline The metabolism of Dyphylline can be decreased when combined with Thiabendazole.
Pentoxifylline The metabolism of Pentoxifylline can be decreased when combined with Thiabendazole.
Mercaptopurine The metabolism of Mercaptopurine can be decreased when combined with Thiabendazole.
Aminophylline The metabolism of Aminophylline can be decreased when combined with Thiabendazole.
Oxtriphylline The metabolism of Oxtriphylline can be decreased when combined with Thiabendazole.
Theobromine The metabolism of Theobromine can be decreased when combined with Thiabendazole.
Fenethylline The metabolism of Fenethylline can be decreased when combined with Thiabendazole.
8-azaguanine The metabolism of 8-azaguanine can be decreased when combined with Thiabendazole.
7,9-Dimethylguanine The metabolism of 7,9-Dimethylguanine can be decreased when combined with Thiabendazole.
Xanthine The metabolism of Xanthine can be decreased when combined with Thiabendazole.
7-Deazaguanine The metabolism of 7-Deazaguanine can be decreased when combined with Thiabendazole.
Guanine The metabolism of Guanine can be decreased when combined with Thiabendazole.
9-Methylguanine The metabolism of 9-Methylguanine can be decreased when combined with Thiabendazole.
Peldesine The metabolism of Peldesine can be decreased when combined with Thiabendazole.
Hypoxanthine The metabolism of Hypoxanthine can be decreased when combined with Thiabendazole.
9-Deazaguanine The metabolism of 9-Deazaguanine can be decreased when combined with Thiabendazole.
Propentofylline The metabolism of Propentofylline can be decreased when combined with Thiabendazole.
Valomaciclovir The metabolism of Valomaciclovir can be decreased when combined with Thiabendazole.
3-isobutyl-1-methyl-7H-xanthine The metabolism of 3-isobutyl-1-methyl-7H-xanthine can be decreased when combined with Thiabendazole.
Uric acid The metabolism of Uric acid can be decreased when combined with Thiabendazole.
Doxofylline The metabolism of Doxofylline can be decreased when combined with Thiabendazole.
6-O-benzylguanine The metabolism of 6-O-benzylguanine can be decreased when combined with Thiabendazole.
Lisofylline The metabolism of Lisofylline can be decreased when combined with Thiabendazole.
Lobucavir The metabolism of Lobucavir can be decreased when combined with Thiabendazole.
Cafedrine The metabolism of Cafedrine can be decreased when combined with Thiabendazole.
Theodrenaline The metabolism of Theodrenaline can be decreased when combined with Thiabendazole.
Bamifylline The metabolism of Bamifylline can be decreased when combined with Thiabendazole.
Proxyphylline The metabolism of Proxyphylline can be decreased when combined with Thiabendazole.
Acefylline The metabolism of Acefylline can be decreased when combined with Thiabendazole.
Etamiphylline The metabolism of Etamiphylline can be decreased when combined with Thiabendazole.
Pentifylline The metabolism of Pentifylline can be decreased when combined with Thiabendazole.
Bufylline The metabolism of Bufylline can be decreased when combined with Thiabendazole.
Bromotheophylline The metabolism of Bromotheophylline can be decreased when combined with Thiabendazole.
Furafylline The metabolism of Furafylline can be decreased when combined with Thiabendazole.
8-chlorotheophylline The metabolism of 8-chlorotheophylline can be decreased when combined with Thiabendazole.
PCS-499 The metabolism of PCS-499 can be decreased when combined with Thiabendazole.
Zolmitriptan The metabolism of Zolmitriptan can be decreased when combined with Thiabendazole.
Abiraterone The serum concentration of Thiabendazole can be increased when it is combined with Abiraterone.
Cyproterone acetate The metabolism of Thiabendazole can be increased when combined with Cyproterone acetate.
Primidone The metabolism of Thiabendazole can be increased when combined with Primidone.
Rifampin The metabolism of Thiabendazole can be increased when combined with Rifampicin.
Albendazole The metabolism of Thiabendazole can be increased when combined with Albendazole.
Carbamazepine The metabolism of Thiabendazole can be increased when combined with Carbamazepine.
Moxifloxacin The metabolism of Thiabendazole can be decreased when combined with Moxifloxacin.
Lidocaine The metabolism of Thiabendazole can be decreased when combined with Lidocaine.
Mexiletine The metabolism of Thiabendazole can be decreased when combined with Mexiletine.
Alosetron The metabolism of Thiabendazole can be decreased when combined with Alosetron.
Ketoconazole The metabolism of Thiabendazole can be decreased when combined with Ketoconazole.
Gatifloxacin The metabolism of Thiabendazole can be decreased when combined with Gatifloxacin.
Simeprevir The metabolism of Thiabendazole can be decreased when combined with Simeprevir.
Lobeglitazone The metabolism of Thiabendazole can be decreased when combined with Lobeglitazone.
Pazufloxacin The metabolism of Thiabendazole can be decreased when combined with Pazufloxacin.
Osilodrostat The metabolism of Thiabendazole can be decreased when combined with Osilodrostat.
Osimertinib The serum concentration of Thiabendazole can be decreased when it is combined with Osimertinib.
Vemurafenib The serum concentration of Thiabendazole can be increased when it is combined with Vemurafenib.
Cyclosporine Cyclosporine may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Icosapent Icosapent may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Cefotiam Cefotiam may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Mesalazine Mesalazine may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Cefmenoxime Cefmenoxime may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Cefmetazole Cefmetazole may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Pamidronic acid Pamidronic acid may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Tenofovir disoproxil Tenofovir disoproxil may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Indomethacin Indomethacin may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Cidofovir Cidofovir may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Cefpiramide Cefpiramide may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Ceftazidime Ceftazidime may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Loracarbef Loracarbef may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Cefalotin Cefalotin may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Ketorolac Ketorolac may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Tenoxicam Tenoxicam may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Celecoxib Celecoxib may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Cefotaxime Cefotaxime may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Tolmetin Tolmetin may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Foscarnet Foscarnet may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Piroxicam Piroxicam may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Cephalexin Cephalexin may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Fenoprofen Fenoprofen may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Valaciclovir Valaciclovir may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Valdecoxib Valdecoxib may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Sulindac Sulindac may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Bacitracin Bacitracin may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Amphotericin B Amphotericin B may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Cephaloglycin Cephaloglycin may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Flurbiprofen Flurbiprofen may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Adefovir dipivoxil Adefovir dipivoxil may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Pentamidine Pentamidine may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Etodolac Etodolac may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Sulfasalazine Sulfasalazine may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Phenylbutazone Phenylbutazone may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Meloxicam Meloxicam may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Carprofen Carprofen may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Cefaclor Cefaclor may decrease the excretion rate of Thiabendazole which could result in a higher serum level.
Diflunisal Diflunisal may decrease the excretion rate of Thiabendazole which could result in a higher serum level.

Target Protein

Fumarate reductase flavoprotein subunit frdA

Referensi & Sumber

Synthesis reference: Lynn E. Applegate, Carl A. Renner, "Preparation of high purity thiabendazole." U.S. Patent US5310923, issued October, 1977.

Contoh Produk & Brand

Produk: 3 • International brands: 2
Produk
  • Mintezol
    Tablet, chewable • 500 mg/1 • Oral • US • Approved
  • Mintezol
    Suspension • 500 mg/5mL • Oral • US • Approved
  • Mintezol Chewable Tab 500mg
    Tablet • 500 mg / tab • Oral • Canada • Approved
International Brands
  • Equizole
  • Thibenzole

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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