Peringatan Keamanan

LD50=956-1034 mg/kg (Orally in rats); Agitation, blurred vision, coma, confusion, constipation, difficulty breathing, dilated or constricted pupils, diminished flow of urine, dry mouth, dry skin, excessively high or low body temperature, extremely low blood pressure, fluid in the lungs, heart abnormalities, inability to urinate, intestinal blockage, nasal congestion, restlessness, sedation, seizures, shock

Thioridazine

DB00679

small molecule approved withdrawn

Deskripsi

A phenothiazine antipsychotic used in the management of psychoses, including schizophrenia, and in the control of severely disturbed or agitated behavior. It has little antiemetic activity. Thioridazine has a higher incidence of antimuscarinic effects, but a lower incidence of extrapyramidal symptoms, than chlorpromazine. (From Martindale, The Extra Pharmacopoeia, 30th ed, p618).

Thioridazine was withdrawn worldwide in 2005 due to its association with cardiac arrythmias.

Struktur Molekul 2D

Berat 370.575
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 21-25 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

60%

Metabolisme

Hepatic

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

1 Data
  • 1. Avoid alcohol. Ingesting alcohol may potentiate the CNS depressant actions of thioridazine.

Interaksi Obat

1656 Data
Duloxetine The risk or severity of orthostatic hypotension and syncope can be increased when Thioridazine is combined with Duloxetine.
Levodopa The risk or severity of hypotension and orthostatic hypotension can be increased when Thioridazine is combined with Levodopa.
Risperidone Thioridazine may increase the hypotensive activities of Risperidone.
Fluvoxamine The serum concentration of Thioridazine can be increased when it is combined with Fluvoxamine.
Furosemide Thioridazine may decrease the antihypertensive activities of Furosemide.
Valsartan Thioridazine may decrease the antihypertensive activities of Valsartan.
Ramipril Thioridazine may decrease the antihypertensive activities of Ramipril.
Remikiren Thioridazine may decrease the antihypertensive activities of Remikiren.
Guanadrel Thioridazine may decrease the antihypertensive activities of Guanadrel.
Olmesartan Thioridazine may decrease the antihypertensive activities of Olmesartan.
Chlorthalidone Thioridazine may decrease the antihypertensive activities of Chlorthalidone.
Nitroprusside Thioridazine may decrease the antihypertensive activities of Nitroprusside.
Minoxidil Thioridazine may decrease the antihypertensive activities of Minoxidil.
Bendroflumethiazide Thioridazine may decrease the antihypertensive activities of Bendroflumethiazide.
Fosinopril Thioridazine may decrease the antihypertensive activities of Fosinopril.
Trandolapril Thioridazine may decrease the antihypertensive activities of Trandolapril.
Metolazone Thioridazine may decrease the antihypertensive activities of Metolazone.
Benazepril Thioridazine may decrease the antihypertensive activities of Benazepril.
Bosentan Thioridazine may decrease the antihypertensive activities of Bosentan.
Enalapril Thioridazine may decrease the antihypertensive activities of Enalapril.
Cyclothiazide Thioridazine may decrease the antihypertensive activities of Cyclothiazide.
Candoxatril Thioridazine may decrease the antihypertensive activities of Candoxatril.
Mecamylamine Thioridazine may decrease the antihypertensive activities of Mecamylamine.
Eplerenone Thioridazine may decrease the antihypertensive activities of Eplerenone.
Lisinopril Thioridazine may decrease the antihypertensive activities of Lisinopril.
Nitroglycerin Thioridazine may decrease the antihypertensive activities of Nitroglycerin.
Hydroflumethiazide Thioridazine may decrease the antihypertensive activities of Hydroflumethiazide.
Cryptenamine Thioridazine may decrease the antihypertensive activities of Cryptenamine.
Perindopril Thioridazine may decrease the antihypertensive activities of Perindopril.
Candesartan cilexetil Thioridazine may decrease the antihypertensive activities of Candesartan cilexetil.
Eprosartan Thioridazine may decrease the antihypertensive activities of Eprosartan.
Chlorothiazide Thioridazine may decrease the antihypertensive activities of Chlorothiazide.
Quinapril Thioridazine may decrease the antihypertensive activities of Quinapril.
Omapatrilat Thioridazine may decrease the antihypertensive activities of Omapatrilat.
Trichlormethiazide Thioridazine may decrease the antihypertensive activities of Trichlormethiazide.
Deserpidine Thioridazine may decrease the antihypertensive activities of Deserpidine.
Pentolinium Thioridazine may decrease the antihypertensive activities of Pentolinium.
Trimethaphan Thioridazine may decrease the antihypertensive activities of Trimethaphan.
Diazoxide Thioridazine may decrease the antihypertensive activities of Diazoxide.
Guanethidine Thioridazine may decrease the antihypertensive activities of Guanethidine.
Rescinnamine Thioridazine may decrease the antihypertensive activities of Rescinnamine.
Epoprostenol Thioridazine may decrease the antihypertensive activities of Epoprostenol.
Hydralazine Thioridazine may decrease the antihypertensive activities of Hydralazine.
Polythiazide Thioridazine may decrease the antihypertensive activities of Polythiazide.
Cilazapril Thioridazine may decrease the antihypertensive activities of Cilazapril.
Saprisartan Thioridazine may decrease the antihypertensive activities of Saprisartan.
Spirapril Thioridazine may decrease the antihypertensive activities of Spirapril.
Tienilic acid Thioridazine may decrease the antihypertensive activities of Tienilic acid.
Ambrisentan Thioridazine may decrease the antihypertensive activities of Ambrisentan.
Diethylnorspermine Thioridazine may decrease the antihypertensive activities of Diethylnorspermine.
Pinacidil Thioridazine may decrease the antihypertensive activities of Pinacidil.
Temocapril Thioridazine may decrease the antihypertensive activities of Temocapril.
Macitentan Thioridazine may decrease the antihypertensive activities of Macitentan.
Aliskiren Thioridazine may decrease the antihypertensive activities of Aliskiren.
Rauwolfia serpentina root Thioridazine may decrease the antihypertensive activities of Rauwolfia serpentina root.
Enalaprilat Thioridazine may decrease the antihypertensive activities of Enalaprilat.
Angiotensin 1-7 Thioridazine may decrease the antihypertensive activities of Angiotensin 1-7.
Imidapril Thioridazine may decrease the antihypertensive activities of Imidapril.
BQ-123 Thioridazine may decrease the antihypertensive activities of BQ-123.
Dihydralazine Thioridazine may decrease the antihypertensive activities of Dihydralazine.
Zofenopril Thioridazine may decrease the antihypertensive activities of Zofenopril.
Guanoxan Thioridazine may decrease the antihypertensive activities of Guanoxan.
Delapril Thioridazine may decrease the antihypertensive activities of Delapril.
Vincamine Thioridazine may decrease the antihypertensive activities of Vincamine.
Linsidomine Thioridazine may decrease the antihypertensive activities of Linsidomine.
Guanoxabenz Thioridazine may decrease the antihypertensive activities of Guanoxabenz.
Tolonidine Thioridazine may decrease the antihypertensive activities of Tolonidine.
Endralazine Thioridazine may decrease the antihypertensive activities of Endralazine.
Cadralazine Thioridazine may decrease the antihypertensive activities of Cadralazine.
Cyclopenthiazide Thioridazine may decrease the antihypertensive activities of Cyclopenthiazide.
Bietaserpine Thioridazine may decrease the antihypertensive activities of Bietaserpine.
Guanazodine Thioridazine may decrease the antihypertensive activities of Guanazodine.
Methoserpidine Thioridazine may decrease the antihypertensive activities of Methoserpidine.
Guanoclor Thioridazine may decrease the antihypertensive activities of Guanoclor.
Muzolimine Thioridazine may decrease the antihypertensive activities of Muzolimine.
Xipamide Thioridazine may decrease the antihypertensive activities of Xipamide.
Candesartan Thioridazine may decrease the antihypertensive activities of Candesartan.
Tocopherylquinone Thioridazine may decrease the antihypertensive activities of Tocopherylquinone.
Benazeprilat Thioridazine may decrease the antihypertensive activities of Benazeprilat.
Fosinoprilat Thioridazine may decrease the antihypertensive activities of Fosinoprilat.
Ramiprilat Thioridazine may decrease the antihypertensive activities of Ramiprilat.
Perindoprilat Thioridazine may decrease the antihypertensive activities of Perindoprilat.
Quinaprilat Thioridazine may decrease the antihypertensive activities of Quinaprilat.
Torasemide Thioridazine may decrease the antihypertensive activities of Torasemide.
Irbesartan Thioridazine may decrease the antihypertensive activities of Irbesartan.
Captopril Thioridazine may decrease the antihypertensive activities of Captopril.
Riociguat Thioridazine may decrease the antihypertensive activities of Riociguat.
Selexipag Thioridazine may decrease the antihypertensive activities of Selexipag.
Levamlodipine Thioridazine may decrease the antihypertensive activities of Levamlodipine.
Buthiazide Thioridazine may decrease the antihypertensive activities of Buthiazide.
Buprenorphine Thioridazine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Thioridazine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Thioridazine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Thioridazine.
Hydrocodone Thioridazine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Magnesium sulfate The therapeutic efficacy of Thioridazine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Thioridazine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Thioridazine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Thioridazine.
Orphenadrine Thioridazine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.

Target Protein

D(2) dopamine receptor DRD2
D(1A) dopamine receptor DRD1
Alpha-1A adrenergic receptor ADRA1A
Alpha-1B adrenergic receptor ADRA1B
5-hydroxytryptamine receptor 2A HTR2A
Voltage-gated inwardly rectifying potassium channel KCNH2 KCNH2

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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