Peringatan Keamanan

Symptoms of overdose include nausea and vomiting. Estrogen related side effects include nausea, breast tenderness, fluid retention and edema, headaches and/or migraines, chloasma and poor contact lens fit. Estrogen hormone deficiency is associated with breakthrough bleeding, hypomenorrhea, irritability, depression and menopausal symptoms. Withdrawal bleeds may occur in females.

Estrone

DB00655

small molecule approved

Deskripsi

Estrone, one of the major mammalian estrogens, is an aromatized C18 steroid with a 3-hydroxyl group and a 17-ketone. It is produced in vivo from androstenedione or from testosterone via estradiol. It is produced primarily in the ovaries, placenta, and in peripheral tissues (especially adipose tissue) through conversion of adrostenedione. Estrone may be further metabolized to 16-alpha-hydroxyestrone, which may be reduced to estriol by estradiol dehydrogenase.

Struktur Molekul 2D

Berat 270.3661
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 19 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

43%

Metabolisme

Hepatic.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol. Ingesting alcohol may increase serum concentrations of estradiol.
  • 2. Avoid grapefruit products. Grapefruit inhibits CYP3A4 and therefore, may increase estrone concentrations, potentially increasing its adverse effects.

Interaksi Obat

449 Data
Prasterone The risk or severity of adverse effects can be increased when Prasterone is combined with Estrone.
Exemestane The therapeutic efficacy of Exemestane can be decreased when used in combination with Estrone.
Lenalidomide Estrone may increase the thrombogenic activities of Lenalidomide.
Ospemifene The risk or severity of adverse effects can be increased when Estrone is combined with Ospemifene.
Ropinirole Estrone may increase the excretion rate of Ropinirole which could result in a lower serum level and potentially a reduction in efficacy.
Thalidomide Estrone may increase the thrombogenic activities of Thalidomide.
Cetuximab Estrone may increase the thrombogenic activities of Cetuximab.
Human immunoglobulin G Estrone may increase the thrombogenic activities of Human immunoglobulin G.
Omalizumab Estrone may increase the thrombogenic activities of Omalizumab.
Gemtuzumab ozogamicin Estrone may increase the thrombogenic activities of Gemtuzumab ozogamicin.
Indium In-111 satumomab pendetide Estrone may increase the thrombogenic activities of Indium In-111 satumomab pendetide.
Trastuzumab Estrone may increase the thrombogenic activities of Trastuzumab.
Rituximab Estrone may increase the thrombogenic activities of Rituximab.
Basiliximab Estrone may increase the thrombogenic activities of Basiliximab.
Muromonab Estrone may increase the thrombogenic activities of Muromonab.
Digoxin Immune Fab (Ovine) Estrone may increase the thrombogenic activities of Digoxin Immune Fab (Ovine).
Ibritumomab tiuxetan Estrone may increase the thrombogenic activities of Ibritumomab tiuxetan.
Tositumomab Estrone may increase the thrombogenic activities of Tositumomab.
Alemtuzumab Estrone may increase the thrombogenic activities of Alemtuzumab.
Capromab pendetide Estrone may increase the thrombogenic activities of Capromab pendetide.
Efalizumab Estrone may increase the thrombogenic activities of Efalizumab.
Antithymocyte immunoglobulin (rabbit) Estrone may increase the thrombogenic activities of Antithymocyte immunoglobulin (rabbit).
Natalizumab Estrone may increase the thrombogenic activities of Natalizumab.
Palivizumab Estrone may increase the thrombogenic activities of Palivizumab.
Daclizumab Estrone may increase the thrombogenic activities of Daclizumab.
Bevacizumab Estrone may increase the thrombogenic activities of Bevacizumab.
Technetium Tc-99m arcitumomab Estrone may increase the thrombogenic activities of Technetium Tc-99m arcitumomab.
Eculizumab Estrone may increase the thrombogenic activities of Eculizumab.
Panitumumab Estrone may increase the thrombogenic activities of Panitumumab.
Ranibizumab Estrone may increase the thrombogenic activities of Ranibizumab.
Galiximab Estrone may increase the thrombogenic activities of Galiximab.
Pexelizumab Estrone may increase the thrombogenic activities of Pexelizumab.
Epratuzumab Estrone may increase the thrombogenic activities of Epratuzumab.
Bectumomab Estrone may increase the thrombogenic activities of Bectumomab.
Oregovomab Estrone may increase the thrombogenic activities of Oregovomab.
IGN311 Estrone may increase the thrombogenic activities of IGN311.
Adecatumumab Estrone may increase the thrombogenic activities of Adecatumumab.
Labetuzumab Estrone may increase the thrombogenic activities of Labetuzumab.
Matuzumab Estrone may increase the thrombogenic activities of Matuzumab.
Fontolizumab Estrone may increase the thrombogenic activities of Fontolizumab.
Bavituximab Estrone may increase the thrombogenic activities of Bavituximab.
CR002 Estrone may increase the thrombogenic activities of CR002.
Rozrolimupab Estrone may increase the thrombogenic activities of Rozrolimupab.
Girentuximab Estrone may increase the thrombogenic activities of Girentuximab.
Obiltoxaximab Estrone may increase the thrombogenic activities of Obiltoxaximab.
XTL-001 Estrone may increase the thrombogenic activities of XTL-001.
NAV 1800 Estrone may increase the thrombogenic activities of NAV 1800.
Briakinumab Estrone may increase the thrombogenic activities of Briakinumab.
Otelixizumab Estrone may increase the thrombogenic activities of Otelixizumab.
AMG 108 Estrone may increase the thrombogenic activities of AMG 108.
Iratumumab Estrone may increase the thrombogenic activities of Iratumumab.
Enokizumab Estrone may increase the thrombogenic activities of Enokizumab.
Ramucirumab Estrone may increase the thrombogenic activities of Ramucirumab.
Farletuzumab Estrone may increase the thrombogenic activities of Farletuzumab.
Veltuzumab Estrone may increase the thrombogenic activities of Veltuzumab.
Ustekinumab Estrone may increase the thrombogenic activities of Ustekinumab.
PRO-542 Estrone may increase the thrombogenic activities of PRO-542.
TNX-901 Estrone may increase the thrombogenic activities of TNX-901.
Inotuzumab ozogamicin Estrone may increase the thrombogenic activities of Inotuzumab ozogamicin.
RI 624 Estrone may increase the thrombogenic activities of RI 624.
Stamulumab Estrone may increase the thrombogenic activities of MYO-029.
CT-011 Estrone may increase the thrombogenic activities of CT-011.
Leronlimab Estrone may increase the thrombogenic activities of Leronlimab.
Glembatumumab vedotin Estrone may increase the thrombogenic activities of Glembatumumab vedotin.
Olaratumab Estrone may increase the thrombogenic activities of Olaratumab.
IPH 2101 Estrone may increase the thrombogenic activities of IPH 2101.
TB-402 Estrone may increase the thrombogenic activities of TB-402.
Caplacizumab Estrone may increase the thrombogenic activities of Caplacizumab.
IMC-1C11 Estrone may increase the thrombogenic activities of IMC-1C11.
Eldelumab Estrone may increase the thrombogenic activities of Eldelumab.
Lumiliximab Estrone may increase the thrombogenic activities of Lumiliximab.
Ipilimumab Estrone may increase the thrombogenic activities of Ipilimumab.
Nimotuzumab Estrone may increase the thrombogenic activities of Nimotuzumab.
Clenoliximab Estrone may increase the thrombogenic activities of Clenoliximab.
BIIB015 Estrone may increase the thrombogenic activities of BIIB015.
Sonepcizumab Estrone may increase the thrombogenic activities of Sonepcizumab.
Motavizumab Estrone may increase the thrombogenic activities of Motavizumab.
Elotuzumab Estrone may increase the thrombogenic activities of Elotuzumab.
AVE9633 Estrone may increase the thrombogenic activities of AVE9633.
Carotuximab Estrone may increase the thrombogenic activities of Carotuximab.
XmAb 2513 Estrone may increase the thrombogenic activities of XmAb 2513.
Coltuximab ravtansine Estrone may increase the thrombogenic activities of Coltuximab ravtansine.
Lucatumumab Estrone may increase the thrombogenic activities of Lucatumumab.
Pertuzumab Estrone may increase the thrombogenic activities of Pertuzumab.
Siplizumab Estrone may increase the thrombogenic activities of Siplizumab.
Apolizumab Estrone may increase the thrombogenic activities of Apolizumab.
Sibrotuzumab Estrone may increase the thrombogenic activities of Sibrotuzumab.
Bivatuzumab Estrone may increase the thrombogenic activities of Bivatuzumab.
Lerdelimumab Estrone may increase the thrombogenic activities of Lerdelimumab.
Lexatumumab Estrone may increase the thrombogenic activities of Lexatumumab.
Reslizumab Estrone may increase the thrombogenic activities of Reslizumab.
Teplizumab Estrone may increase the thrombogenic activities of Teplizumab.
Catumaxomab Estrone may increase the thrombogenic activities of Catumaxomab.
Mepolizumab Estrone may increase the thrombogenic activities of Mepolizumab.
Denosumab Estrone may increase the thrombogenic activities of Denosumab.
Volociximab Estrone may increase the thrombogenic activities of Volociximab.
Ofatumumab Estrone may increase the thrombogenic activities of Ofatumumab.
Brentuximab vedotin Estrone may increase the thrombogenic activities of Brentuximab vedotin.
Belimumab Estrone may increase the thrombogenic activities of Belimumab.
Raxibacumab Estrone may increase the thrombogenic activities of Raxibacumab.

Target Protein

Estrogen receptor ESR1
Estrogen receptor beta ESR2
Androgen receptor AR
Aromatase CYP19A1
Sex hormone-binding globulin SHBG

Referensi & Sumber

Synthesis reference: Seiichi Takano, Kunio Ogasawara, "Method for producing (+)-estrone derivatives." U.S. Patent US5424462, issued January, 1965.
Artikel (PubMed)
  • PMID: 12796390
    Miyoshi Y, Tanji Y, Taguchi T, Tamaki Y, Noguchi S: Association of serum estrone levels with estrogen receptor-positive breast cancer risk in postmenopausal Japanese women. Clin Cancer Res. 2003 Jun;9(6):2229-33.
  • PMID: 12866733
    Kajta M, Lason W, Bien E, Marszal M: Neuroprotective effects of estrone on NMDA-induced toxicity in primary cultures of rat cortical neurons are independent of estrogen receptors. Pol J Pharmacol. 2002 Nov-Dec;54(6):727-9.

Contoh Produk & Brand

Produk: 3 • International brands: 1
Produk
  • Estragyn Vaginal Cream
    Cream • 0.1 % w/w • Vaginal • Canada • Approved
  • Oestrilin Cones Vaginaux
    Suppository • .25 mg / sup • Vaginal • Canada • Approved
  • Oestrilin Creme Vaginale 1mg
    Cream • 1 mg / g • Vaginal • Canada • Approved
International Brands
  • Estrone — Watson

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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