Peringatan Keamanan

LD50 = 1200 mg/kg (rat, subcutaneous). May be harmful if swallowed. May act as an irritant. Adverse reactions include hypotension, ECG changes, diarrhea, urinary retention, CNS depression and respiratory depression.

Magnesium sulfate

DB00653

small molecule approved investigational vet_approved

Deskripsi

A small colorless crystal used as an anticonvulsant, a cathartic, and an electrolyte replenisher in the treatment of pre-eclampsia and eclampsia. It causes direct inhibition of action potentials in myometrial muscle cells. Excitation and contraction are uncoupled, which decreases the frequency and force of contractions. (From AMA Drug Evaluations Annual, 1992, p1083)

Struktur Molekul 2D

Berat 120.368
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 43.2 hours (for newborns)
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

None

Rute Eliminasi

Magnesium is excreted solely by the kidney at a rate proportional to the serum concentration and glomerular filtration.

Interaksi Obat

1607 Data
Ceritinib Magnesium sulfate may increase the bradycardic activities of Ceritinib.
Ivabradine Magnesium sulfate may increase the bradycardic activities of Ivabradine.
Ruxolitinib Ruxolitinib may increase the bradycardic activities of Magnesium sulfate.
Buprenorphine Magnesium sulfate may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Magnesium sulfate.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Magnesium sulfate.
Botulinum toxin type B The therapeutic efficacy of Botulinum toxin type B can be increased when used in combination with Magnesium sulfate.
Botulinum toxin type A The therapeutic efficacy of Botulinum toxin type A can be increased when used in combination with Magnesium sulfate.
Fluvoxamine The therapeutic efficacy of Fluvoxamine can be increased when used in combination with Magnesium sulfate.
Baclofen The therapeutic efficacy of Baclofen can be increased when used in combination with Magnesium sulfate.
Lorazepam The therapeutic efficacy of Lorazepam can be increased when used in combination with Magnesium sulfate.
Ethchlorvynol The therapeutic efficacy of Ethchlorvynol can be increased when used in combination with Magnesium sulfate.
Tramadol The therapeutic efficacy of Tramadol can be increased when used in combination with Magnesium sulfate.
Succinylcholine The therapeutic efficacy of Succinylcholine can be increased when used in combination with Magnesium sulfate.
Reserpine The therapeutic efficacy of Reserpine can be increased when used in combination with Magnesium sulfate.
Citalopram The therapeutic efficacy of Citalopram can be increased when used in combination with Magnesium sulfate.
Eletriptan The therapeutic efficacy of Eletriptan can be increased when used in combination with Magnesium sulfate.
Enflurane The therapeutic efficacy of Enflurane can be increased when used in combination with Magnesium sulfate.
Pregabalin The therapeutic efficacy of Pregabalin can be increased when used in combination with Magnesium sulfate.
Temazepam The therapeutic efficacy of Temazepam can be increased when used in combination with Magnesium sulfate.
Reboxetine The therapeutic efficacy of Reboxetine can be increased when used in combination with Magnesium sulfate.
Butabarbital The therapeutic efficacy of Butabarbital can be increased when used in combination with Magnesium sulfate.
Butalbital The therapeutic efficacy of Butalbital can be increased when used in combination with Magnesium sulfate.
Ziprasidone The therapeutic efficacy of Ziprasidone can be increased when used in combination with Magnesium sulfate.
Methysergide The therapeutic efficacy of Methysergide can be increased when used in combination with Magnesium sulfate.
Cabergoline The therapeutic efficacy of Cabergoline can be increased when used in combination with Magnesium sulfate.
Phenytoin The therapeutic efficacy of Phenytoin can be increased when used in combination with Magnesium sulfate.
Topiramate The therapeutic efficacy of Topiramate can be increased when used in combination with Magnesium sulfate.
Clemastine The therapeutic efficacy of Clemastine can be increased when used in combination with Magnesium sulfate.
Venlafaxine The therapeutic efficacy of Venlafaxine can be increased when used in combination with Magnesium sulfate.
Etomidate The therapeutic efficacy of Etomidate can be increased when used in combination with Magnesium sulfate.
Morphine The therapeutic efficacy of Morphine can be increased when used in combination with Magnesium sulfate.
Talbutal The therapeutic efficacy of Talbutal can be increased when used in combination with Magnesium sulfate.
Pentobarbital The therapeutic efficacy of Pentobarbital can be increased when used in combination with Magnesium sulfate.
Valproic acid The therapeutic efficacy of Valproic acid can be increased when used in combination with Magnesium sulfate.
Zolmitriptan The therapeutic efficacy of Zolmitriptan can be increased when used in combination with Magnesium sulfate.
Codeine The therapeutic efficacy of Codeine can be increased when used in combination with Magnesium sulfate.
Dihydroergotamine The therapeutic efficacy of Dihydroergotamine can be increased when used in combination with Magnesium sulfate.
Amitriptyline The therapeutic efficacy of Amitriptyline can be increased when used in combination with Magnesium sulfate.
Tolcapone The therapeutic efficacy of Tolcapone can be increased when used in combination with Magnesium sulfate.
Hydromorphone The therapeutic efficacy of Hydromorphone can be increased when used in combination with Magnesium sulfate.
Olanzapine The therapeutic efficacy of Olanzapine can be increased when used in combination with Magnesium sulfate.
Cetirizine The therapeutic efficacy of Cetirizine can be increased when used in combination with Magnesium sulfate.
Protriptyline The therapeutic efficacy of Protriptyline can be increased when used in combination with Magnesium sulfate.
Trimethadione The therapeutic efficacy of Trimethadione can be increased when used in combination with Magnesium sulfate.
Clobazam The therapeutic efficacy of Clobazam can be increased when used in combination with Magnesium sulfate.
Chlorzoxazone The therapeutic efficacy of Chlorzoxazone can be increased when used in combination with Magnesium sulfate.
Clozapine The therapeutic efficacy of Clozapine can be increased when used in combination with Magnesium sulfate.
Mirtazapine The therapeutic efficacy of Mirtazapine can be increased when used in combination with Magnesium sulfate.
Meprobamate The therapeutic efficacy of Meprobamate can be increased when used in combination with Magnesium sulfate.
Thiethylperazine The therapeutic efficacy of Thiethylperazine can be increased when used in combination with Magnesium sulfate.
Palonosetron The therapeutic efficacy of Palonosetron can be increased when used in combination with Magnesium sulfate.
Sulpiride The therapeutic efficacy of Sulpiride can be increased when used in combination with Magnesium sulfate.
Carisoprodol The therapeutic efficacy of Carisoprodol can be increased when used in combination with Magnesium sulfate.
Eszopiclone The therapeutic efficacy of Eszopiclone can be increased when used in combination with Magnesium sulfate.
Alprazolam The therapeutic efficacy of Alprazolam can be increased when used in combination with Magnesium sulfate.
Dexbrompheniramine The therapeutic efficacy of Dexbrompheniramine can be increased when used in combination with Magnesium sulfate.
Loxapine The therapeutic efficacy of Loxapine can be increased when used in combination with Magnesium sulfate.
Remoxipride The therapeutic efficacy of Remoxipride can be increased when used in combination with Magnesium sulfate.
Metocurine iodide The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium sulfate.
Secobarbital The therapeutic efficacy of Secobarbital can be increased when used in combination with Magnesium sulfate.
Promazine The therapeutic efficacy of Promazine can be increased when used in combination with Magnesium sulfate.
Methocarbamol The therapeutic efficacy of Methocarbamol can be increased when used in combination with Magnesium sulfate.
Zolpidem The therapeutic efficacy of Zolpidem can be increased when used in combination with Magnesium sulfate.
Triprolidine The therapeutic efficacy of Triprolidine can be increased when used in combination with Magnesium sulfate.
Prochlorperazine The therapeutic efficacy of Prochlorperazine can be increased when used in combination with Magnesium sulfate.
Cyproheptadine The therapeutic efficacy of Cyproheptadine can be increased when used in combination with Magnesium sulfate.
Droperidol The therapeutic efficacy of Droperidol can be increased when used in combination with Magnesium sulfate.
Meperidine The therapeutic efficacy of Meperidine can be increased when used in combination with Magnesium sulfate.
Imipramine The therapeutic efficacy of Imipramine can be increased when used in combination with Magnesium sulfate.
Metharbital The therapeutic efficacy of Metharbital can be increased when used in combination with Magnesium sulfate.
Quinine The therapeutic efficacy of Quinine can be increased when used in combination with Magnesium sulfate.
Dronabinol The therapeutic efficacy of Dronabinol can be increased when used in combination with Magnesium sulfate.
Fluoxetine The therapeutic efficacy of Fluoxetine can be increased when used in combination with Magnesium sulfate.
Methohexital The therapeutic efficacy of Methohexital can be increased when used in combination with Magnesium sulfate.
Chlordiazepoxide The therapeutic efficacy of Chlordiazepoxide can be increased when used in combination with Magnesium sulfate.
Duloxetine The therapeutic efficacy of Duloxetine can be increased when used in combination with Magnesium sulfate.
Chlorpromazine The therapeutic efficacy of Chlorpromazine can be increased when used in combination with Magnesium sulfate.
Gallamine triethiodide The therapeutic efficacy of Gallamine triethiodide can be increased when used in combination with Magnesium sulfate.
Nabilone The therapeutic efficacy of Nabilone can be increased when used in combination with Magnesium sulfate.
Entacapone The therapeutic efficacy of Entacapone can be increased when used in combination with Magnesium sulfate.
Oxycodone The therapeutic efficacy of Oxycodone can be increased when used in combination with Magnesium sulfate.
Haloperidol The therapeutic efficacy of Haloperidol can be increased when used in combination with Magnesium sulfate.
Triflupromazine The therapeutic efficacy of Triflupromazine can be increased when used in combination with Magnesium sulfate.
Dextromethorphan The therapeutic efficacy of Dextromethorphan can be increased when used in combination with Magnesium sulfate.
Mephenytoin The therapeutic efficacy of Mephenytoin can be increased when used in combination with Magnesium sulfate.
Nortriptyline The therapeutic efficacy of Nortriptyline can be increased when used in combination with Magnesium sulfate.
Amoxapine The therapeutic efficacy of Amoxapine can be increased when used in combination with Magnesium sulfate.
Adinazolam The therapeutic efficacy of Adinazolam can be increased when used in combination with Magnesium sulfate.
Lamotrigine The therapeutic efficacy of Lamotrigine can be increased when used in combination with Magnesium sulfate.
Carbamazepine The therapeutic efficacy of Carbamazepine can be increased when used in combination with Magnesium sulfate.
Cisatracurium The therapeutic efficacy of Cisatracurium can be increased when used in combination with Magnesium sulfate.
Fenfluramine The therapeutic efficacy of Fenfluramine can be increased when used in combination with Magnesium sulfate.
Mazindol The therapeutic efficacy of Mazindol can be increased when used in combination with Magnesium sulfate.
Fluticasone propionate The therapeutic efficacy of Fluticasone propionate can be increased when used in combination with Magnesium sulfate.
Lisuride The therapeutic efficacy of Lisuride can be increased when used in combination with Magnesium sulfate.
Ethosuximide The therapeutic efficacy of Ethosuximide can be increased when used in combination with Magnesium sulfate.
Thiopental The therapeutic efficacy of Thiopental can be increased when used in combination with Magnesium sulfate.
Cisapride The therapeutic efficacy of Cisapride can be increased when used in combination with Magnesium sulfate.
Butorphanol The therapeutic efficacy of Butorphanol can be increased when used in combination with Magnesium sulfate.

Target Protein

Voltage-dependent L-type calcium channel CACNA1C

Referensi & Sumber

Synthesis reference: Shinichi Yamamoto, Akifumi Sekitani, "BASIC MAGNESIUM SULFATE GRANULE, AND PROCESS FOR PRODUCTION THEREOF." U.S. Patent US20110042297, issued February 24, 2011.
Artikel (PubMed)
  • PMID: 16002955
    Blitz M, Blitz S, Hughes R, Diner B, Beasley R, Knopp J, Rowe BH: Aerosolized magnesium sulfate for acute asthma: a systematic review. Chest. 2005 Jul;128(1):337-44.
  • PMID: 20226604
    Yokoyama K, Takahashi N, Yada Y, Koike Y, Kawamata R, Uehara R, Kono Y, Honma Y, Momoi MY: Prolonged maternal magnesium administration and bone metabolism in neonates. Early Hum Dev. 2010 Mar;86(3):187-91. doi: 10.1016/j.earlhumdev.2010.02.007. Epub 2010 Mar 12.
  • PMID: 16724078
    Wedig KE, Kogan J, Schorry EK, Whitsett JA: Skeletal demineralization and fractures caused by fetal magnesium toxicity. J Perinatol. 2006 Jun;26(6):371-4.
  • PMID: 16929415
    Nassar AH, Sakhel K, Maarouf H, Naassan GR, Usta IM: Adverse maternal and neonatal outcome of prolonged course of magnesium sulfate tocolysis. Acta Obstet Gynecol Scand. 2006;85(9):1099-103.
  • PMID: 14985884
    Malaeb SN, Rassi AI, Haddad MC, Seoud MA, Yunis KA: Bone mineralization in newborns whose mothers received magnesium sulphate for tocolysis of premature labour. Pediatr Radiol. 2004 May;34(5):384-6. Epub 2004 Feb 18.
  • PMID: 9286718
    Matsuda Y, Maeda Y, Ito M, Sakamoto H, Masaoka N, Takada M, Sato K: Effect of magnesium sulfate treatment on neonatal bone abnormalities. Gynecol Obstet Invest. 1997;44(2):82-8.
  • PMID: 9194621
    Schanler RJ, Smith LG Jr, Burns PA: Effects of long-term maternal intravenous magnesium sulfate therapy on neonatal calcium metabolism and bone mineral content. Gynecol Obstet Invest. 1997;43(4):236-41.
  • PMID: 8188843
    Santi MD, Henry GW, Douglas GL: Magnesium sulfate treatment of preterm labor as a cause of abnormal neonatal bone mineralization. J Pediatr Orthop. 1994 Mar-Apr;14(2):249-53.
Menampilkan 8 dari 13 artikel.

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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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