Pentazocine

DB00652

small molecule approved vet_approved

Deskripsi

The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor. (From AMA Drug Evaluations Annual, 1991, p97)

Struktur Molekul 2D

Berat 285.431
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 2 to 3 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Well absorbed from the gastro-intestinal tract.

Metabolisme

Hepatic

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol.
  • 2. Take with or without food. Food does not significantly affect absorption.

Interaksi Obat

921 Data
Buprenorphine Pentazocine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Pentazocine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Pentazocine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Pentazocine.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Pentazocine.
Magnesium sulfate The therapeutic efficacy of Pentazocine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Pentazocine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Pentazocine may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Pentazocine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Pentazocine.
Orphenadrine Pentazocine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Pentazocine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Pentazocine.
Pramipexole Pentazocine may increase the sedative activities of Pramipexole.
Ropinirole Pentazocine may increase the sedative activities of Ropinirole.
Rotigotine Pentazocine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Pentazocine.
Sodium oxybate Pentazocine may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Pentazocine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol The therapeutic efficacy of Tapentadol can be decreased when used in combination with Pentazocine.
Thalidomide Pentazocine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Pentazocine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Alvimopan The risk or severity of adverse effects can be increased when Pentazocine is combined with Alvimopan.
Desmopressin The risk or severity of hyponatremia can be increased when Pentazocine is combined with Desmopressin.
Pegvisomant The therapeutic efficacy of Pegvisomant can be decreased when used in combination with Pentazocine.
Succinylcholine The risk or severity of bradycardia can be increased when Succinylcholine is combined with Pentazocine.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Pentazocine.
Linezolid The risk or severity of serotonin syndrome can be increased when Linezolid is combined with Pentazocine.
Methylnaltrexone Pentazocine may increase the opioid antagonism activities of Methylnaltrexone.
Naloxegol Pentazocine may increase the opioid antagonism activities of Naloxegol.
Mirtazapine Pentazocine may increase the serotonergic activities of Mirtazapine.
Fluvoxamine The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Fluvoxamine.
Citalopram The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Citalopram.
Duloxetine The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Duloxetine.
Paroxetine The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Paroxetine.
Sertraline The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Sertraline.
Sibutramine The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Sibutramine.
Nefazodone The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Nefazodone.
Zimelidine The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Zimelidine.
Dapoxetine The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Dapoxetine.
Milnacipran The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Milnacipran.
Desvenlafaxine The risk or severity of serotonin syndrome can be increased when Desvenlafaxine is combined with Pentazocine.
Seproxetine The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Seproxetine.
Levomilnacipran The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Levomilnacipran.
Indalpine The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Indalpine.
Ritanserin The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Ritanserin.
Alaproclate The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Alaproclate.
Ethanol Pentazocine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Pentazocine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Pentazocine.
Phentermine Phentermine may increase the analgesic activities of Pentazocine.
Pseudoephedrine Pseudoephedrine may increase the analgesic activities of Pentazocine.
Benzphetamine Benzphetamine may increase the analgesic activities of Pentazocine.
Diethylpropion Diethylpropion may increase the analgesic activities of Pentazocine.
Lisdexamfetamine The risk or severity of serotonin syndrome can be increased when Pentazocine is combined with Lisdexamfetamine.
Mephentermine Mephentermine may increase the analgesic activities of Pentazocine.
MMDA MMDA may increase the analgesic activities of Pentazocine.
Midomafetamine Midomafetamine may increase the analgesic activities of Pentazocine.
2,5-Dimethoxy-4-ethylamphetamine 2,5-Dimethoxy-4-ethylamphetamine may increase the analgesic activities of Pentazocine.
4-Bromo-2,5-dimethoxyamphetamine 4-Bromo-2,5-dimethoxyamphetamine may increase the analgesic activities of Pentazocine.
Tenamfetamine Tenamfetamine may increase the analgesic activities of Pentazocine.
Chlorphentermine Chlorphentermine may increase the analgesic activities of Pentazocine.
Methylenedioxyethamphetamine Methylenedioxyethamphetamine may increase the analgesic activities of Pentazocine.
Dextroamphetamine Dextroamphetamine may increase the analgesic activities of Pentazocine.
Metamfetamine Metamfetamine may increase the analgesic activities of Pentazocine.
Iofetamine I-123 Iofetamine I-123 may increase the analgesic activities of Pentazocine.
Ritobegron Ritobegron may increase the analgesic activities of Pentazocine.
Mephedrone Mephedrone may increase the analgesic activities of Pentazocine.
Methoxyphenamine Methoxyphenamine may increase the analgesic activities of Pentazocine.
Gepefrine Gepefrine may increase the analgesic activities of Pentazocine.
2,5-Dimethoxy-4-ethylthioamphetamine 2,5-Dimethoxy-4-ethylthioamphetamine may increase the analgesic activities of Pentazocine.
Amphetamine Amphetamine may increase the analgesic activities of Pentazocine.
Phendimetrazine Phendimetrazine may increase the analgesic activities of Pentazocine.
Mecamylamine The risk or severity of adverse effects can be increased when Mecamylamine is combined with Pentazocine.
Pentolinium The risk or severity of adverse effects can be increased when Pentolinium is combined with Pentazocine.
Trimethaphan The risk or severity of adverse effects can be increased when Trimethaphan is combined with Pentazocine.
Chloroprocaine The risk or severity of CNS depression can be increased when Pentazocine is combined with Chloroprocaine.
Fenoterol The risk or severity of adverse effects can be increased when Fenoterol is combined with Pentazocine.
Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione The risk or severity of adverse effects can be increased when Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione is combined with Pentazocine.
Agmatine The risk or severity of adverse effects can be increased when Agmatine is combined with Pentazocine.
Promazine The risk or severity of adverse effects can be increased when Promazine is combined with Pentazocine.
Chlorpromazine The risk or severity of adverse effects can be increased when Chlorpromazine is combined with Pentazocine.
Triflupromazine The risk or severity of adverse effects can be increased when Triflupromazine is combined with Pentazocine.
Promethazine The risk or severity of adverse effects can be increased when Promethazine is combined with Pentazocine.
Trospium The risk or severity of adverse effects can be increased when Trospium is combined with Pentazocine.
Oxyphenonium The risk or severity of adverse effects can be increased when Oxyphenonium is combined with Pentazocine.
Benzatropine The risk or severity of adverse effects can be increased when Benzatropine is combined with Pentazocine.
Disopyramide The risk or severity of adverse effects can be increased when Disopyramide is combined with Pentazocine.
Ipratropium The risk or severity of adverse effects can be increased when Ipratropium is combined with Pentazocine.
Metixene The risk or severity of adverse effects can be increased when Metixene is combined with Pentazocine.
Buclizine The risk or severity of adverse effects can be increased when Buclizine is combined with Pentazocine.
Trihexyphenidyl The risk or severity of adverse effects can be increased when Trihexyphenidyl is combined with Pentazocine.
Oxyphencyclimine The risk or severity of adverse effects can be increased when Oxyphencyclimine is combined with Pentazocine.
Procyclidine The risk or severity of adverse effects can be increased when Procyclidine is combined with Pentazocine.
Profenamine The risk or severity of adverse effects can be increased when Profenamine is combined with Pentazocine.
Hyoscyamine The risk or severity of adverse effects can be increased when Hyoscyamine is combined with Pentazocine.
Cyproheptadine The risk or severity of adverse effects can be increased when Cyproheptadine is combined with Pentazocine.
Methscopolamine bromide The risk or severity of adverse effects can be increased when Methscopolamine bromide is combined with Pentazocine.
Darifenacin The risk or severity of adverse effects can be increased when Darifenacin is combined with Pentazocine.
Tridihexethyl The risk or severity of adverse effects can be increased when Tridihexethyl is combined with Pentazocine.

Target Protein

Sigma non-opioid intracellular receptor 1 SIGMAR1
Mu-type opioid receptor OPRM1
Kappa-type opioid receptor OPRK1

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 24 • International brands: 8
Produk
  • Pentazocine and naloxone
    Tablet • - • Oral • US • Generic • Approved
  • Pentazocine and naloxone
    Tablet • - • Oral • US • Generic • Approved
  • Pentazocine and Naloxone
    Tablet • - • Oral • US • Generic • Approved
  • Pentazocine and naloxone
    Tablet • - • Oral • US • Generic • Approved
  • Pentazocine and Naloxone
    Tablet • - • Oral • US • Generic • Approved
  • Pentazocine and naloxone
    Tablet • - • Oral • US • Generic • Approved
  • Pentazocine and naloxone
    Tablet • - • Oral • US • Generic • Approved
  • Pentazocine and naloxone hydrochlorides
    Tablet • - • Oral • US • Generic • Approved
Menampilkan 8 dari 24 produk.
International Brands
  • Fortal — Sanofi-Aventis
  • Fortral — Sanofi-Aventis
  • Fortwin — Terapia
  • Pangon — L.B.S.
  • Pentagin — Daiichi Sankyo
  • Sosegon — Sanofi-Aventis
  • Stopain — Beximco
  • Talwin PX — Sanofi-Aventis

Sekuens Gen/Protein (FASTA)

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