Peringatan Keamanan

Symptoms of overdose include clumsiness or unsteadiness, coma, severe dizziness, severe drowsiness, severe nausea, and problems with vision.

Paramethadione

DB00617

small molecule approved

Deskripsi

Paramethadione is an anticonvulsant in the oxazolidinedione class. It is associated with fetal trimethadione syndrome, which is also known as paramethadione syndrome.

Struktur Molekul 2D

Berat 157.1671
Wujud liquid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 12 to 24 hours (however the half-life for the active metabolite is not known)
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Rapid via the digestive tract.

Metabolisme

Primarily hepatic (mainly via cytochrome P450 isozyme 2C9), paramethadione is completely demethylated to 5-ethyl-5-methyl-2,4-oxazolidinedione, the active metabolite.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1174 Data
Buprenorphine Paramethadione may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Paramethadione.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Paramethadione.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Paramethadione.
Hydrocodone Paramethadione may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Paramethadione.
Magnesium sulfate The therapeutic efficacy of Paramethadione can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Paramethadione may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Paramethadione may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Paramethadione.
Mirtazapine Paramethadione may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Paramethadione.
Orphenadrine Paramethadione may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Paramethadione may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Paramethadione.
Pramipexole Paramethadione may increase the sedative activities of Pramipexole.
Ropinirole Paramethadione may increase the sedative activities of Ropinirole.
Rotigotine Paramethadione may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Paramethadione.
Sodium oxybate Paramethadione may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Paramethadione may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Paramethadione.
Thalidomide Paramethadione may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Paramethadione may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Mefloquine The therapeutic efficacy of Paramethadione can be decreased when used in combination with Mefloquine.
Mianserin The therapeutic efficacy of Paramethadione can be decreased when used in combination with Mianserin.
Orlistat Orlistat can cause a decrease in the absorption of Paramethadione resulting in a reduced serum concentration and potentially a decrease in efficacy.
Topotecan Paramethadione may increase the excretion rate of Topotecan which could result in a lower serum level and potentially a reduction in efficacy.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Paramethadione.
Mifepristone The serum concentration of Paramethadione can be increased when it is combined with Mifepristone.
Tetracosactide The risk or severity of liver damage can be increased when Tetracosactide is combined with Paramethadione.
Ethanol Paramethadione may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Paramethadione may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Paramethadione.
Fluvoxamine The risk or severity of adverse effects can be increased when Paramethadione is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Paramethadione is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Paramethadione is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Paramethadione is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Paramethadione is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Paramethadione is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Paramethadione is combined with Sibutramine.
Escitalopram The risk or severity of adverse effects can be increased when Paramethadione is combined with Escitalopram.
Zimelidine The risk or severity of adverse effects can be increased when Paramethadione is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Paramethadione is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Paramethadione is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Paramethadione is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Paramethadione is combined with Seproxetine.
Indalpine The risk or severity of adverse effects can be increased when Paramethadione is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Paramethadione is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Paramethadione is combined with Alaproclate.
Cyproheptadine The risk or severity of CNS depression can be increased when Cyproheptadine is combined with Paramethadione.
Amoxapine The risk or severity of CNS depression can be increased when Amoxapine is combined with Paramethadione.
Propiomazine The risk or severity of CNS depression can be increased when Paramethadione is combined with Propiomazine.
Maprotiline The risk or severity of CNS depression can be increased when Paramethadione is combined with Maprotiline.
Tolterodine The metabolism of Tolterodine can be decreased when combined with Paramethadione.
Desipramine The risk or severity of CNS depression can be increased when Paramethadione is combined with Desipramine.
Pizotifen The risk or severity of CNS depression can be increased when Paramethadione is combined with Pizotifen.
Dosulepin The risk or severity of CNS depression can be increased when Paramethadione is combined with Dosulepin.
Imipramine The risk or severity of CNS depression can be increased when Imipramine is combined with Paramethadione.
Nortriptyline The risk or severity of CNS depression can be increased when Nortriptyline is combined with Paramethadione.
Quetiapine The risk or severity of CNS depression can be increased when Paramethadione is combined with Quetiapine.
Doxepin The risk or severity of CNS depression can be increased when Paramethadione is combined with Doxepin.
Cocaine The risk or severity of methemoglobinemia can be increased when Paramethadione is combined with Cocaine.
Quinidine The metabolism of Paramethadione can be decreased when combined with Quinidine.
Zopiclone The risk or severity of adverse effects can be increased when Paramethadione is combined with Zopiclone.
Botulinum toxin type B The risk or severity of CNS depression can be increased when Botulinum toxin type B is combined with Paramethadione.
Botulinum toxin type A The risk or severity of CNS depression can be increased when Botulinum toxin type A is combined with Paramethadione.
Tryptophan The risk or severity of CNS depression can be increased when Tryptophan is combined with Paramethadione.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of Paramethadione.
Lorazepam The risk or severity of CNS depression can be increased when Lorazepam is combined with Paramethadione.
Ethchlorvynol The risk or severity of CNS depression can be increased when Ethchlorvynol is combined with Paramethadione.
Succinylcholine The risk or severity of CNS depression can be increased when Succinylcholine is combined with Paramethadione.
Reserpine The risk or severity of CNS depression can be increased when Reserpine is combined with Paramethadione.
Enflurane The risk or severity of CNS depression can be increased when Enflurane is combined with Paramethadione.
Temazepam The risk or severity of CNS depression can be increased when Temazepam is combined with Paramethadione.
Reboxetine The risk or severity of CNS depression can be increased when Reboxetine is combined with Paramethadione.
Butabarbital The risk or severity of CNS depression can be increased when Butabarbital is combined with Paramethadione.
Butalbital The risk or severity of CNS depression can be increased when Butalbital is combined with Paramethadione.
Cabergoline The risk or severity of CNS depression can be increased when Cabergoline is combined with Paramethadione.
Topiramate The risk or severity of CNS depression can be increased when Topiramate is combined with Paramethadione.
Clemastine The risk or severity of CNS depression can be increased when Clemastine is combined with Paramethadione.
Venlafaxine The risk or severity of CNS depression can be increased when Venlafaxine is combined with Paramethadione.
Etomidate The risk or severity of CNS depression can be increased when Etomidate is combined with Paramethadione.
Morphine The risk or severity of CNS depression can be increased when Morphine is combined with Paramethadione.
Talbutal The risk or severity of CNS depression can be increased when Talbutal is combined with Paramethadione.
Zolmitriptan The risk or severity of CNS depression can be increased when Zolmitriptan is combined with Paramethadione.
Codeine The risk or severity of CNS depression can be increased when Codeine is combined with Paramethadione.
Tolcapone The risk or severity of CNS depression can be increased when Tolcapone is combined with Paramethadione.
Hydromorphone The risk or severity of CNS depression can be increased when Hydromorphone is combined with Paramethadione.
Olanzapine The risk or severity of CNS depression can be increased when Olanzapine is combined with Paramethadione.
Cetirizine The risk or severity of CNS depression can be increased when Cetirizine is combined with Paramethadione.
Protriptyline The risk or severity of CNS depression can be increased when Protriptyline is combined with Paramethadione.
Trimethadione The risk or severity of CNS depression can be increased when Trimethadione is combined with Paramethadione.
Clobazam The risk or severity of sedation, somnolence, and CNS depression can be increased when Clobazam is combined with Paramethadione.
Chlorzoxazone The risk or severity of CNS depression can be increased when Chlorzoxazone is combined with Paramethadione.
Clozapine The metabolism of Paramethadione can be decreased when combined with Clozapine.
Meprobamate The risk or severity of CNS depression can be increased when Meprobamate is combined with Paramethadione.
Thiethylperazine The risk or severity of CNS depression can be increased when Thiethylperazine is combined with Paramethadione.
Palonosetron The risk or severity of CNS depression can be increased when Palonosetron is combined with Paramethadione.
Sulpiride The risk or severity of CNS depression can be increased when Sulpiride is combined with Paramethadione.

Target Protein

Voltage-dependent T-type calcium channel subunit alpha-1G CACNA1G
Voltage-dependent T-type calcium channel subunit alpha-1I CACNA1I

Referensi & Sumber

Artikel (PubMed)
  • PMID: 1185541
    Hoffman DJ, Chun AH: Paramethadione and metabolite serum levels in humans after a single oral paramethadione dose. J Pharm Sci. 1975 Oct;64(10):1702-3.
  • PMID: 412416
    Feldman GL, Weaver DD, Lovrien EW: The fetal trimethadione syndrome: report of an additional family and further delineation of this syndrome. Am J Dis Child. 1977 Dec;131(12):1389-92.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Paradione

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul