Peringatan Keamanan

LD50 = 5 g/kg (Human, oral). Symptoms of overdose include muscle fatigue, seizures, and difficulty breathing.

Piperazine

DB00592

small molecule approved vet_approved

Deskripsi

Piperazine is an organic compound that consists of a six-membered ring containing two opposing nitrogen atoms. First used as a solvent for uric acid, the use of piperazine as an anthelmintic agent was first introduced in 1953. Upon entry into the systemic circulation, the drug is partly oxidized and partly eliminated as an unchanged compound. Outside the body, piperazine has a remarkable power to dissolve uric acid and producing a soluble urate, but in clinical experience it has not proved equally successful. Piperazine was first introduced as an anthelmintic in 1953. Piperazine compounds mediate their anthelmintic action by generally paralyzing parasites, allowing the host body to easily remove or expel the invading organism.

Struktur Molekul 2D

Berat 86.1356
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Rapidly absorbed from the gastrointestinal tract

Metabolisme

About 25% is metabolized in the liver. Piperazine is nitrosated to form N -mononitrosopiperazine (MNPz) in gastric juice, which is then metabolized to N-nitroso-3-hydroxypyrrolidine (NHPYR).

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

1 Data
  • 1. Take with or without food. The absorption is unaffected by food.

Interaksi Obat

443 Data
Mirabegron The serum concentration of Piperazine can be increased when it is combined with Mirabegron.
Insulin human The therapeutic efficacy of Insulin human can be decreased when used in combination with Piperazine.
Insulin lispro The therapeutic efficacy of Insulin lispro can be decreased when used in combination with Piperazine.
Insulin glargine The therapeutic efficacy of Insulin glargine can be decreased when used in combination with Piperazine.
Insulin pork The therapeutic efficacy of Insulin pork can be decreased when used in combination with Piperazine.
Troglitazone The therapeutic efficacy of Troglitazone can be decreased when used in combination with Piperazine.
Glimepiride The therapeutic efficacy of Glimepiride can be decreased when used in combination with Piperazine.
Sulfisoxazole The therapeutic efficacy of Sulfisoxazole can be decreased when used in combination with Piperazine.
Disopyramide The therapeutic efficacy of Disopyramide can be decreased when used in combination with Piperazine.
Acarbose The therapeutic efficacy of Acarbose can be decreased when used in combination with Piperazine.
Sulfadiazine The therapeutic efficacy of Sulfadiazine can be decreased when used in combination with Piperazine.
Rosiglitazone The therapeutic efficacy of Rosiglitazone can be decreased when used in combination with Piperazine.
Acetohexamide The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Piperazine.
Miglitol The therapeutic efficacy of Miglitol can be decreased when used in combination with Piperazine.
Chlorpropamide The therapeutic efficacy of Chlorpropamide can be decreased when used in combination with Piperazine.
Nateglinide The therapeutic efficacy of Nateglinide can be decreased when used in combination with Piperazine.
Pentamidine The therapeutic efficacy of Pentamidine can be decreased when used in combination with Piperazine.
Mifepristone The therapeutic efficacy of Mifepristone can be decreased when used in combination with Piperazine.
Tolazamide The therapeutic efficacy of Tolazamide can be decreased when used in combination with Piperazine.
Repaglinide The therapeutic efficacy of Repaglinide can be decreased when used in combination with Piperazine.
Phenformin The therapeutic efficacy of Phenformin can be decreased when used in combination with Piperazine.
Sulfamethoxazole The therapeutic efficacy of Sulfamethoxazole can be decreased when used in combination with Piperazine.
Glyburide The therapeutic efficacy of Glyburide can be decreased when used in combination with Piperazine.
Glipizide The therapeutic efficacy of Glipizide can be decreased when used in combination with Piperazine.
Gliclazide The therapeutic efficacy of Gliclazide can be decreased when used in combination with Piperazine.
Tolbutamide The therapeutic efficacy of Tolbutamide can be decreased when used in combination with Piperazine.
Pioglitazone The therapeutic efficacy of Pioglitazone can be decreased when used in combination with Piperazine.
Bromocriptine The therapeutic efficacy of Bromocriptine can be decreased when used in combination with Piperazine.
Gliquidone The therapeutic efficacy of Gliquidone can be decreased when used in combination with Piperazine.
Mitiglinide The therapeutic efficacy of Mitiglinide can be decreased when used in combination with Piperazine.
Sitagliptin The therapeutic efficacy of Sitagliptin can be decreased when used in combination with Piperazine.
Sunitinib The therapeutic efficacy of Sunitinib can be decreased when used in combination with Piperazine.
Exenatide The therapeutic efficacy of Exenatide can be decreased when used in combination with Piperazine.
Mecasermin The therapeutic efficacy of Mecasermin can be decreased when used in combination with Piperazine.
Pramlintide The therapeutic efficacy of Pramlintide can be decreased when used in combination with Piperazine.
Glisoxepide The therapeutic efficacy of Glisoxepide can be decreased when used in combination with Piperazine.
Insulin aspart The therapeutic efficacy of Insulin aspart can be decreased when used in combination with Piperazine.
Insulin detemir The therapeutic efficacy of Insulin detemir can be decreased when used in combination with Piperazine.
Insulin glulisine The therapeutic efficacy of Insulin glulisine can be decreased when used in combination with Piperazine.
Glymidine The therapeutic efficacy of Glymidine can be decreased when used in combination with Piperazine.
AICA ribonucleotide The therapeutic efficacy of AICA ribonucleotide can be decreased when used in combination with Piperazine.
Buformin The therapeutic efficacy of Buformin can be decreased when used in combination with Piperazine.
Vildagliptin The therapeutic efficacy of Vildagliptin can be decreased when used in combination with Piperazine.
Voglibose The therapeutic efficacy of Voglibose can be decreased when used in combination with Piperazine.
NN344 The therapeutic efficacy of NN344 can be decreased when used in combination with Piperazine.
AMG-222 The therapeutic efficacy of AMG-222 can be decreased when used in combination with Piperazine.
Bisegliptin The therapeutic efficacy of Bisegliptin can be decreased when used in combination with Piperazine.
Alogliptin The therapeutic efficacy of Alogliptin can be decreased when used in combination with Piperazine.
Dapagliflozin The therapeutic efficacy of Dapagliflozin can be decreased when used in combination with Piperazine.
Saxagliptin The therapeutic efficacy of Saxagliptin can be decreased when used in combination with Piperazine.
Liraglutide The therapeutic efficacy of Liraglutide can be decreased when used in combination with Piperazine.
Gosogliptin The therapeutic efficacy of Gosogliptin can be decreased when used in combination with Piperazine.
Linagliptin The therapeutic efficacy of Linagliptin can be decreased when used in combination with Piperazine.
Canagliflozin The therapeutic efficacy of Canagliflozin can be decreased when used in combination with Piperazine.
Glibornuride The therapeutic efficacy of Glibornuride can be decreased when used in combination with Piperazine.
Benfluorex The therapeutic efficacy of Benfluorex can be decreased when used in combination with Piperazine.
Empagliflozin The therapeutic efficacy of Empagliflozin can be decreased when used in combination with Piperazine.
Albiglutide The therapeutic efficacy of Albiglutide can be decreased when used in combination with Piperazine.
Dulaglutide The therapeutic efficacy of Dulaglutide can be decreased when used in combination with Piperazine.
Lobeglitazone The therapeutic efficacy of Lobeglitazone can be decreased when used in combination with Piperazine.
Netoglitazone The therapeutic efficacy of Netoglitazone can be decreased when used in combination with Piperazine.
Rivoglitazone The therapeutic efficacy of Rivoglitazone can be decreased when used in combination with Piperazine.
Ciglitazone The therapeutic efficacy of Ciglitazone can be decreased when used in combination with Piperazine.
Lixisenatide The therapeutic efficacy of Lixisenatide can be decreased when used in combination with Piperazine.
Insulin beef The therapeutic efficacy of Insulin beef can be decreased when used in combination with Piperazine.
Insulin degludec The therapeutic efficacy of Insulin degludec can be decreased when used in combination with Piperazine.
Insulin peglispro The therapeutic efficacy of Insulin peglispro can be decreased when used in combination with Piperazine.
Insulin tregopil The therapeutic efficacy of Insulin tregopil can be decreased when used in combination with Piperazine.
Ipragliflozin The therapeutic efficacy of Ipragliflozin can be decreased when used in combination with Piperazine.
Dutogliptin The therapeutic efficacy of Dutogliptin can be decreased when used in combination with Piperazine.
Allicin The therapeutic efficacy of Allicin can be decreased when used in combination with Piperazine.
Tofogliflozin The therapeutic efficacy of Tofogliflozin can be decreased when used in combination with Piperazine.
Ertugliflozin The therapeutic efficacy of Ertugliflozin can be decreased when used in combination with Piperazine.
2,4-thiazolidinedione The therapeutic efficacy of 2,4-thiazolidinedione can be decreased when used in combination with Piperazine.
Teneligliptin The therapeutic efficacy of Teneligliptin can be decreased when used in combination with Piperazine.
Omarigliptin The therapeutic efficacy of Omarigliptin can be decreased when used in combination with Piperazine.
Carmegliptin The therapeutic efficacy of Carmegliptin can be decreased when used in combination with Piperazine.
Gemigliptin The therapeutic efficacy of Gemigliptin can be decreased when used in combination with Piperazine.
Anagliptin The therapeutic efficacy of Anagliptin can be decreased when used in combination with Piperazine.
Evogliptin The therapeutic efficacy of Evogliptin can be decreased when used in combination with Piperazine.
Sotagliflozin The therapeutic efficacy of Sotagliflozin can be decreased when used in combination with Piperazine.
Balaglitazone The therapeutic efficacy of Balaglitazone can be decreased when used in combination with Piperazine.
Remogliflozin etabonate The therapeutic efficacy of Remogliflozin etabonate can be decreased when used in combination with Piperazine.
Carbutamide The therapeutic efficacy of Carbutamide can be decreased when used in combination with Piperazine.
Guar gum The therapeutic efficacy of Guar gum can be decreased when used in combination with Piperazine.
Metahexamide The therapeutic efficacy of Metahexamide can be decreased when used in combination with Piperazine.
Semaglutide The therapeutic efficacy of Semaglutide can be decreased when used in combination with Piperazine.
Taspoglutide The therapeutic efficacy of Taspoglutide can be decreased when used in combination with Piperazine.
Englitazone The therapeutic efficacy of Englitazone can be decreased when used in combination with Piperazine.
Tirzepatide The therapeutic efficacy of Tirzepatide can be decreased when used in combination with Piperazine.
Gastric inhibitory polypeptide The therapeutic efficacy of Gastric inhibitory polypeptide can be decreased when used in combination with Piperazine.
Cyclosporine The metabolism of Piperazine can be decreased when combined with Cyclosporine.
Cholecalciferol The metabolism of Piperazine can be decreased when combined with Cholecalciferol.
Fluvoxamine The metabolism of Piperazine can be decreased when combined with Fluvoxamine.
Metoprolol The metabolism of Piperazine can be decreased when combined with Metoprolol.
Venlafaxine The metabolism of Piperazine can be decreased when combined with Venlafaxine.
Terfenadine The metabolism of Piperazine can be decreased when combined with Terfenadine.
Clobazam The serum concentration of Piperazine can be increased when it is combined with Clobazam.
Clozapine The serum concentration of Piperazine can be increased when it is combined with Clozapine.
Quinine The metabolism of Piperazine can be decreased when combined with Quinine.

Target Protein

Gamma-aminobutyric acid receptor subunit beta-3 GABRB3

Referensi & Sumber

Synthesis reference: Hong-Xin Li, Jose Guadalupe Santiesteban, Lenore Ann Emig, John Nelson Armor, "Triethylenediamine and piperazine synthesis using zeolite catalysts modified with a silicon-containing compound." U.S. Patent US6084096, issued 0000.

Contoh Produk & Brand

Produk: 8 • International brands: 4
Produk
  • Entacyl Granules
    Powder, for solution • 2 g / pck • Oral • Canada • OTC • Approved
  • Entacyl Granules 2.0gm
    Powder • 2 g / 4 g • Oral • Canada • OTC • Approved
  • Entacyl Susp 0.6gm/5ml
    Suspension • 600 mg / 5 mL • Oral • Canada • OTC • Approved
  • Entacyl Suspension-600mg/5ml
    Suspension • 600 mg / 5 mL • Oral • Canada • OTC • Approved
  • Formule C34
    Liquid • 100 mg / mL • Oral • Canada • OTC • Approved
  • Veriga 125
    Liquid • 110 mg / mL • Oral • Canada • OTC • Approved
  • Vermirex Syr
    Syrup • 110 mg / mL • Oral • Canada • OTC • Approved
  • Versol 100mg
    Liquid • 100 mg / mL • Oral • Canada • Approved
International Brands
  • Antepar
  • Uvilon
  • Vermidol
  • Vermizine

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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