Peringatan Keamanan

Intravenous LD50 values in the mouse and rat were approximately 75 mg/kg and in the cat and dog were 40 to 80 mg/kg. Symptoms of overdosage are extensions of the pharmacologic effects of the drug. Excessive pressor effect, tachycardia, skeletal muscle hyperactivity, and enhanced deep tendon reflexes may be early signs of overdosage.

Doxapram

DB00561

small molecule approved vet_approved

Deskripsi

A central respiratory stimulant with a brief duration of action. (From Martindale, The Extra Pharmocopoeia, 30th ed, p1225)

Struktur Molekul 2D

Berat 378.5072
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

538 Data
Valsartan Doxapram may decrease the antihypertensive activities of Valsartan.
Ramipril Doxapram may decrease the antihypertensive activities of Ramipril.
Esmolol Doxapram may decrease the antihypertensive activities of Esmolol.
Betaxolol Doxapram may decrease the antihypertensive activities of Betaxolol.
Reserpine Doxapram may decrease the antihypertensive activities of Reserpine.
Remikiren Doxapram may decrease the antihypertensive activities of Remikiren.
Torasemide Doxapram may decrease the antihypertensive activities of Torasemide.
Guanadrel Doxapram may decrease the antihypertensive activities of Guanadrel.
Metoprolol Doxapram may decrease the antihypertensive activities of Metoprolol.
Isradipine Doxapram may decrease the antihypertensive activities of Isradipine.
Olmesartan Doxapram may decrease the antihypertensive activities of Olmesartan.
Chlorthalidone Doxapram may decrease the antihypertensive activities of Chlorthalidone.
Nitroprusside Doxapram may decrease the antihypertensive activities of Nitroprusside.
Atenolol Doxapram may decrease the antihypertensive activities of Atenolol.
Diltiazem Doxapram may decrease the antihypertensive activities of Diltiazem.
Minoxidil Doxapram may decrease the antihypertensive activities of Minoxidil.
Timolol Doxapram may decrease the antihypertensive activities of Timolol.
Treprostinil Doxapram may decrease the antihypertensive activities of Treprostinil.
Amlodipine Doxapram may decrease the antihypertensive activities of Amlodipine.
Nimodipine Doxapram may decrease the antihypertensive activities of Nimodipine.
Nisoldipine Doxapram may decrease the antihypertensive activities of Nisoldipine.
Bendroflumethiazide Doxapram may decrease the antihypertensive activities of Bendroflumethiazide.
Prazosin Doxapram may decrease the antihypertensive activities of Prazosin.
Fosinopril Doxapram may decrease the antihypertensive activities of Fosinopril.
Trandolapril Doxapram may decrease the antihypertensive activities of Trandolapril.
Metolazone Doxapram may decrease the antihypertensive activities of Metolazone.
Lercanidipine Doxapram may decrease the antihypertensive activities of Lercanidipine.
Benazepril Doxapram may decrease the antihypertensive activities of Benazepril.
Bosentan Doxapram may decrease the antihypertensive activities of Bosentan.
Propranolol Doxapram may decrease the antihypertensive activities of Propranolol.
Enalapril Doxapram may decrease the antihypertensive activities of Enalapril.
Doxazosin Doxapram may decrease the antihypertensive activities of Doxazosin.
Labetalol Doxapram may decrease the antihypertensive activities of Labetalol.
Cyclothiazide Doxapram may decrease the antihypertensive activities of Cyclothiazide.
Bisoprolol Doxapram may decrease the antihypertensive activities of Bisoprolol.
Candoxatril Doxapram may decrease the antihypertensive activities of Candoxatril.
Nicardipine Doxapram may decrease the antihypertensive activities of Nicardipine.
Mecamylamine Doxapram may decrease the antihypertensive activities of Mecamylamine.
Losartan Doxapram may decrease the antihypertensive activities of Losartan.
Moexipril Doxapram may decrease the antihypertensive activities of Moexipril.
Eplerenone Doxapram may decrease the antihypertensive activities of Eplerenone.
Lisinopril Doxapram may decrease the antihypertensive activities of Lisinopril.
Nitroglycerin Doxapram may decrease the antihypertensive activities of Nitroglycerin.
Metyrosine Doxapram may decrease the antihypertensive activities of Metyrosine.
Hydroflumethiazide Doxapram may decrease the antihypertensive activities of Hydroflumethiazide.
Cryptenamine Doxapram may decrease the antihypertensive activities of Cryptenamine.
Perindopril Doxapram may decrease the antihypertensive activities of Perindopril.
Candesartan cilexetil Doxapram may decrease the antihypertensive activities of Candesartan cilexetil.
Fenoldopam Doxapram may decrease the antihypertensive activities of Fenoldopam.
Indapamide Doxapram may decrease the antihypertensive activities of Indapamide.
Tadalafil Doxapram may decrease the antihypertensive activities of Tadalafil.
Alprenolol Doxapram may decrease the antihypertensive activities of Alprenolol.
Eprosartan Doxapram may decrease the antihypertensive activities of Eprosartan.
Chlorothiazide Doxapram may decrease the antihypertensive activities of Chlorothiazide.
Quinapril Doxapram may decrease the antihypertensive activities of Quinapril.
Pindolol Doxapram may decrease the antihypertensive activities of Pindolol.
Telmisartan Doxapram may decrease the antihypertensive activities of Telmisartan.
Methyldopa Doxapram may decrease the antihypertensive activities of Methyldopa.
Hydrochlorothiazide Doxapram may decrease the antihypertensive activities of Hydrochlorothiazide.
Trichlormethiazide Doxapram may decrease the antihypertensive activities of Trichlormethiazide.
Felodipine Doxapram may decrease the antihypertensive activities of Felodipine.
Irbesartan Doxapram may decrease the antihypertensive activities of Irbesartan.
Nitrendipine Doxapram may decrease the antihypertensive activities of Nitrendipine.
Deserpidine Doxapram may decrease the antihypertensive activities of Deserpidine.
Pentolinium Doxapram may decrease the antihypertensive activities of Pentolinium.
Trimethaphan Doxapram may decrease the antihypertensive activities of Trimethaphan.
Diazoxide Doxapram may decrease the antihypertensive activities of Diazoxide.
Carvedilol Doxapram may decrease the antihypertensive activities of Carvedilol.
Bretylium Doxapram may decrease the antihypertensive activities of Bretylium.
Terazosin Doxapram may decrease the antihypertensive activities of Terazosin.
Guanethidine Doxapram may decrease the antihypertensive activities of Guanethidine.
Acebutolol Doxapram may decrease the antihypertensive activities of Acebutolol.
Captopril Doxapram may decrease the antihypertensive activities of Captopril.
Nadolol Doxapram may decrease the antihypertensive activities of Nadolol.
Epoprostenol Doxapram may decrease the antihypertensive activities of Epoprostenol.
Bepridil Doxapram may decrease the antihypertensive activities of Bepridil.
Hydralazine Doxapram may decrease the antihypertensive activities of Hydralazine.
Bevantolol Doxapram may decrease the antihypertensive activities of Bevantolol.
Practolol Doxapram may decrease the antihypertensive activities of Practolol.
Polythiazide Doxapram may decrease the antihypertensive activities of Polythiazide.
Cilazapril Doxapram may decrease the antihypertensive activities of Cilazapril.
Saprisartan Doxapram may decrease the antihypertensive activities of Saprisartan.
Spirapril Doxapram may decrease the antihypertensive activities of Spirapril.
Penbutolol Doxapram may decrease the antihypertensive activities of Penbutolol.
Mibefradil Doxapram may decrease the antihypertensive activities of Mibefradil.
Oxprenolol Doxapram may decrease the antihypertensive activities of Oxprenolol.
Dexpropranolol Doxapram may decrease the antihypertensive activities of Dexpropranolol.
Tienilic acid Doxapram may decrease the antihypertensive activities of Tienilic acid.
Debrisoquine Doxapram may decrease the antihypertensive activities of Debrisoquine.
Celiprolol Doxapram may decrease the antihypertensive activities of Celiprolol.
Nebivolol Doxapram may decrease the antihypertensive activities of Nebivolol.
Sitaxentan Doxapram may decrease the antihypertensive activities of Sitaxentan.
Ambrisentan Doxapram may decrease the antihypertensive activities of Ambrisentan.
Diethylnorspermine Doxapram may decrease the antihypertensive activities of Diethylnorspermine.
Nilvadipine Doxapram may decrease the antihypertensive activities of Nilvadipine.
Pinacidil Doxapram may decrease the antihypertensive activities of Pinacidil.
Bupranolol Doxapram may decrease the antihypertensive activities of Bupranolol.
Temocapril Doxapram may decrease the antihypertensive activities of Temocapril.
Riociguat Doxapram may decrease the antihypertensive activities of Riociguat.
Macitentan Doxapram may decrease the antihypertensive activities of Macitentan.

Target Protein

Potassium channel subfamily K member 3 KCNK3
Potassium channel subfamily K member 9 KCNK9

Referensi & Sumber

Synthesis reference: Lunsford, C.D. and Cale, A.D. Jr.; U S . Patent 3,192,230; June 29, 1965; assigned to A.H. Robins Company, Inc.
Artikel (PubMed)
  • PMID: 8251281
    Singh P, Dimitriou V, Mahajan RP, Crossley AW: Double-blind comparison between doxapram and pethidine in the treatment of postanaesthetic shivering. Br J Anaesth. 1993 Nov;71(5):685-8.
  • PMID: 17227289
    Yost CS: A new look at the respiratory stimulant doxapram. CNS Drug Rev. 2006 Fall-Winter;12(3-4):236-49.

Contoh Produk & Brand

Produk: 6 • International brands: 5
Produk
  • Dopram
    Injection • 20 mg/1mL • Intravenous • US • Approved
  • Dopram
    Injection • 20 mg/1mL • Intravenous • US • Approved
  • Dopram Inj 20mg/ml
    Liquid • 20 mg / mL • Intravenous • Canada • Approved
  • Dopram Injectable Liq 20mg/ml
    Liquid • 20 mg / mL • Intravenous • Canada • Approved
  • Doxapram Hydrochloride
    Injection • 20 mg/1mL • Intravenous • US • Generic • Approved
  • Doxapram Hydrochloride
    Injection • 20 mg/1mL • Intravenous • US • Approved
International Brands
  • Caropram — Khandelwal
  • Dai Er Song — Bosen Bio Pharmaceutical
  • Jia Su Lun — Nhwa
  • Stimulex
  • Ze Lun — Jiuxu Pharmaceutical

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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