Peringatan Keamanan

LD50 = 475 mg/kg (oral, rat). Can cause severe gastrointestinal symptoms (nausea, vomiting and diarrhea), bone marrow suppression, renal insufficiency and other hematologic abnormalities (anemia, leucopenia). Severe guanidine intoxication is characterized by nervous hyperirritability, fibrillary tremors and convulsive contractions of muscle, salivation, vomiting, diarrhea, hypoglycemia, and circulatory disturbances.

Guanidine

DB00536

small molecule approved

Deskripsi

A strong organic base existing primarily as guanidium ions at physiological pH. It is found in the urine as a normal product of protein metabolism. It is also used in laboratory research as a protein denaturant. (From Martindale, the Extra Pharmacopoeia, 30th ed and Merck Index, 12th ed) It is also used in the treatment of myasthenia and as a fluorescent probe in HPLC.

Struktur Molekul 2D

Berat 59.0705
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 7-8 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Rapidly absorbed and distributed

Metabolisme

Not metabolized.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

151 Data
Succinic acid The excretion of Succinic acid can be decreased when combined with Guanidine.
Citrulline The excretion of Citrulline can be decreased when combined with Guanidine.
Pravastatin The excretion of Pravastatin can be decreased when combined with Guanidine.
Oseltamivir The excretion of Oseltamivir can be decreased when combined with Guanidine.
Cefotiam The excretion of Cefotiam can be decreased when combined with Guanidine.
Conjugated estrogens The excretion of Conjugated estrogens can be decreased when combined with Guanidine.
Tenofovir disoproxil The excretion of Tenofovir disoproxil can be decreased when combined with Guanidine.
Piperacillin The excretion of Piperacillin can be decreased when combined with Guanidine.
Indomethacin The excretion of Indomethacin can be decreased when combined with Guanidine.
Aminohippuric acid The excretion of Aminohippuric acid can be decreased when combined with Guanidine.
Trifluridine The excretion of Trifluridine can be decreased when combined with Guanidine.
Allopurinol The excretion of Allopurinol can be decreased when combined with Guanidine.
Zidovudine The excretion of Zidovudine can be decreased when combined with Guanidine.
Cefdinir The excretion of Cefdinir can be decreased when combined with Guanidine.
Methotrexate The excretion of Methotrexate can be decreased when combined with Guanidine.
Valaciclovir The excretion of Valaciclovir can be decreased when combined with Guanidine.
Levocarnitine The excretion of Levocarnitine can be decreased when combined with Guanidine.
Leucovorin The excretion of Leucovorin can be decreased when combined with Guanidine.
Fluorescein The excretion of Fluorescein can be decreased when combined with Guanidine.
Hydrocortisone The excretion of Hydrocortisone can be decreased when combined with Guanidine.
Tetracycline The excretion of Tetracycline can be decreased when combined with Guanidine.
Estradiol The excretion of Estradiol can be decreased when combined with Guanidine.
Cefaclor The excretion of Cefaclor can be decreased when combined with Guanidine.
Quinapril The excretion of Quinapril can be decreased when combined with Guanidine.
Bumetanide The excretion of Bumetanide can be decreased when combined with Guanidine.
Dinoprostone The excretion of Dinoprostone can be decreased when combined with Guanidine.
Famotidine The excretion of Famotidine can be decreased when combined with Guanidine.
Fexofenadine The excretion of Fexofenadine can be decreased when combined with Guanidine.
Benzylpenicillin The excretion of Benzylpenicillin can be decreased when combined with Guanidine.
Rosuvastatin The excretion of Rosuvastatin can be decreased when combined with Guanidine.
Captopril The excretion of Captopril can be decreased when combined with Guanidine.
Sitagliptin The excretion of Sitagliptin can be decreased when combined with Guanidine.
Cefazolin The excretion of Cefazolin can be decreased when combined with Guanidine.
Ceftizoxime The excretion of Ceftizoxime can be decreased when combined with Guanidine.
Cefacetrile The excretion of Cefacetrile can be decreased when combined with Guanidine.
Ceftibuten The excretion of Ceftibuten can be decreased when combined with Guanidine.
Tazobactam The excretion of Tazobactam can be decreased when combined with Guanidine.
Cyclic adenosine monophosphate The excretion of Cyclic adenosine monophosphate can be decreased when combined with Guanidine.
Cholic Acid The excretion of Cholic Acid can be decreased when combined with Guanidine.
Glutaric Acid The excretion of Glutaric Acid can be decreased when combined with Guanidine.
Oxalic Acid The excretion of Oxalic Acid can be decreased when combined with Guanidine.
Taurocholic acid The excretion of Taurocholic acid can be decreased when combined with Guanidine.
Doripenem The excretion of Doripenem can be decreased when combined with Guanidine.
Saxagliptin The excretion of Saxagliptin can be decreased when combined with Guanidine.
Ellagic acid The excretion of Ellagic acid can be decreased when combined with Guanidine.
Cefaloridine The excretion of Cefaloridine can be decreased when combined with Guanidine.
Avibactam The excretion of Avibactam can be decreased when combined with Guanidine.
Eluxadoline The excretion of Eluxadoline can be decreased when combined with Guanidine.
Silibinin The excretion of Silibinin can be decreased when combined with Guanidine.
Tenofovir alafenamide The excretion of Tenofovir alafenamide can be decreased when combined with Guanidine.
Tenofovir The excretion of Tenofovir can be decreased when combined with Guanidine.
Hydrochlorothiazide The excretion of Hydrochlorothiazide can be decreased when combined with Guanidine.
Dexamethasone The excretion of Dexamethasone can be decreased when combined with Guanidine.
Cephalexin The excretion of Cephalexin can be decreased when combined with Guanidine.
Acyclovir The excretion of Acyclovir can be decreased when combined with Guanidine.
Relebactam The excretion of Relebactam can be decreased when combined with Guanidine.
Cimetidine The excretion of Cimetidine can be decreased when combined with Guanidine.
Oxytetracycline The excretion of Oxytetracycline can be decreased when combined with Guanidine.
Polythiazide The excretion of Polythiazide can be decreased when combined with Guanidine.
Prednisolone phosphate The excretion of Prednisolone phosphate can be decreased when combined with Guanidine.
Dexamethasone acetate The excretion of Dexamethasone acetate can be decreased when combined with Guanidine.
Tipiracil The excretion of Tipiracil can be decreased when combined with Guanidine.
Varenicline The excretion of Varenicline can be decreased when combined with Guanidine.
Prazosin The serum concentration of Prazosin can be increased when it is combined with Guanidine.
Linagliptin The serum concentration of Linagliptin can be increased when it is combined with Guanidine.
Choline salicylate The serum concentration of Choline salicylate can be increased when it is combined with Guanidine.
Choline The serum concentration of Choline can be increased when it is combined with Guanidine.
Metformin The serum concentration of Metformin can be increased when it is combined with Guanidine.
Norepinephrine The serum concentration of Norepinephrine can be increased when it is combined with Guanidine.
Solriamfetol The serum concentration of Solriamfetol can be increased when it is combined with Guanidine.
Reserpine The serum concentration of Reserpine can be increased when it is combined with Guanidine.
Pramipexole The serum concentration of Pramipexole can be increased when it is combined with Guanidine.
Epinephrine The serum concentration of Epinephrine can be increased when it is combined with Guanidine.
Lamivudine The serum concentration of Lamivudine can be increased when it is combined with Guanidine.
Amantadine The serum concentration of Amantadine can be increased when it is combined with Guanidine.
Dopamine The serum concentration of Dopamine can be increased when it is combined with Guanidine.
Memantine The serum concentration of Memantine can be increased when it is combined with Guanidine.
Histamine The serum concentration of Histamine can be increased when it is combined with Guanidine.
Agmatine The serum concentration of Agmatine can be increased when it is combined with Guanidine.
Nafamostat The serum concentration of Nafamostat can be increased when it is combined with Guanidine.
Pemetrexed Guanidine may decrease the excretion rate of Pemetrexed which could result in a higher serum level.
Mercaptopurine The excretion of Mercaptopurine can be decreased when combined with Guanidine.
Valproic acid The excretion of Valproic acid can be decreased when combined with Guanidine.
Emtricitabine The excretion of Emtricitabine can be decreased when combined with Guanidine.
Ganciclovir The excretion of Ganciclovir can be decreased when combined with Guanidine.
Levofloxacin The excretion of Levofloxacin can be decreased when combined with Guanidine.
Nadolol The excretion of Nadolol can be decreased when combined with Guanidine.
Cefradine The excretion of Cefradine can be decreased when combined with Guanidine.
Estrone sulfate The excretion of Estrone sulfate can be decreased when combined with Guanidine.
N-methylnicotinamide The excretion of N-methylnicotinamide can be decreased when combined with Guanidine.
Procainamide The excretion of Procainamide can be decreased when combined with Guanidine.
Topotecan The excretion of Topotecan can be decreased when combined with Guanidine.
Abemaciclib The excretion of Abemaciclib can be decreased when combined with Guanidine.
Baricitinib The serum concentration of Baricitinib can be increased when it is combined with Guanidine.
Pyrimethamine The excretion of Guanidine can be decreased when combined with Pyrimethamine.
Ciprofloxacin The excretion of Guanidine can be decreased when combined with Ciprofloxacin.
Flecainide The excretion of Flecainide can be decreased when combined with Guanidine.
Lofexidine The excretion of Guanidine can be decreased when combined with Lofexidine.
Tafenoquine The excretion of Guanidine can be decreased when combined with Tafenoquine.
Tucatinib The excretion of Guanidine can be decreased when combined with Tucatinib.

Target Protein

Aldehyde dehydrogenase, mitochondrial ALDH2
Ribonuclease pancreatic RNASE1
DNA
Disks large homolog 4 DLG4
Endolysin E
Guanidinoacetate N-methyltransferase GAMT
Arginase rocF

Referensi & Sumber

Synthesis reference: Helmut Hoffmann, Carlhans Suling, "Process for the production of guanidine salts of aliphatic mercaptosulphonic acids." U.S. Patent US3956368, issued November, 1954.

Contoh Produk & Brand

Produk: 1 • International brands: 0
Produk
  • Guanidine hydrochloride
    Tablet • 125 mg/1 • Oral • US • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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