Peringatan Keamanan

Subcutaneous LD50 in rat is 27 mg/kg. Symptoms of overdose include convulsions, hypoxia, acidosis, bradycardia, arrhythmias and cardiac arrest.

Cinchocaine

DB00527

small molecule approved vet_approved

Deskripsi

A local anesthetic of the amide type now generally used for surface anesthesia. It is one of the most potent and toxic of the long-acting local anesthetics and its parenteral use is restricted to spinal anesthesia. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1006)

Struktur Molekul 2D

Berat 343.4632
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

In general, ionized forms (salts) of local anesthetics are not readily absorbed through intact skin. However, both nonionized (bases) and ionized forms of local anesthetics are readily absorbed through traumatized or abraded skin into the systemic circulation.

Metabolisme

Primarily hepatic.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1784 Data
Buprenorphine Cinchocaine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Cinchocaine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Cinchocaine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Cinchocaine.
Hydrocodone Cinchocaine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Cinchocaine.
Magnesium sulfate The therapeutic efficacy of Cinchocaine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Cinchocaine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Cinchocaine may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Cinchocaine.
Mirtazapine Cinchocaine may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Cinchocaine.
Orphenadrine Cinchocaine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Cinchocaine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Cinchocaine.
Pramipexole Cinchocaine may increase the sedative activities of Pramipexole.
Ropinirole Cinchocaine may increase the sedative activities of Ropinirole.
Rotigotine Cinchocaine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Cinchocaine.
Sodium oxybate Cinchocaine may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Cinchocaine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Cinchocaine.
Thalidomide Cinchocaine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Cinchocaine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Hyaluronidase (ovine) Hyaluronidase (ovine) can cause an increase in the absorption of Cinchocaine resulting in an increased serum concentration and potentially a worsening of adverse effects.
Hyaluronidase (human recombinant) Hyaluronidase (human recombinant) can cause an increase in the absorption of Cinchocaine resulting in an increased serum concentration and potentially a worsening of adverse effects.
Hyaluronidase Hyaluronidase can cause an increase in the absorption of Cinchocaine resulting in an increased serum concentration and potentially a worsening of adverse effects.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Cinchocaine.
Dipyridamole The therapeutic efficacy of Cinchocaine can be decreased when used in combination with Dipyridamole.
Irinotecan The risk or severity of methemoglobinemia can be increased when Irinotecan is combined with Cinchocaine.
Ephedrine Cinchocaine may increase the neuromuscular blocking activities of Ephedrine.
Bambuterol Cinchocaine may increase the neuromuscular blocking activities of Bambuterol.
Clevidipine Cinchocaine may increase the neuromuscular blocking activities of Clevidipine.
Sar9, Met (O2)11-Substance P Cinchocaine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Mirabegron Cinchocaine may increase the neuromuscular blocking activities of Mirabegron.
Moxisylyte Cinchocaine may increase the neuromuscular blocking activities of Moxisylyte.
Propacetamol Cinchocaine may increase the neuromuscular blocking activities of Propacetamol.
Procaine The risk or severity of methemoglobinemia can be increased when Cinchocaine is combined with Procaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Cinchocaine is combined with Cocaine.
Trimethaphan Cinchocaine may increase the neuromuscular blocking activities of Trimethaphan.
Doxacurium Cinchocaine may increase the neuromuscular blocking activities of Doxacurium.
Chloroprocaine The risk or severity of adverse effects can be increased when Cinchocaine is combined with Chloroprocaine.
Tubocurarine Cinchocaine may increase the neuromuscular blocking activities of Tubocurarine.
Aclidinium Cinchocaine may increase the neuromuscular blocking activities of Aclidinium.
Butyrylthiocholine Cinchocaine may increase the neuromuscular blocking activities of Butyrylthiocholine.
Oxybuprocaine The risk or severity of methemoglobinemia can be increased when Cinchocaine is combined with Oxybuprocaine.
Benzonatate Cinchocaine may increase the neuromuscular blocking activities of Benzonatate.
Succinylcholine The metabolism of Succinylcholine can be decreased when combined with Cinchocaine.
Ethanol Cinchocaine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Cinchocaine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Cinchocaine.
Paroxetine The risk or severity of adverse effects can be increased when Cinchocaine is combined with Paroxetine.
Escitalopram The risk or severity of adverse effects can be increased when Cinchocaine is combined with Escitalopram.
Fluvoxamine The risk or severity of adverse effects can be increased when Cinchocaine is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Cinchocaine is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Cinchocaine is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Cinchocaine is combined with Trazodone.
Sertraline The risk or severity of adverse effects can be increased when Cinchocaine is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Cinchocaine is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Cinchocaine is combined with Nefazodone.
Zimelidine The risk or severity of adverse effects can be increased when Cinchocaine is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Cinchocaine is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Cinchocaine is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Cinchocaine is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Cinchocaine is combined with Seproxetine.
Indalpine The risk or severity of adverse effects can be increased when Cinchocaine is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Cinchocaine is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Cinchocaine is combined with Alaproclate.
Technetium Tc-99m tilmanocept Cinchocaine may decrease effectiveness of Technetium Tc-99m tilmanocept as a diagnostic agent.
Mecamylamine The therapeutic efficacy of Mecamylamine can be decreased when used in combination with Cinchocaine.
Amantadine The therapeutic efficacy of Amantadine can be decreased when used in combination with Cinchocaine.
Pentolinium The therapeutic efficacy of Pentolinium can be decreased when used in combination with Cinchocaine.
Fenoterol The therapeutic efficacy of Fenoterol can be decreased when used in combination with Cinchocaine.
Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione The therapeutic efficacy of Dihydro-2-thioxo-5-((5-(2-(trifluoromethyl)phenyl)-2-furanyl)methyl)-4,6(1H,5H)-pyrimidinedione can be decreased when used in combination with Cinchocaine.
Agmatine The therapeutic efficacy of Agmatine can be decreased when used in combination with Cinchocaine.
Esmolol Cinchocaine may increase the bradycardic activities of Esmolol.
Betaxolol Cinchocaine may increase the bradycardic activities of Betaxolol.
Metoprolol Cinchocaine may increase the bradycardic activities of Metoprolol.
Atenolol Cinchocaine may increase the bradycardic activities of Atenolol.
Timolol Cinchocaine may increase the bradycardic activities of Timolol.
Sotalol Cinchocaine may increase the bradycardic activities of Sotalol.
Propranolol Cinchocaine may increase the bradycardic activities of Propranolol.
Labetalol Cinchocaine may increase the bradycardic activities of Labetalol.
Bisoprolol Cinchocaine may increase the bradycardic activities of Bisoprolol.
Alprenolol Cinchocaine may increase the bradycardic activities of Alprenolol.
Pindolol Cinchocaine may increase the bradycardic activities of Pindolol.
Carvedilol Cinchocaine may increase the bradycardic activities of Carvedilol.
Propafenone Cinchocaine may increase the bradycardic activities of Propafenone.
Acebutolol Cinchocaine may increase the bradycardic activities of Acebutolol.
Nadolol Cinchocaine may increase the bradycardic activities of Nadolol.
Bevantolol Cinchocaine may increase the bradycardic activities of Bevantolol.
Practolol Cinchocaine may increase the bradycardic activities of Practolol.
Penbutolol Cinchocaine may increase the bradycardic activities of Penbutolol.
Oxprenolol Cinchocaine may increase the bradycardic activities of Oxprenolol.
Dexpropranolol Cinchocaine may increase the bradycardic activities of Dexpropranolol.
Celiprolol Cinchocaine may increase the bradycardic activities of Celiprolol.
Nebivolol Cinchocaine may increase the bradycardic activities of Nebivolol.
Bufuralol Cinchocaine may increase the bradycardic activities of Bufuralol.
Bopindolol Cinchocaine may increase the bradycardic activities of Bopindolol.
Bupranolol Cinchocaine may increase the bradycardic activities of Bupranolol.

Target Protein

Sodium channel protein type 5 subunit alpha SCN5A
Sodium channel protein type 10 subunit alpha SCN10A
Calmodulin CALM1

Referensi & Sumber

Artikel (PubMed)
  • PMID: 15910814
    Abdel-Ghani NT, Youssef AF, Awady MA: Cinchocaine hydrochloride determination by atomic absorption spectrometry and spectrophotometry. Farmaco. 2005 May;60(5):419-24.
  • PMID: 16612626
    Souto-Padron T, Lima AP, Ribeiro Rde O: Effects of dibucaine on the endocytic/exocytic pathways in Trypanosoma cruzi. Parasitol Res. 2006 Sep;99(4):317-20. Epub 2006 Apr 13.
  • PMID: 16459486
    Nounou MM, El-Khordagui LK, Khalafallah N: Effect of various formulation variables on the encapsulation and stability of dibucaine base in multilamellar vesicles. Acta Pol Pharm. 2005 Sep-Oct;62(5):369-79.

Contoh Produk & Brand

Produk: 31 • International brands: 3
Produk
  • CVS Hemorrhoidal Topical Analgesic
    Ointment • 10 mg/1g • Topical • US • OTC
  • Dibucaine
    Cream • 10 mg/1g • Topical • US • OTC
  • Dibucaine
    Ointment • 1 g/100g • Topical • US • OTC
  • Dibucaine
    Ointment • 1 g/100g • Topical • US • OTC
  • Dibucaine
    Ointment • 0.28 g/28g • Topical • US • OTC
  • Dibucaine
    Ointment • 0.28 g/28g • Topical • US • OTC
  • Dibucaine
    Ointment • 1 g/100g • Topical • US • OTC
  • Dibucaine
    Ointment • 0.01 g/1g • Topical • US • OTC
Menampilkan 8 dari 31 produk.
International Brands
  • Cincain
  • Nupercaine
  • Sovcaine

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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