Anisotropine methylbromide

DB00517

small molecule approved

Deskripsi

Anisotropine methylbromide is a quaternary ammonium compound. Its use as treatment adjunct in peptic ulcer has been replaced by the use of more effective agents. Depending on the dose, anisotropine methylbromide may reduce the motility and secretory activity of the gastrointestinal system, and the tone of the ureter and urinary bladder and may have a slight relaxant action on the bile ducts and gallbladder. In general, smaller doses of anisotropine methylbromide inhibit salivary and bronchial secretions, sweating, and accommodation; cause dilatation of the pupil; and increase the heart rate. Larger doses are required to decrease motility of the gastrointestinal and urinary tracts and to inhibit gastric acid secretion.

Struktur Molekul 2D

Berat 362.345
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Not Known
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Gastrointestinal absorption is poor and irregular. Total absorption after an oral dose is about 10 to 25%.

Metabolisme

Hepatic, by enzymatic hydrolysis.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

516 Data
Aclidinium The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Aclidinium.
Mianserin Mianserin may increase the anticholinergic activities of Anisotropine methylbromide.
Mirabegron The risk or severity of urinary retention can be increased when Anisotropine methylbromide is combined with Mirabegron.
Potassium chloride The risk or severity of gastrointestinal ulceration can be increased when Anisotropine methylbromide is combined with Potassium chloride.
Pramlintide The risk or severity of reduced gastrointestinal motility can be increased when Pramlintide is combined with Anisotropine methylbromide.
Secretin porcine The therapeutic efficacy of Secretin porcine can be decreased when used in combination with Anisotropine methylbromide.
Tiotropium The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Tiotropium.
Topiramate The risk or severity of hyperthermia and oligohydrosis can be increased when Anisotropine methylbromide is combined with Topiramate.
Umeclidinium The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Umeclidinium.
Glycopyrronium The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Glycopyrronium.
Botulinum toxin type A The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Botulinum toxin type A.
Glucagon Anisotropine methylbromide may increase the gastrointestinal motility reducing activities of Glucagon.
Sulpiride Anisotropine methylbromide may increase the anticholinergic activities of Sulpiride.
Botulinum toxin type B The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Botulinum toxin type B.
Eluxadoline The risk or severity of constipation can be increased when Anisotropine methylbromide is combined with Eluxadoline.
Ramosetron The risk or severity of constipation can be increased when Anisotropine methylbromide is combined with Ramosetron.
Naltrexone The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Naltrexone.
Bezitramide The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Bezitramide.
Tramadol The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Tramadol.
Morphine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Morphine.
Codeine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Codeine.
Hydromorphone The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Hydromorphone.
Methadone The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Methadone.
Meperidine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Meperidine.
Oxycodone The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Oxycodone.
Butorphanol The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Butorphanol.
Dextropropoxyphene The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Dextropropoxyphene.
Pentazocine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Pentazocine.
Sufentanil The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Sufentanil.
Alfentanil The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Alfentanil.
Fentanyl The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Fentanyl.
Nalbuphine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Nalbuphine.
Levorphanol The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Levorphanol.
Remifentanil The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Remifentanil.
Buprenorphine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Buprenorphine.
Hydrocodone The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Hydrocodone.
Diphenoxylate The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Diphenoxylate.
Oxymorphone The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Oxymorphone.
Dezocine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Dezocine.
Levacetylmethadol The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Levacetylmethadol.
Methadyl acetate The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Methadyl acetate.
Dihydroetorphine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Dihydroetorphine.
Diamorphine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Diamorphine.
Ethylmorphine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Ethylmorphine.
Etorphine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Etorphine.
Dextromoramide The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Dextromoramide.
Desomorphine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Desomorphine.
Carfentanil The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Carfentanil.
Dihydrocodeine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Dihydrocodeine.
Alphacetylmethadol The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Alphacetylmethadol.
Dihydromorphine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Dihydromorphine.
Tapentadol The risk or severity of urinary retention and constipation can be increased when Anisotropine methylbromide is combined with Tapentadol.
Ketobemidone The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Ketobemidone.
DPDPE The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with DPDPE.
Lofentanil The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Lofentanil.
Opium The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Opium.
Normethadone The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Normethadone.
Piritramide The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Piritramide.
Alphaprodine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Alphaprodine.
Nicomorphine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Nicomorphine.
Meptazinol The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Meptazinol.
Phenoperidine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Phenoperidine.
Phenazocine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Phenazocine.
Tilidine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Tilidine.
Carfentanil, C-11 The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Carfentanil, C-11.
Benzhydrocodone The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Benzhydrocodone.
Naloxegol The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Naloxegol.
Trospium The risk or severity of adverse effects can be increased when Trospium is combined with Anisotropine methylbromide.
Oxyphenonium The risk or severity of adverse effects can be increased when Oxyphenonium is combined with Anisotropine methylbromide.
Benzatropine The risk or severity of adverse effects can be increased when Benzatropine is combined with Anisotropine methylbromide.
Disopyramide The risk or severity of adverse effects can be increased when Disopyramide is combined with Anisotropine methylbromide.
Metixene The risk or severity of adverse effects can be increased when Metixene is combined with Anisotropine methylbromide.
Terfenadine The risk or severity of adverse effects can be increased when Terfenadine is combined with Anisotropine methylbromide.
Buclizine The risk or severity of adverse effects can be increased when Buclizine is combined with Anisotropine methylbromide.
Trihexyphenidyl The risk or severity of adverse effects can be increased when Trihexyphenidyl is combined with Anisotropine methylbromide.
Oxyphencyclimine The risk or severity of adverse effects can be increased when Oxyphencyclimine is combined with Anisotropine methylbromide.
Procyclidine The risk or severity of adverse effects can be increased when Procyclidine is combined with Anisotropine methylbromide.
Hyoscyamine The risk or severity of adverse effects can be increased when Hyoscyamine is combined with Anisotropine methylbromide.
Methscopolamine bromide The risk or severity of adverse effects can be increased when Methscopolamine bromide is combined with Anisotropine methylbromide.
Darifenacin The risk or severity of adverse effects can be increased when Darifenacin is combined with Anisotropine methylbromide.
Tridihexethyl The risk or severity of adverse effects can be increased when Tridihexethyl is combined with Anisotropine methylbromide.
Atropine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Atropine.
Nicardipine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Nicardipine.
Mecamylamine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Mecamylamine.
Pirenzepine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Pirenzepine.
Homatropine methylbromide The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Homatropine methylbromide.
Benzquinamide The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Benzquinamide.
Propantheline The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Propantheline.
Dicyclomine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Dicyclomine.
Tropicamide The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Tropicamide.
Cocaine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Cocaine.
Quinidine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Quinidine.
Amantadine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Amantadine.
Methantheline The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Methantheline.
Cycrimine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Cycrimine.
Cyclopentolate The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Cyclopentolate.
Tolterodine The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Tolterodine.
Oxybutynin The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Oxybutynin.
Pentolinium The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Pentolinium.
Trimethaphan The risk or severity of adverse effects can be increased when Anisotropine methylbromide is combined with Trimethaphan.

Target Protein

Muscarinic acetylcholine receptor M5 CHRM5
Muscarinic acetylcholine receptor M1 CHRM1
Muscarinic acetylcholine receptor M2 CHRM2
Muscarinic acetylcholine receptor M3 CHRM3

Referensi & Sumber

Synthesis reference: Weiner, N. and Gordon, S.M.; US. Patent 2,962,499; November 29,1960; assigned to Endo Laboratories, Inc.

Contoh Produk & Brand

Produk: 0 • International brands: 3
International Brands
  • Endovalpin
  • Lytispasm
  • Valpin — Endo

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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