Peringatan Keamanan

A few cases of acute overdosage with intravenous administration have been reported. The effects have ranged from no reaction to transient hypotension to severe acute renal failure leading to death. The intravenous and oral LD50 were 3.0 and 12.0 g/kg respectively in the mouse and 3.2 and 16.4 g/kg respectively in the rat. An intravenous infusion dose of 2.3 g/kg was lethal in the dog.

Aminocaproic acid

DB00513

small molecule approved investigational

Deskripsi

An antifibrinolytic agent that acts by inhibiting plasminogen activators which have fibrinolytic properties.

Struktur Molekul 2D

Berat 131.1729
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The terminal elimination half-life is approximately 2 hours.
Volume Distribusi * 23.1 ± 6.6 L
Klirens (Clearance) * 169 mL/min

Absorpsi

Absorbed rapidly following oral administration. In adults, oral absorption appears to be a zero-order process with an absorption rate of 5.2 g/hr. The mean lag time in absorption is 10 minutes. After a single oral dose of 5 g, absorption was complete (F=1).

Metabolisme

Sixty-five percent of the dose is recovered in the urine as unchanged drug and 11% of the dose appears as the metabolite adipic acid.

Rute Eliminasi

Renal excretion is the primary route of elimination, whether aminocaproic acid is administered orally or intravenously.

Interaksi Makanan

1 Data
  • 1. Take with or without food. The absorption is unaffected by food.

Interaksi Obat

56 Data
Alpha-1-proteinase inhibitor Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Aminocaproic acid.
Menadione Menadione may increase the thrombogenic activities of Aminocaproic acid.
Tranexamic acid Tranexamic acid may increase the thrombogenic activities of Aminocaproic acid.
Aprotinin Aminocaproic acid may increase the thrombogenic activities of Aprotinin.
Hydrogen peroxide Aminocaproic acid may increase the thrombogenic activities of Hydrogen peroxide.
Aminomethylbenzoic acid Aminocaproic acid may increase the thrombogenic activities of Aminomethylbenzoic acid.
Camostat Aminocaproic acid may increase the thrombogenic activities of Camostat.
Menadione bisulfite Aminocaproic acid may increase the thrombogenic activities of Menadione bisulfite.
Tretinoin The risk or severity of Thrombosis can be increased when Aminocaproic acid is combined with Tretinoin.
Antihemophilic factor, human recombinant The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Antihemophilic factor, human recombinant.
Coagulation factor VIIa Recombinant Human The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Coagulation factor VIIa Recombinant Human.
Coagulation Factor IX (Recombinant) The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Coagulation Factor IX (Recombinant).
Calcium The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Calcium.
Pantothenic acid The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Pantothenic acid.
Formic acid The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Formic acid.
Platelet Activating Factor The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Platelet Activating Factor.
Turoctocog alfa The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Turoctocog alfa.
Fibrinogen human The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Fibrinogen human.
Catridecacog The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Catridecacog.
Antihemophilic factor (recombinant), PEGylated The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Antihemophilic factor (recombinant), PEGylated.
Prothrombin The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Prothrombin.
Factor IX Complex (Human) The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Factor IX Complex (Human).
Susoctocog alfa The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Susoctocog alfa.
Eftrenonacog alfa The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Eftrenonacog alfa.
Rusalatide acetate The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Rusalatide acetate.
Vatreptacog alfa The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Vatreptacog alfa.
Factor XIII (human) The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Factor XIII (human).
Von Willebrand factor human The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Von Willebrand factor human.
Coagulation factor X human The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Coagulation factor X human.
Coagulation factor VII human The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Coagulation factor VII human.
Anti-inhibitor coagulant complex The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Anti-inhibitor coagulant complex.
Coagulation Factor IX Human The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Coagulation Factor IX Human.
Antihemophilic factor human The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Antihemophilic factor human.
Kallidinogenase The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Kallidinogenase.
Trenonacog alfa The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Trenonacog alfa.
Albutrepenonacog alfa The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Albutrepenonacog alfa.
Emicizumab The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Emicizumab.
Nonacog beta pegol The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Nonacog beta pegol.
Moroctocog alfa The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Moroctocog alfa.
Beroctocog alfa The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Beroctocog alfa.
Andexanet alfa The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Andexanet alfa.
Calcium cation The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Calcium cation.
Damoctocog alfa pegol The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Damoctocog alfa pegol.
Turoctocog alfa pegol The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Turoctocog alfa pegol.
Alteplase The therapeutic efficacy of Aminocaproic acid can be decreased when used in combination with Alteplase.
Urokinase The therapeutic efficacy of Aminocaproic acid can be decreased when used in combination with Urokinase.
Reteplase The therapeutic efficacy of Aminocaproic acid can be decreased when used in combination with Reteplase.
Anistreplase The therapeutic efficacy of Aminocaproic acid can be decreased when used in combination with Anistreplase.
Tenecteplase The therapeutic efficacy of Aminocaproic acid can be decreased when used in combination with Tenecteplase.
Streptokinase The therapeutic efficacy of Aminocaproic acid can be decreased when used in combination with Streptokinase.
Lanoteplase The therapeutic efficacy of Aminocaproic acid can be decreased when used in combination with Lanoteplase.
Amediplase The therapeutic efficacy of Aminocaproic acid can be decreased when used in combination with Amediplase.
Saruplase The therapeutic efficacy of Aminocaproic acid can be decreased when used in combination with Saruplase.
Protein S human The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Protein S human.
Rurioctocog alfa pegol The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Rurioctocog alfa pegol.
Etranacogene dezaparvovec The risk or severity of adverse effects can be increased when Aminocaproic acid is combined with Etranacogene dezaparvovec.

Target Protein

Plasminogen PLG
Tissue-type plasminogen activator PLAT
Apolipoprotein(a) LPA

Referensi & Sumber

Synthesis reference: Frantisek Mares, "Process for producing caprolactam from 6-aminocaproic acid." U.S. Patent US3988319, issued August, 1955.

Contoh Produk & Brand

Produk: 105 • International brands: 15
Produk
  • 28tak Gum Care Tooth
    Paste, dentifrice • - • Oral • US • OTC
  • Amicar
    Tablet • 500 mg/1 • Oral • US • Approved
  • Amicar
    Tablet • 500 mg/1 • Oral • US • Approved
  • Amicar
    Tablet • 1000 mg/1 • Oral • US • Approved
  • Amicar
    Solution • 0.25 g/1mL • Oral • US • Approved
  • Amicar
    Tablet • 500 mg/1 • Oral • US • Approved
  • Amicar
    Injection, solution • 250 mg/1mL • Intravenous • US • Approved
  • Amicar
    Solution • 0.25 g/1mL • Oral • US • Approved
Menampilkan 8 dari 105 produk.
International Brands
  • Acepramin — Pannonpharma
  • Amocap — Celon
  • Caproamin — Rottapharm
  • Caprocat — Catalysis
  • Caprolisin — Menarini
  • E-Capro — Edruc
  • Epsicaprom
  • Hemocid — GlaxoSmithKline
  • Inselon — Ying Yuan
  • Ipron — Johnson

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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