Peringatan Keamanan

Oral, mouse: LD50 = 175 mg/kg; Oral, rat: LD50 = 163 mg/kg.

Phenindione

DB00498

small molecule approved investigational

Deskripsi

An indandione that has been used as an anticoagulant. Phenindione has actions similar to warfarin, but it is now rarely employed because of its higher incidence of severe adverse effects. (From Martindale, The Extra Pharmacopoeia, 30th ed, p234)

Struktur Molekul 2D

Berat 222.2387
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 5-10 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Absorbed slowly from the gastrointestinal tract.

Metabolisme

Hepatic.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

1 Data
  • 1. Avoid herbs and supplements with anticoagulant/antiplatelet activity. Examples include ginseng, ginkgo, ginger, and garlic.

Interaksi Obat

1293 Data
Apixaban Apixaban may increase the anticoagulant activities of Phenindione.
Dabigatran etexilate Dabigatran etexilate may increase the anticoagulant activities of Phenindione.
Dasatinib The risk or severity of bleeding and hemorrhage can be increased when Dasatinib is combined with Phenindione.
Deferasirox The risk or severity of gastrointestinal bleeding can be increased when Phenindione is combined with Deferasirox.
Ursodeoxycholic acid The risk or severity of bleeding and bruising can be increased when Phenindione is combined with Ursodeoxycholic acid.
Glycochenodeoxycholic Acid The risk or severity of bleeding and bruising can be increased when Phenindione is combined with Glycochenodeoxycholic Acid.
Cholic Acid The risk or severity of bleeding and bruising can be increased when Phenindione is combined with Cholic Acid.
Glycocholic acid The risk or severity of bleeding and bruising can be increased when Phenindione is combined with Glycocholic acid.
Deoxycholic acid The risk or severity of bleeding and bruising can be increased when Phenindione is combined with Deoxycholic acid.
Taurocholic acid The risk or severity of bleeding and bruising can be increased when Phenindione is combined with Taurocholic acid.
Obeticholic acid The risk or severity of bleeding and bruising can be increased when Phenindione is combined with Obeticholic acid.
Chenodeoxycholic acid The risk or severity of bleeding and bruising can be increased when Phenindione is combined with Chenodeoxycholic acid.
Taurochenodeoxycholic acid The risk or severity of bleeding and bruising can be increased when Phenindione is combined with Taurochenodeoxycholic acid.
Tauroursodeoxycholic acid The risk or severity of bleeding and bruising can be increased when Phenindione is combined with Tauroursodeoxycholic acid.
Bamet-UD2 The risk or severity of bleeding and bruising can be increased when Phenindione is combined with Bamet-UD2.
Dehydrocholic acid The risk or severity of bleeding and bruising can be increased when Phenindione is combined with Dehydrocholic acid.
Hyodeoxycholic Acid The risk or severity of bleeding and bruising can be increased when Phenindione is combined with Hyodeoxycholic Acid.
Edoxaban The risk or severity of bleeding can be increased when Edoxaban is combined with Phenindione.
Ibrutinib The risk or severity of bleeding and hemorrhage can be increased when Ibrutinib is combined with Phenindione.
Obinutuzumab The risk or severity of bleeding and hemorrhage can be increased when Phenindione is combined with Obinutuzumab.
Rivaroxaban Phenindione may increase the anticoagulant activities of Rivaroxaban.
Sugammadex The risk or severity of bleeding and hemorrhage can be increased when Phenindione is combined with Sugammadex.
Tibolone Tibolone may increase the anticoagulant activities of Phenindione.
Tipranavir The risk or severity of bleeding and hemorrhage can be increased when Tipranavir is combined with Phenindione.
Urokinase Urokinase may increase the anticoagulant activities of Phenindione.
Vitamin E Vitamin E may increase the anticoagulant activities of Phenindione.
Vorapaxar The risk or severity of bleeding and hemorrhage can be increased when Vorapaxar is combined with Phenindione.
Gemcitabine The therapeutic efficacy of Phenindione can be increased when used in combination with Gemcitabine.
Flunisolide Flunisolide may increase the anticoagulant activities of Phenindione.
Beclomethasone dipropionate Beclomethasone dipropionate may increase the anticoagulant activities of Phenindione.
Betamethasone Betamethasone may increase the anticoagulant activities of Phenindione.
Fluticasone propionate Fluticasone propionate may increase the anticoagulant activities of Phenindione.
Fluocinolone acetonide Fluocinolone acetonide may increase the anticoagulant activities of Phenindione.
Prednisone Prednisone may increase the anticoagulant activities of Phenindione.
Fludrocortisone Fludrocortisone may increase the anticoagulant activities of Phenindione.
Hydrocortisone Hydrocortisone may increase the anticoagulant activities of Phenindione.
Prednisolone Prednisolone may increase the anticoagulant activities of Phenindione.
Methylprednisolone Methylprednisolone may increase the anticoagulant activities of Phenindione.
Trilostane Trilostane may increase the anticoagulant activities of Phenindione.
Budesonide Budesonide may increase the anticoagulant activities of Phenindione.
Dexamethasone Dexamethasone may increase the anticoagulant activities of Phenindione.
Corticotropin Corticotropin may increase the anticoagulant activities of Phenindione.
Cortisone acetate Cortisone acetate may increase the anticoagulant activities of Phenindione.
Paramethasone Paramethasone may increase the anticoagulant activities of Phenindione.
Ciclesonide Ciclesonide may increase the anticoagulant activities of Phenindione.
Aldosterone Aldosterone may increase the anticoagulant activities of Phenindione.
Fluticasone furoate Fluticasone furoate may increase the anticoagulant activities of Phenindione.
Fluprednidene Fluprednidene may increase the anticoagulant activities of Phenindione.
Tixocortol Tixocortol may increase the anticoagulant activities of Phenindione.
Fluprednisolone Fluprednisolone may increase the anticoagulant activities of Phenindione.
Meprednisone Meprednisone may increase the anticoagulant activities of Phenindione.
Dexamethasone isonicotinate Dexamethasone isonicotinate may increase the anticoagulant activities of Phenindione.
Melengestrol Melengestrol may increase the anticoagulant activities of Phenindione.
Deflazacort Deflazacort may increase the anticoagulant activities of Phenindione.
Cortivazol Cortivazol may increase the anticoagulant activities of Phenindione.
Prednylidene Prednylidene may increase the anticoagulant activities of Phenindione.
Fluocortin Fluocortin may increase the anticoagulant activities of Phenindione.
Fluperolone Fluperolone may increase the anticoagulant activities of Phenindione.
Cloprednol Cloprednol may increase the anticoagulant activities of Phenindione.
Fluclorolone Fluclorolone may increase the anticoagulant activities of Phenindione.
Fluticasone Fluticasone may increase the anticoagulant activities of Phenindione.
Mometasone furoate Mometasone furoate may increase the anticoagulant activities of Phenindione.
Hydrocortisone acetate Hydrocortisone acetate may increase the anticoagulant activities of Phenindione.
Hydrocortisone cypionate Hydrocortisone cypionate may increase the anticoagulant activities of Phenindione.
Hydrocortisone succinate Hydrocortisone succinate may increase the anticoagulant activities of Phenindione.
Prednisolone phosphate Prednisolone phosphate may increase the anticoagulant activities of Phenindione.
Prednisolone hemisuccinate Prednisolone hemisuccinate may increase the anticoagulant activities of Phenindione.
Methylprednisolone hemisuccinate Methylprednisolone hemisuccinate may increase the anticoagulant activities of Phenindione.
Prednisone acetate Prednisone acetate may increase the anticoagulant activities of Phenindione.
Clocortolone acetate Clocortolone acetate may increase the anticoagulant activities of Phenindione.
Melengestrol acetate Melengestrol acetate may increase the anticoagulant activities of Phenindione.
Betamethasone phosphate Betamethasone phosphate may increase the anticoagulant activities of Phenindione.
Cortisone Cortisone may increase the anticoagulant activities of Phenindione.
Clobetasol propionate Clobetasol propionate may increase the anticoagulant activities of Phenindione.
Fluocinonide Fluocinonide may increase the anticoagulant activities of Phenindione.
Hydrocortisone butyrate Hydrocortisone butyrate may increase the anticoagulant activities of Phenindione.
Desoximetasone Desoximetasone may increase the anticoagulant activities of Phenindione.
Mometasone Mometasone may increase the anticoagulant activities of Phenindione.
Fluocortolone Fluocortolone may increase the anticoagulant activities of Phenindione.
Prednisolone acetate Prednisolone acetate may increase the anticoagulant activities of Phenindione.
Fluorometholone Fluorometholone may increase the anticoagulant activities of Phenindione.
Difluocortolone Difluocortolone may increase the anticoagulant activities of Phenindione.
Flumethasone Flumethasone may increase the anticoagulant activities of Phenindione.
Methylprednisolone aceponate Methylprednisolone aceponate may increase the anticoagulant activities of Phenindione.
Erlotinib The serum concentration of Phenindione can be increased when it is combined with Erlotinib.
Acetaminophen Acetaminophen may increase the anticoagulant activities of Phenindione.
Allopurinol The risk or severity of bleeding can be increased when Allopurinol is combined with Phenindione.
Azathioprine The therapeutic efficacy of Phenindione can be decreased when used in combination with Azathioprine.
Chloral hydrate The protein binding of Phenindione can be decreased when combined with Chloral hydrate.
Methylphenidate The metabolism of Phenindione can be decreased when combined with Methylphenidate.
Dexmethylphenidate The metabolism of Phenindione can be decreased when combined with Dexmethylphenidate.
Disulfiram Disulfiram may increase the anticoagulant activities of Phenindione.
Etacrynic acid The protein binding of Phenindione can be decreased when combined with Etacrynic acid.
Ethotoin The therapeutic efficacy of Phenindione can be increased when used in combination with Ethotoin.
Etoposide The therapeutic efficacy of Phenindione can be increased when used in combination with Etoposide.
Exenatide Exenatide can cause an increase in the absorption of Phenindione resulting in an increased serum concentration and potentially a worsening of adverse effects.
Gefitinib Gefitinib may increase the anticoagulant activities of Phenindione.
Ginkgo biloba Ginkgo biloba may increase the anticoagulant activities of Phenindione.
Glutethimide The therapeutic efficacy of Phenindione can be decreased when used in combination with Glutethimide.
Ifosfamide The risk or severity of bleeding can be increased when Ifosfamide is combined with Phenindione.

Target Protein

Vitamin K epoxide reductase complex subunit 1 VKORC1

Referensi & Sumber

Link

Contoh Produk & Brand

Produk: 0 • International brands: 4
International Brands
  • Dindevan — Sigma
  • Fenindion — Souriree
  • Phenindione — Goldshield
  • Soluthrombine — Cooper

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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