Peringatan Keamanan

Signs of overdose include confusion (severe), decrease in or loss of reflexes, drowsiness (severe), fever, irritability (continuing), low body temperature, poor judgment, shortness of breath or slow or troubled breathing, slow heartbeat, slurred speech, staggering, trouble in sleeping, unusual movements of the eyes, weakness (severe).

Metharbital

DB00463

small molecule withdrawn

Deskripsi

Metharbital is a barbiturate anticonvulsant, similar to phenobarbital, marketed as Gemonil by Abbott Laboratories. It was patented in 1905 by Emil Fischer of Merck.

Struktur Molekul 2D

Berat 198.2191
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1020 Data
Buprenorphine Metharbital may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Metharbital.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Metharbital.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Metharbital.
Hydrocodone Metharbital may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Metharbital.
Magnesium sulfate The therapeutic efficacy of Metharbital can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Metharbital may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Metharbital may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Metharbital.
Mirtazapine Metharbital may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Metharbital.
Orphenadrine Metharbital may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Metharbital may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Metharbital.
Pramipexole Metharbital may increase the sedative activities of Pramipexole.
Ropinirole Metharbital may increase the sedative activities of Ropinirole.
Rotigotine Metharbital may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Metharbital.
Sodium oxybate Metharbital may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Metharbital may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Metharbital.
Thalidomide Metharbital may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Metharbital may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Secretin porcine The therapeutic efficacy of Secretin porcine can be decreased when used in combination with Metharbital.
Mefloquine The therapeutic efficacy of Metharbital can be decreased when used in combination with Mefloquine.
Mianserin The therapeutic efficacy of Metharbital can be decreased when used in combination with Mianserin.
Orlistat Orlistat can cause a decrease in the absorption of Metharbital resulting in a reduced serum concentration and potentially a decrease in efficacy.
Topotecan Metharbital may increase the excretion rate of Topotecan which could result in a lower serum level and potentially a reduction in efficacy.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Metharbital.
Tetracosactide The risk or severity of liver damage can be increased when Tetracosactide is combined with Metharbital.
Botulinum toxin type A The risk or severity of adverse effects can be increased when Metharbital is combined with Botulinum toxin type A.
Botulinum toxin type B The risk or severity of adverse effects can be increased when Metharbital is combined with Botulinum toxin type B.
Ethanol Metharbital may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Metharbital may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Metharbital.
Fluvoxamine The risk or severity of adverse effects can be increased when Metharbital is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Metharbital is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Metharbital is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Metharbital is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Metharbital is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Metharbital is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Metharbital is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Metharbital is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Metharbital is combined with Escitalopram.
Zimelidine The risk or severity of adverse effects can be increased when Metharbital is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Metharbital is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Metharbital is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Metharbital is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Metharbital is combined with Seproxetine.
Indalpine The risk or severity of adverse effects can be increased when Metharbital is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Metharbital is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Metharbital is combined with Alaproclate.
Naltrexone The risk or severity of adverse effects can be increased when Metharbital is combined with Naltrexone.
Bezitramide The risk or severity of adverse effects can be increased when Metharbital is combined with Bezitramide.
Morphine The risk or severity of adverse effects can be increased when Metharbital is combined with Morphine.
Codeine The risk or severity of adverse effects can be increased when Metharbital is combined with Codeine.
Hydromorphone The risk or severity of adverse effects can be increased when Metharbital is combined with Hydromorphone.
Meperidine The risk or severity of adverse effects can be increased when Metharbital is combined with Meperidine.
Oxycodone The risk or severity of adverse effects can be increased when Metharbital is combined with Oxycodone.
Butorphanol The risk or severity of adverse effects can be increased when Metharbital is combined with Butorphanol.
Dextropropoxyphene The risk or severity of adverse effects can be increased when Metharbital is combined with Dextropropoxyphene.
Pentazocine The risk or severity of adverse effects can be increased when Metharbital is combined with Pentazocine.
Sufentanil The risk or severity of adverse effects can be increased when Metharbital is combined with Sufentanil.
Alfentanil The risk or severity of adverse effects can be increased when Metharbital is combined with Alfentanil.
Fentanyl The risk or severity of adverse effects can be increased when Metharbital is combined with Fentanyl.
Nalbuphine The risk or severity of adverse effects can be increased when Metharbital is combined with Nalbuphine.
Levorphanol The risk or severity of adverse effects can be increased when Metharbital is combined with Levorphanol.
Remifentanil The risk or severity of adverse effects can be increased when Metharbital is combined with Remifentanil.
Diphenoxylate The risk or severity of adverse effects can be increased when Metharbital is combined with Diphenoxylate.
Oxymorphone The risk or severity of adverse effects can be increased when Metharbital is combined with Oxymorphone.
Dezocine The risk or severity of adverse effects can be increased when Metharbital is combined with Dezocine.
Levacetylmethadol The risk or severity of adverse effects can be increased when Metharbital is combined with Levacetylmethadol.
Methadyl acetate The risk or severity of adverse effects can be increased when Metharbital is combined with Methadyl acetate.
Dihydroetorphine The risk or severity of adverse effects can be increased when Metharbital is combined with Dihydroetorphine.
Diamorphine The risk or severity of adverse effects can be increased when Metharbital is combined with Diamorphine.
Ethylmorphine The risk or severity of adverse effects can be increased when Metharbital is combined with Ethylmorphine.
Etorphine The risk or severity of adverse effects can be increased when Metharbital is combined with Etorphine.
Dextromoramide The risk or severity of adverse effects can be increased when Metharbital is combined with Dextromoramide.
Desomorphine The risk or severity of adverse effects can be increased when Metharbital is combined with Desomorphine.
Carfentanil The risk or severity of adverse effects can be increased when Metharbital is combined with Carfentanil.
Dihydrocodeine The risk or severity of adverse effects can be increased when Metharbital is combined with Dihydrocodeine.
Alphacetylmethadol The risk or severity of adverse effects can be increased when Metharbital is combined with Alphacetylmethadol.
Dihydromorphine The risk or severity of adverse effects can be increased when Metharbital is combined with Dihydromorphine.
Ketobemidone The risk or severity of adverse effects can be increased when Metharbital is combined with Ketobemidone.
DPDPE The risk or severity of adverse effects can be increased when Metharbital is combined with DPDPE.
Lofentanil The risk or severity of adverse effects can be increased when Metharbital is combined with Lofentanil.
Opium The risk or severity of adverse effects can be increased when Metharbital is combined with Opium.
Normethadone The risk or severity of adverse effects can be increased when Metharbital is combined with Normethadone.
Piritramide The risk or severity of adverse effects can be increased when Metharbital is combined with Piritramide.
Alphaprodine The risk or severity of adverse effects can be increased when Metharbital is combined with Alphaprodine.
Nicomorphine The risk or severity of adverse effects can be increased when Metharbital is combined with Nicomorphine.
Meptazinol The risk or severity of adverse effects can be increased when Metharbital is combined with Meptazinol.
Phenoperidine The risk or severity of adverse effects can be increased when Metharbital is combined with Phenoperidine.
Phenazocine The risk or severity of adverse effects can be increased when Metharbital is combined with Phenazocine.
Tilidine The risk or severity of adverse effects can be increased when Metharbital is combined with Tilidine.
Carfentanil, C-11 The risk or severity of adverse effects can be increased when Metharbital is combined with Carfentanil, C-11.
Benzhydrocodone The risk or severity of adverse effects can be increased when Metharbital is combined with Benzhydrocodone.
Naloxegol The risk or severity of adverse effects can be increased when Metharbital is combined with Naloxegol.
Mecamylamine The risk or severity of adverse effects can be increased when Metharbital is combined with Mecamylamine.

Target Protein

Gamma-aminobutyric acid receptor subunit alpha-2 GABRA2
Gamma-aminobutyric acid receptor subunit gamma-3 GABRG3
Gamma-aminobutyric acid receptor subunit alpha-3 GABRA3
Gamma-aminobutyric acid receptor subunit alpha-4 GABRA4
Gamma-aminobutyric acid receptor subunit alpha-5 GABRA5
Gamma-aminobutyric acid receptor subunit alpha-6 GABRA6
GABA(A) Receptor GABRA1
Gamma-aminobutyric acid receptor subunit alpha-1 GABRA1
Neuronal acetylcholine receptor subunit alpha-4 CHRNA4
Neuronal acetylcholine receptor subunit alpha-7 CHRNA7
Glutamate receptor 2 GRIA2
Glutamate receptor ionotropic, kainate 2 GRIK2

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Gemonil — Abbott Laboratories

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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