Peringatan Keamanan

The intravenous LD50 of droperidol is 20-43 mg/kg in mice; 30 mg/kg in rats; 25 mg/kg in dogs and 11-13 mg/kg in rabbits. The intramuscular LD50 of droperidol is 195 mg/kg in mice, 104-110 mg/kg in rats; 97 mg/kg in rabbits and 200 mg/kg in guinea pigs. The manifestations of droperidol overdosage are an extension of its pharmacologic actions.

Droperidol

DB00450

small molecule approved vet_approved

Deskripsi

A butyrophenone with general properties similar to those of haloperidol. It is used in conjunction with an opioid analgesic such as fentanyl to maintain the patient in a calm state of neuroleptanalgesia with indifference to surroundings but still able to cooperate with the surgeon. It is also used as a premedicant, as an antiemetic, and for the control of agitation in acute psychoses. (From Martindale, The Extra Pharmacopoeia, 29th ed, p593)

Struktur Molekul 2D

Berat 379.4274
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Biphasic distribution. The rapid distribution phase is 1.4 ± 0.5 minutes and the slower distribution phase is 14.3 ± 6.5 minutes. Elimination half-life in adults is 134 ± 13 minutes and may be increased in geriatric patients. In children, it is 101.5 ± 26.4 minutes.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Completely absorbed following intramuscular administration.

Metabolisme

Extensively metabolized.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1371 Data
Ivabradine Ivabradine may increase the QTc-prolonging activities of Droperidol.
Valsartan Droperidol may decrease the antihypertensive activities of Valsartan.
Ramipril Droperidol may decrease the antihypertensive activities of Ramipril.
Remikiren Droperidol may decrease the antihypertensive activities of Remikiren.
Torasemide Droperidol may decrease the antihypertensive activities of Torasemide.
Guanadrel Droperidol may decrease the antihypertensive activities of Guanadrel.
Olmesartan Droperidol may decrease the antihypertensive activities of Olmesartan.
Chlorthalidone Droperidol may decrease the antihypertensive activities of Chlorthalidone.
Nitroprusside Droperidol may decrease the antihypertensive activities of Nitroprusside.
Minoxidil Droperidol may decrease the antihypertensive activities of Minoxidil.
Bendroflumethiazide Droperidol may decrease the antihypertensive activities of Bendroflumethiazide.
Fosinopril Droperidol may decrease the antihypertensive activities of Fosinopril.
Trandolapril Droperidol may decrease the antihypertensive activities of Trandolapril.
Metolazone Droperidol may decrease the antihypertensive activities of Metolazone.
Benazepril Droperidol may decrease the antihypertensive activities of Benazepril.
Bosentan Droperidol may decrease the antihypertensive activities of Bosentan.
Enalapril Droperidol may decrease the antihypertensive activities of Enalapril.
Cyclothiazide Droperidol may decrease the antihypertensive activities of Cyclothiazide.
Candoxatril Droperidol may decrease the antihypertensive activities of Candoxatril.
Mecamylamine Droperidol may decrease the antihypertensive activities of Mecamylamine.
Eplerenone Droperidol may decrease the antihypertensive activities of Eplerenone.
Lisinopril Droperidol may decrease the antihypertensive activities of Lisinopril.
Nitroglycerin Droperidol may decrease the antihypertensive activities of Nitroglycerin.
Hydroflumethiazide Droperidol may decrease the antihypertensive activities of Hydroflumethiazide.
Cryptenamine Droperidol may decrease the antihypertensive activities of Cryptenamine.
Perindopril Droperidol may decrease the antihypertensive activities of Perindopril.
Candesartan cilexetil Droperidol may decrease the antihypertensive activities of Candesartan cilexetil.
Eprosartan Droperidol may decrease the antihypertensive activities of Eprosartan.
Chlorothiazide Droperidol may decrease the antihypertensive activities of Chlorothiazide.
Quinapril Droperidol may decrease the antihypertensive activities of Quinapril.
Telmisartan Droperidol may decrease the antihypertensive activities of Telmisartan.
Trichlormethiazide Droperidol may decrease the antihypertensive activities of Trichlormethiazide.
Irbesartan Droperidol may decrease the antihypertensive activities of Irbesartan.
Deserpidine Droperidol may decrease the antihypertensive activities of Deserpidine.
Pentolinium Droperidol may decrease the antihypertensive activities of Pentolinium.
Trimethaphan Droperidol may decrease the antihypertensive activities of Trimethaphan.
Diazoxide Droperidol may decrease the antihypertensive activities of Diazoxide.
Guanethidine Droperidol may decrease the antihypertensive activities of Guanethidine.
Captopril Droperidol may decrease the antihypertensive activities of Captopril.
Epoprostenol Droperidol may decrease the antihypertensive activities of Epoprostenol.
Hydralazine Droperidol may decrease the antihypertensive activities of Hydralazine.
Polythiazide Droperidol may decrease the antihypertensive activities of Polythiazide.
Cilazapril Droperidol may decrease the antihypertensive activities of Cilazapril.
Saprisartan Droperidol may decrease the antihypertensive activities of Saprisartan.
Spirapril Droperidol may decrease the antihypertensive activities of Spirapril.
Tienilic acid Droperidol may decrease the antihypertensive activities of Tienilic acid.
Debrisoquine Droperidol may decrease the antihypertensive activities of Debrisoquine.
Sitaxentan Droperidol may decrease the antihypertensive activities of Sitaxentan.
Ambrisentan Droperidol may decrease the antihypertensive activities of Ambrisentan.
Diethylnorspermine Droperidol may decrease the antihypertensive activities of Diethylnorspermine.
Pinacidil Droperidol may decrease the antihypertensive activities of Pinacidil.
Temocapril Droperidol may decrease the antihypertensive activities of Temocapril.
Riociguat Droperidol may decrease the antihypertensive activities of Riociguat.
Macitentan Droperidol may decrease the antihypertensive activities of Macitentan.
Aliskiren Droperidol may decrease the antihypertensive activities of Aliskiren.
Nicorandil Droperidol may decrease the antihypertensive activities of Nicorandil.
Rauwolfia serpentina root Droperidol may decrease the antihypertensive activities of Rauwolfia serpentina root.
Enalaprilat Droperidol may decrease the antihypertensive activities of Enalaprilat.
Selexipag Droperidol may decrease the antihypertensive activities of Selexipag.
Angiotensin 1-7 Droperidol may decrease the antihypertensive activities of Angiotensin 1-7.
Imidapril Droperidol may decrease the antihypertensive activities of Imidapril.
BQ-123 Droperidol may decrease the antihypertensive activities of BQ-123.
Dihydralazine Droperidol may decrease the antihypertensive activities of Dihydralazine.
Zofenopril Droperidol may decrease the antihypertensive activities of Zofenopril.
Guanoxan Droperidol may decrease the antihypertensive activities of Guanoxan.
Delapril Droperidol may decrease the antihypertensive activities of Delapril.
Vincamine Droperidol may decrease the antihypertensive activities of Vincamine.
Linsidomine Droperidol may decrease the antihypertensive activities of Linsidomine.
Guanoxabenz Droperidol may decrease the antihypertensive activities of Guanoxabenz.
Tolonidine Droperidol may decrease the antihypertensive activities of Tolonidine.
Endralazine Droperidol may decrease the antihypertensive activities of Endralazine.
Cadralazine Droperidol may decrease the antihypertensive activities of Cadralazine.
Cyclopenthiazide Droperidol may decrease the antihypertensive activities of Cyclopenthiazide.
Bietaserpine Droperidol may decrease the antihypertensive activities of Bietaserpine.
Guanazodine Droperidol may decrease the antihypertensive activities of Guanazodine.
Methoserpidine Droperidol may decrease the antihypertensive activities of Methoserpidine.
Guanoclor Droperidol may decrease the antihypertensive activities of Guanoclor.
Muzolimine Droperidol may decrease the antihypertensive activities of Muzolimine.
Xipamide Droperidol may decrease the antihypertensive activities of Xipamide.
Candesartan Droperidol may decrease the antihypertensive activities of Candesartan.
Tocopherylquinone Droperidol may decrease the antihypertensive activities of Tocopherylquinone.
Benazeprilat Droperidol may decrease the antihypertensive activities of Benazeprilat.
Fosinoprilat Droperidol may decrease the antihypertensive activities of Fosinoprilat.
Ramiprilat Droperidol may decrease the antihypertensive activities of Ramiprilat.
Perindoprilat Droperidol may decrease the antihypertensive activities of Perindoprilat.
Quinaprilat Droperidol may decrease the antihypertensive activities of Quinaprilat.
Furosemide Droperidol may decrease the antihypertensive activities of Furosemide.
Levamlodipine Droperidol may decrease the antihypertensive activities of Levamlodipine.
Buthiazide Droperidol may decrease the antihypertensive activities of Buthiazide.
Azilsartan medoxomil Droperidol may decrease the antihypertensive activities of Azilsartan medoxomil.
Buprenorphine Droperidol may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Droperidol.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Droperidol.
Botulinum toxin type B Droperidol may increase the central nervous system depressant (CNS depressant) activities of Botulinum toxin type B.
Botulinum toxin type A Droperidol may increase the central nervous system depressant (CNS depressant) activities of Botulinum toxin type A.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of Droperidol.
Ethchlorvynol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Ethchlorvynol.
Succinylcholine Droperidol may increase the central nervous system depressant (CNS depressant) activities of Succinylcholine.
Eletriptan Droperidol may increase the central nervous system depressant (CNS depressant) activities of Eletriptan.
Enflurane Droperidol may increase the central nervous system depressant (CNS depressant) activities of Enflurane.

Target Protein

Alpha-1A adrenergic receptor ADRA1A
D(2) dopamine receptor DRD2

Referensi & Sumber

Synthesis reference: Janssen, P.A.J. and Gardocki, J.F.; U.S. Patent 3,141,823; July 21, 1964; assigned to Research Laboratorium Dr. C. Janssen NV, Belgium. Januen, P.A.J.; U.S. Patent 3,161,645; December 15,1964: assigned to Research Laboratorium Dr. C. Janssen NV, Belgium.

Contoh Produk & Brand

Produk: 15 • International brands: 8
Produk
  • Droperidol
    Injection, solution • 2.5 mg/1mL • Intramuscular; Intravenous • US • Generic • Approved
  • Droperidol
    Injection, solution • 2.5 mg/1mL • Intramuscular; Intravenous • US • Generic • Approved
  • Droperidol
    Injection, solution • 2.5 mg/1mL • Intramuscular; Intravenous • US • Generic • Approved
  • Droperidol
    Injection, solution • 2.5 mg/1mL • Intramuscular; Intravenous • US • Generic • Approved
  • Droperidol
    Injection, solution • 2.5 mg/1mL • Intramuscular; Intravenous • US • Generic • Approved
  • Droperidol
    Injection, solution • 2.5 mg/1mL • Intramuscular; Intravenous • US • Generic • Approved
  • Droperidol
    Injection, solution • 2.5 mg/1mL • Intramuscular; Intravenous • US • Generic • Approved
  • Droperidol Injection
    Liquid • 2.5 mg / mL • Intramuscular; Intravenous • Canada • Approved
Menampilkan 8 dari 15 produk.
International Brands
  • Dehydrobenzperidol — Janssen
  • Dridol — Prostrakan
  • Droleptan — Daiichi Sankyo
  • Dropedol — Excelsior
  • Dropel — Siu Guan
  • Droperdal — Cristália
  • Droperidols — Grindeks
  • Xomolix — Arzneimittel ProStrakan

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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