Peringatan Keamanan

Lindane is a moderately toxic compound via oral exposure, with a reported oral LD50 of 88 to 190 mg/kg in rats. Gamma-HCH (which constitutes 99% of lindane) is generally considered to be the most acutely toxic of the isomers following single administration. It is moderately toxic via the dermal route as well, with reported dermal LD50 values of 500 to 1000 mg/kg in rats, 300 mg/kg in mice, 400 mg/kg in guinea pigs, and 300 mg/kg in rabbits. Acute exposure to lindane may lead to central nervous system stimulation (usually developing within 1 hour), mental/motor impairment, excitation, clonic (intermittent) and tonic (continuous) convulsion. Other adverse reactions include central nervous system toxicity, as well as skin and gastrointestinal changes.

Lindane

DB00431

small molecule approved withdrawn

Deskripsi

An organochlorine insecticide that has been used as a pediculicide and a scabicide. Lindane has been banned in California, United Kingdom, Australia, and many western countries due to concerns about neurotoxicity and adverse effects on the environment. In Canada, Lindane is not recommmended as a first-line therapy due to reports of resistance, neurotoxicity, and bone marrow suppression, but has been approved by the FDA as a second-line therapy for topical treatment of pediculosis capitis (head lice), pediculosis pubis (pubic lice), or scabies in patients greater than two years of age who cannot tolerate or have failed first-line treatment. Lindane is still allowed for pharmaceutical use until 2015.

Struktur Molekul 2D

Berat 290.83
Wujud liquid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 18 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Lindane is absorbed significantly through the skin. A mean peak blood concentration of 28 nanograms per mL occurred in infants and children 6 hours after total body application of lindane lotion for scabies.

Metabolisme

Primarily hepatic through dechlorination leading to 2-chlorophenol, 0-chlorophenol, chlorocyclohexane, chlorocyclohexanol.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

1 Data
  • 1. Avoid excessive or chronic alcohol consumption.

Interaksi Obat

3 Data
Dalfampridine The risk or severity of seizure can be increased when Lindane is combined with Dalfampridine.
Bupropion The risk or severity of seizure can be increased when Bupropion is combined with Lindane.
Hydroxychloroquine The risk or severity of seizure can be increased when Hydroxychloroquine is combined with Lindane.

Target Protein

Gamma-aminobutyric acid receptor subunit beta-1 GABRB1
Glycine receptor subunit alpha-1 GLRA1
Glycine receptor subunit alpha-2 GLRA2
Glycine receptor subunit alpha-3 GLRA3
Glycine receptor subunit beta GLRB
Gamma-aminobutyric acid receptor subunit beta-3 GABRB3
Gamma-aminobutyric acid receptor subunit rho-1 GABRR1
Progesterone receptor PGR
Estrogen receptor ESR1
Nuclear receptor subfamily 1 group I member 2 NR1I2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 18335087
    Brown VJ: Life after lindane in California. Environ Health Perspect. 2008 Mar;116(3):A128.
  • PMID: 17636630
    Strong M, Johnstone P: Interventions for treating scabies. Cochrane Database Syst Rev. 2007 Jul 18;(3):CD000320.

Contoh Produk & Brand

Produk: 17 • International brands: 3
Produk
  • Dom-lindane Lotion - 1%
    Liquid • 1 % • Topical • Canada • Generic • OTC • Approved
  • Hexit Lotion
    Lotion • 1 % • Topical • Canada • OTC • Approved
  • Hexit Shampoo 1.0%
    Shampoo • 1 % • Topical • Canada • OTC • Approved
  • Kwellada Lotion 1%
    Lotion • 1 % • Topical • Canada • OTC • Approved
  • Kwellada Shampoo 1%
    Shampoo • 1 % • Topical • Canada • OTC • Approved
  • Lindane
    Lotion • 10 mg/1mL • Topical • US • Approved
  • Lindane
    Shampoo • 10 mg/1mL • Topical • US • Approved
  • Lindane
    Shampoo • 10 mg/1mL • Topical • US • Generic • Approved
Menampilkan 8 dari 17 produk.
International Brands
  • Gamene
  • Kwell
  • Scabene

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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