Peringatan Keamanan

Symptoms of an overdose typically include sluggishness, incoordination, difficulty in thinking, slowness of speech, faulty judgment, drowsiness or coma, shallow breathing, staggering, and in severe cases coma and death.

Secobarbital

DB00418

small molecule approved vet_approved

Deskripsi

Secobarbital (marketed by Eli Lilly and Company under the brand names Seconal and Tuinal) is a barbiturate derivative drug with anaesthetic, anticonvulsant, sedative and hypnotic properties. It is commonly known as quinalbarbitone in the United Kingdom.

Struktur Molekul 2D

Berat 238.2829
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Barbiturates are metabolized primarily by the hepatic microsomal enzyme system, and the metabolic products are excreted in the urine and, less commonly, in the feces.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol. Taking with alcohol may cause additive CNS depression.
  • 2. Take on an empty stomach. This may increase the rate of absorption.

Interaksi Obat

1875 Data
Aripiprazole The metabolism of Aripiprazole can be increased when combined with Secobarbital.
Aripiprazole lauroxil The metabolism of Aripiprazole lauroxil can be increased when combined with Secobarbital.
Buprenorphine Secobarbital may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Secobarbital.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Secobarbital.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Secobarbital.
Hydrocodone Secobarbital may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Secobarbital.
Magnesium sulfate The therapeutic efficacy of Secobarbital can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Secobarbital may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Secobarbital may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Secobarbital.
Mirtazapine Secobarbital may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Secobarbital.
Orphenadrine Secobarbital may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Secobarbital may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Pramipexole Secobarbital may increase the sedative activities of Pramipexole.
Rotigotine Secobarbital may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Secobarbital.
Suvorexant Secobarbital may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Secobarbital.
Thalidomide Secobarbital may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Secobarbital may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Secretin porcine The therapeutic efficacy of Secretin porcine can be decreased when used in combination with Secobarbital.
Mefloquine The therapeutic efficacy of Secobarbital can be decreased when used in combination with Mefloquine.
Orlistat Orlistat can cause a decrease in the absorption of Secobarbital resulting in a reduced serum concentration and potentially a decrease in efficacy.
Acetaminophen The metabolism of Acetaminophen can be increased when combined with Secobarbital.
Chloramphenicol The metabolism of Secobarbital can be decreased when combined with Chloramphenicol.
Doxycycline The serum concentration of Doxycycline can be decreased when it is combined with Secobarbital.
Felbamate The serum concentration of Secobarbital can be increased when it is combined with Felbamate.
Griseofulvin The serum concentration of Griseofulvin can be decreased when it is combined with Secobarbital.
Lamotrigine The serum concentration of Lamotrigine can be decreased when it is combined with Secobarbital.
Mianserin The therapeutic efficacy of Secobarbital can be decreased when used in combination with Mianserin.
Primidone The risk or severity of adverse effects can be increased when Primidone is combined with Secobarbital.
Methylphenobarbital The risk or severity of adverse effects can be increased when Methylphenobarbital is combined with Secobarbital.
Pyridoxine The metabolism of Secobarbital can be increased when combined with Pyridoxine.
Teniposide The serum concentration of Teniposide can be decreased when it is combined with Secobarbital.
Ulipristal The serum concentration of Ulipristal can be decreased when it is combined with Secobarbital.
Voriconazole The serum concentration of Voriconazole can be decreased when it is combined with Secobarbital.
Topotecan Secobarbital may increase the excretion rate of Topotecan which could result in a lower serum level and potentially a reduction in efficacy.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Secobarbital.
Sodium oxybate Secobarbital may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Ifosfamide The metabolism of Ifosfamide can be increased when combined with Secobarbital.
Perampanel The metabolism of Perampanel can be increased when combined with Secobarbital.
Warfarin The metabolism of Warfarin can be increased when combined with Secobarbital.
Acenocoumarol The metabolism of Acenocoumarol can be increased when combined with Secobarbital.
(R)-warfarin The metabolism of (R)-warfarin can be increased when combined with Secobarbital.
R,S-Warfarin alcohol The metabolism of R,S-Warfarin alcohol can be increased when combined with Secobarbital.
S,R-Warfarin alcohol The metabolism of S,R-Warfarin alcohol can be increased when combined with Secobarbital.
(S)-Warfarin The metabolism of (S)-Warfarin can be increased when combined with Secobarbital.
Tetracosactide The risk or severity of liver damage can be increased when Tetracosactide is combined with Secobarbital.
Aminophylline The therapeutic efficacy of Secobarbital can be decreased when used in combination with Aminophylline.
Botulinum toxin type A The risk or severity of adverse effects can be increased when Secobarbital is combined with Botulinum toxin type A.
Botulinum toxin type B The risk or severity of adverse effects can be increased when Secobarbital is combined with Botulinum toxin type B.
Meperidine Secobarbital may increase the hypotensive and central nervous system depressant (CNS depressant) activities of Meperidine.
Somatostatin The risk or severity of adverse effects can be increased when Somatostatin is combined with Secobarbital.
Ethanol Secobarbital may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Secobarbital may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Secobarbital.
Fluvoxamine The risk or severity of adverse effects can be increased when Secobarbital is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Secobarbital is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Secobarbital is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Secobarbital is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Secobarbital is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Secobarbital is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Secobarbital is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Secobarbital is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Secobarbital is combined with Escitalopram.
Zimelidine The risk or severity of adverse effects can be increased when Secobarbital is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Secobarbital is combined with Dapoxetine.
Desvenlafaxine The risk or severity of adverse effects can be increased when Secobarbital is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Secobarbital is combined with Seproxetine.
Indalpine The risk or severity of adverse effects can be increased when Secobarbital is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Secobarbital is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Secobarbital is combined with Alaproclate.
Naltrexone The risk or severity of adverse effects can be increased when Secobarbital is combined with Naltrexone.
Bezitramide The risk or severity of adverse effects can be increased when Secobarbital is combined with Bezitramide.
Hydromorphone The risk or severity of adverse effects can be increased when Secobarbital is combined with Hydromorphone.
Oxycodone The risk or severity of adverse effects can be increased when Secobarbital is combined with Oxycodone.
Butorphanol The risk or severity of adverse effects can be increased when Secobarbital is combined with Butorphanol.
Dextropropoxyphene The risk or severity of adverse effects can be increased when Secobarbital is combined with Dextropropoxyphene.
Pentazocine The risk or severity of adverse effects can be increased when Secobarbital is combined with Pentazocine.
Sufentanil The risk or severity of adverse effects can be increased when Secobarbital is combined with Sufentanil.
Nalbuphine The risk or severity of adverse effects can be increased when Secobarbital is combined with Nalbuphine.
Levorphanol The risk or severity of adverse effects can be increased when Secobarbital is combined with Levorphanol.
Remifentanil The risk or severity of adverse effects can be increased when Secobarbital is combined with Remifentanil.
Diphenoxylate The risk or severity of adverse effects can be increased when Secobarbital is combined with Diphenoxylate.
Oxymorphone The risk or severity of adverse effects can be increased when Secobarbital is combined with Oxymorphone.
Dezocine The risk or severity of adverse effects can be increased when Secobarbital is combined with Dezocine.
Methadyl acetate The risk or severity of adverse effects can be increased when Secobarbital is combined with Methadyl acetate.
Dihydroetorphine The risk or severity of adverse effects can be increased when Secobarbital is combined with Dihydroetorphine.
Diamorphine The risk or severity of adverse effects can be increased when Secobarbital is combined with Diamorphine.
Ethylmorphine The risk or severity of adverse effects can be increased when Secobarbital is combined with Ethylmorphine.
Etorphine The risk or severity of adverse effects can be increased when Secobarbital is combined with Etorphine.
Dextromoramide The risk or severity of adverse effects can be increased when Secobarbital is combined with Dextromoramide.
Desomorphine The risk or severity of adverse effects can be increased when Secobarbital is combined with Desomorphine.
Carfentanil The risk or severity of adverse effects can be increased when Secobarbital is combined with Carfentanil.
Dihydrocodeine The risk or severity of adverse effects can be increased when Secobarbital is combined with Dihydrocodeine.
Alphacetylmethadol The risk or severity of adverse effects can be increased when Secobarbital is combined with Alphacetylmethadol.
Dihydromorphine The risk or severity of adverse effects can be increased when Secobarbital is combined with Dihydromorphine.

Target Protein

Gamma-aminobutyric acid receptor subunit alpha-2 GABRA2
Gamma-aminobutyric acid receptor subunit alpha-3 GABRA3
Gamma-aminobutyric acid receptor subunit alpha-4 GABRA4
Gamma-aminobutyric acid receptor subunit alpha-5 GABRA5
Gamma-aminobutyric acid receptor subunit alpha-6 GABRA6
Gamma-aminobutyric acid receptor subunit alpha-1 GABRA1
Neuronal acetylcholine receptor subunit alpha-4 CHRNA4
Neuronal acetylcholine receptor subunit alpha-7 CHRNA7
Glutamate receptor 2 GRIA2
Glutamate receptor ionotropic, kainate 2 GRIK2
NMDA receptor GRIN1

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 7 • International brands: 2
Produk
  • Novo-secobarb 100mg
    Capsule • 100 mg / cap • Oral • Canada • Generic • Approved
  • Seconal Sodium
    Capsule • 100 mg/1 • Oral • US • Approved
  • Seconal Sodium
    Capsule • 100 mg/1 • Oral • US • Generic • Approved
  • Seconal Sodium
    Capsule • 100 mg/1 • Oral • US • Generic • Approved
  • Seconal Sodium Pulvule 240 0.1gm
    Capsule • 100 mg / cap • Oral • Canada • Approved
  • Tuinal Pulvule 303
    Capsule • - • Oral • Canada • Approved
  • Tuinal Pulvule 304
    Capsule • - • Oral • Canada • Approved
International Brands
  • Seconal
  • Tuinal

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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