Peringatan Keamanan

Excessive doses can be expected to produce enhanced pharmacological effects. Overdosage may increase the risk of histamine release and cardiovascular effects, especially hypotension.

Metocurine iodide

DB00416

small molecule approved withdrawn

Deskripsi

Metocurine iodide is a benzylisoquinolinium competitive nondepolarizing neuromuscular blocking agent. It is used as an anesthesia adjunct to induce skeletal muscle relaxation and to reduce the intensity of muscle contractions in convulsive therapy Metocurine iodide has a moderate risk of inducing histamine release and has some ganglion blocking activity. Metocurine iodide can be used most advantageously if muscle twitch response to peripheral nerve stimulation is monitored to assess degree of muscle relaxation. Metocurine Iodide is no longer available on the US market.

Struktur Molekul 2D

Berat 906.6279
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 3 to 4 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1113 Data
Buprenorphine Metocurine iodide may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Metocurine iodide.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Metocurine iodide.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Metocurine iodide.
Hydrocodone Metocurine iodide may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Metocurine iodide.
Magnesium sulfate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Metocurine iodide may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Metocurine iodide may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Metocurine iodide.
Mirtazapine Metocurine iodide may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Metocurine iodide.
Orphenadrine Metocurine iodide may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Metocurine iodide may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Metocurine iodide.
Pramipexole Metocurine iodide may increase the sedative activities of Pramipexole.
Ropinirole Metocurine iodide may increase the sedative activities of Ropinirole.
Rotigotine Metocurine iodide may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Metocurine iodide.
Sodium oxybate The risk or severity of CNS depression can be increased when Metocurine iodide is combined with Sodium oxybate.
Suvorexant Metocurine iodide may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Metocurine iodide.
Thalidomide Metocurine iodide may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Metocurine iodide may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Capreomycin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Capreomycin.
Cyclosporine The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Cyclosporine.
Doxycycline The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Doxycycline.
Lymecycline The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Lymecycline.
Framycetin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Framycetin.
Clomocycline The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Clomocycline.
Quinine The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Quinine.
Vancomycin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Vancomycin.
Tigecycline The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Tigecycline.
Oxytetracycline The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Oxytetracycline.
Chloroquine The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Chloroquine.
Demeclocycline The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Demeclocycline.
Mecamylamine The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Mecamylamine.
Tobramycin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Tobramycin.
Tetracycline The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Tetracycline.
Gentamicin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Gentamicin.
Etacrynic acid The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Etacrynic acid.
Quinidine The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Quinidine.
Metacycline The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Metacycline.
Netilmicin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Netilmicin.
Neomycin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Neomycin.
Streptomycin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Streptomycin.
Colistimethate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Colistimethate.
Kanamycin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Kanamycin.
Rolitetracycline The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Rolitetracycline.
Magnesium oxide The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium oxide.
Magnesium cation The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium cation.
Paromomycin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Paromomycin.
Lincomycin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Lincomycin.
Ribostamycin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Ribostamycin.
Geneticin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Geneticin.
Apramycin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Apramycin.
Gentamicin C1a The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Gentamicin C1a.
Neamine The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Neamine.
Arbekacin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Arbekacin.
Viomycin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Viomycin.
Puromycin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Puromycin.
Magnesium hydroxide The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium hydroxide.
Magnesium trisilicate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium trisilicate.
Magnesium chloride The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium chloride.
Magnesium acetate tetrahydrate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium acetate tetrahydrate.
Magnesium carbonate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium carbonate.
Magnesium citrate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium citrate.
Magnesium glycinate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium glycinate.
Magnesium Aluminum Silicate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium Aluminum Silicate.
Dihydrostreptomycin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Dihydrostreptomycin.
Hygromycin B The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Hygromycin B.
Sisomicin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Sisomicin.
Plazomicin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Plazomicin.
Magnesium silicate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium silicate.
Penimepicycline The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Penimepicycline.
Magnesium aspartate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium aspartate.
Isepamicin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Isepamicin.
Magnesium gluconate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium gluconate.
Magnesium orotate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium orotate.
Magnesium phosphate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium phosphate.
Magnesium acetate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium acetate.
Procainamide The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Procainamide.
Dantrolene The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Dantrolene.
Piperacillin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Piperacillin.
Magnesium stearate The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Magnesium stearate.
Colistin The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Colistin.
Secretin porcine The therapeutic efficacy of Secretin porcine can be decreased when used in combination with Metocurine iodide.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Metocurine iodide.
Spironolactone Spironolactone may increase the neuromuscular blocking activities of Metocurine iodide.
Botulinum toxin type A The risk or severity of adverse effects can be increased when Metocurine iodide is combined with Botulinum toxin type A.
Botulinum toxin type B The risk or severity of adverse effects can be increased when Metocurine iodide is combined with Botulinum toxin type B.
Ethanol Metocurine iodide may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Metocurine iodide may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Metocurine iodide.
Fluvoxamine The risk or severity of adverse effects can be increased when Metocurine iodide is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Metocurine iodide is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Metocurine iodide is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Metocurine iodide is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Metocurine iodide is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Metocurine iodide is combined with Sertraline.

Target Protein

Neuronal acetylcholine receptor subunit alpha-4 CHRNA4
Neuronal acetylcholine receptor subunit beta-2 CHRNB2
Neuronal acetylcholine receptor subunit alpha-2 CHRNA2

Referensi & Sumber

Synthesis reference: Bray, M.D.; U.S. Patent 2,581,903; January 8, 1952; assigned to Eli Lilly and Company.

Contoh Produk & Brand

Produk: 1 • International brands: 0
Produk
  • Metubine Iodide Inj 2mg/ml
    Liquid • 2 mg / mL • Intravenous • Canada • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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