Peringatan Keamanan

Oral, rat LD50: 5 gm/kg; Oral, mouse LD50: >2500 mg/kg. Symptoms of an acetohexamide overdose include hunger, nausea, anxiety, cold sweats, weakness, drowsiness, unconsciousness, and coma.

Acetohexamide

DB00414

small molecule approved investigational withdrawn

Deskripsi

A sulfonylurea hypoglycemic agent that is metabolized in the liver to 1-hydrohexamide. Acetohexamide has been discontinued in the US market.

Struktur Molekul 2D

Berat 324.395
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Elimination half-life of the parent compound is 1.3 hours and the elimination half-life of the active metabolite is approximately 5-6 hours.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Rapidly absorbed from the GI tract.

Metabolisme

Extensively metabolized in the liver to the active metabolite hydroxyhexamide, which exhibits greater hypoglycemic potency than acetohexamide. Hydroxyhexamide is believed to be responsible for prolonged hypoglycemic effects.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol.
  • 2. Take with or without food. The absorption is unaffected by food.

Interaksi Obat

1035 Data
Pegvisomant The risk or severity of hypoglycemia can be increased when Pegvisomant is combined with Acetohexamide.
Carbocisteine The risk or severity of adverse effects can be increased when Acetohexamide is combined with Carbocisteine.
Chloramphenicol The metabolism of Acetohexamide can be decreased when combined with Chloramphenicol.
Cimetidine The serum concentration of Acetohexamide can be increased when it is combined with Cimetidine.
Fluconazole The serum concentration of Acetohexamide can be increased when it is combined with Fluconazole.
Metreleptin Metreleptin may increase the hypoglycemic activities of Acetohexamide.
Probenecid The protein binding of Acetohexamide can be decreased when combined with Probenecid.
Ranitidine The serum concentration of Acetohexamide can be increased when it is combined with Ranitidine.
Voriconazole The serum concentration of Acetohexamide can be increased when it is combined with Voriconazole.
Clarithromycin The serum concentration of Acetohexamide can be increased when it is combined with Clarithromycin.
Lipoic acid The risk or severity of hypoglycemia can be increased when Lipoic acid is combined with Acetohexamide.
Rifampin The serum concentration of Acetohexamide can be decreased when it is combined with Rifampicin.
Moxifloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Moxifloxacin.
Grepafloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Grepafloxacin.
Enoxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Enoxacin.
Pefloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Pefloxacin.
Ciprofloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Ciprofloxacin.
Trovafloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Trovafloxacin.
Nalidixic acid The therapeutic efficacy of Acetohexamide can be increased when used in combination with Nalidixic acid.
Rosoxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Rosoxacin.
Cinoxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Cinoxacin.
Lomefloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Lomefloxacin.
Gatifloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Gatifloxacin.
Norfloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Norfloxacin.
Levofloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Levofloxacin.
Gemifloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Gemifloxacin.
Ofloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Ofloxacin.
Sparfloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Sparfloxacin.
Temafloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Temafloxacin.
Fleroxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Fleroxacin.
Technetium Tc-99m ciprofloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Technetium Tc-99m ciprofloxacin.
Garenoxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Garenoxacin.
Nemonoxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Nemonoxacin.
Flumequine The therapeutic efficacy of Acetohexamide can be increased when used in combination with Flumequine.
Enrofloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Enrofloxacin.
Orbifloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Orbifloxacin.
Sarafloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Sarafloxacin.
Difloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Difloxacin.
Pazufloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Pazufloxacin.
Prulifloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Prulifloxacin.
Delafloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Delafloxacin.
Sitafloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Sitafloxacin.
Oxolinic acid The therapeutic efficacy of Acetohexamide can be increased when used in combination with Oxolinic acid.
Rufloxacin The therapeutic efficacy of Acetohexamide can be increased when used in combination with Rufloxacin.
Pipemidic acid The therapeutic efficacy of Acetohexamide can be increased when used in combination with Pipemidic acid.
Methyclothiazide The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Methyclothiazide.
Chlorthalidone The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Chlorthalidone.
Bendroflumethiazide The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Bendroflumethiazide.
Metolazone The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Metolazone.
Benzthiazide The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Benzthiazide.
Hydroflumethiazide The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Hydroflumethiazide.
Indapamide The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Indapamide.
Chlorothiazide The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Chlorothiazide.
Hydrochlorothiazide The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Hydrochlorothiazide.
Trichlormethiazide The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Trichlormethiazide.
Polythiazide The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Polythiazide.
Quinethazone The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Quinethazone.
Cyclopenthiazide The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Cyclopenthiazide.
Epitizide The therapeutic efficacy of Acetohexamide can be decreased when used in combination with Epitizide.
Esmolol Esmolol may increase the hypoglycemic activities of Acetohexamide.
Landiolol Landiolol may increase the hypoglycemic activities of Acetohexamide.
Ethanol The risk or severity of adverse effects can be increased when Acetohexamide is combined with Ethanol.
Amitriptyline Amitriptyline may decrease the hypoglycemic activities of Acetohexamide.
Protriptyline Protriptyline may decrease the hypoglycemic activities of Acetohexamide.
Imipramine Imipramine may decrease the hypoglycemic activities of Acetohexamide.
Nortriptyline Nortriptyline may decrease the hypoglycemic activities of Acetohexamide.
Amoxapine Amoxapine may decrease the hypoglycemic activities of Acetohexamide.
Desipramine Desipramine may decrease the hypoglycemic activities of Acetohexamide.
Clomipramine Clomipramine may decrease the hypoglycemic activities of Acetohexamide.
Amineptine Amineptine may decrease the hypoglycemic activities of Acetohexamide.
Dimetacrine Dimetacrine may decrease the hypoglycemic activities of Acetohexamide.
Butriptyline Butriptyline may decrease the hypoglycemic activities of Acetohexamide.
Dosulepin Dosulepin may decrease the hypoglycemic activities of Acetohexamide.
Tianeptine Tianeptine may decrease the hypoglycemic activities of Acetohexamide.
Oxaprotiline Oxaprotiline may decrease the hypoglycemic activities of Acetohexamide.
Opipramol Opipramol may decrease the hypoglycemic activities of Acetohexamide.
Amitriptylinoxide Amitriptylinoxide may decrease the hypoglycemic activities of Acetohexamide.
Dibenzepin Dibenzepin may decrease the hypoglycemic activities of Acetohexamide.
Quinupramine Quinupramine may decrease the hypoglycemic activities of Acetohexamide.
Melitracen Melitracen may decrease the hypoglycemic activities of Acetohexamide.
Lofepramine Lofepramine may decrease the hypoglycemic activities of Acetohexamide.
Iprindole Iprindole may decrease the hypoglycemic activities of Acetohexamide.
Imipramine oxide Imipramine oxide may decrease the hypoglycemic activities of Acetohexamide.
Doxepin Doxepin may decrease the hypoglycemic activities of Acetohexamide.
Clofibrate The risk or severity of hypoglycemia can be increased when Clofibrate is combined with Acetohexamide.
Fenofibrate The risk or severity of hypoglycemia can be increased when Fenofibrate is combined with Acetohexamide.
Bezafibrate The risk or severity of hypoglycemia can be increased when Bezafibrate is combined with Acetohexamide.
Etofibrate The risk or severity of hypoglycemia can be increased when Etofibrate is combined with Acetohexamide.
Ciprofibrate The risk or severity of hypoglycemia can be increased when Ciprofibrate is combined with Acetohexamide.
Simfibrate The risk or severity of hypoglycemia can be increased when Simfibrate is combined with Acetohexamide.
Ronifibrate The risk or severity of hypoglycemia can be increased when Ronifibrate is combined with Acetohexamide.
Aluminium clofibrate The risk or severity of hypoglycemia can be increased when Aluminium clofibrate is combined with Acetohexamide.
Clofibride The risk or severity of hypoglycemia can be increased when Clofibride is combined with Acetohexamide.
Fenofibric acid The risk or severity of hypoglycemia can be increased when Fenofibric acid is combined with Acetohexamide.
Miconazole The serum concentration of Acetohexamide can be increased when it is combined with Miconazole.
Phenindione Acetohexamide may increase the anticoagulant activities of Phenindione.
Coumarin Acetohexamide may increase the anticoagulant activities of Coumarin.
(R)-warfarin Acetohexamide may increase the anticoagulant activities of (R)-warfarin.
Clorindione Acetohexamide may increase the anticoagulant activities of Clorindione.
Diphenadione Acetohexamide may increase the anticoagulant activities of Diphenadione.

Target Protein

ATP-sensitive inward rectifier potassium channel 1 KCNJ1
ATP-binding cassette sub-family C member 8 ABCC8

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 1 • International brands: 4
Produk
  • Dimelor Tablet 1843 500mg
    Tablet • 500 mg / tab • Oral • Canada • Approved
International Brands
  • Acetohexamide — Watson
  • Dimelin — Shionogi Seiyaku
  • Dymelor — Lilly
  • Gamadiabet — Salvat

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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