Peringatan Keamanan

LD50=65 mg/kg (Orally in mice)

Loxapine

DB00408

small molecule approved

Deskripsi

An antipsychotic agent used in schizophrenia. PubChem

Struktur Molekul 2D

Berat 327.808
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Oral-4 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Systemic bioavailability of the parent drug was only about one third that after an equivalent intramuscular dose (25 mg base) in male volunteers

Metabolisme

Hepatic

Rute Eliminasi

Metabolites are excreted in the urine in the form of conjugates and in the feces unconjugated.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol.
  • 2. Take with food. Food reduces irritation.

Interaksi Obat

941 Data
Omalizumab The therapeutic efficacy of Omalizumab can be decreased when used in combination with Loxapine.
Flunisolide The therapeutic efficacy of Flunisolide can be decreased when used in combination with Loxapine.
Ipratropium The therapeutic efficacy of Ipratropium can be decreased when used in combination with Loxapine.
Beclomethasone dipropionate The therapeutic efficacy of Beclomethasone dipropionate can be decreased when used in combination with Loxapine.
Montelukast The therapeutic efficacy of Montelukast can be decreased when used in combination with Loxapine.
Zafirlukast The therapeutic efficacy of Zafirlukast can be decreased when used in combination with Loxapine.
Fluticasone propionate The therapeutic efficacy of Fluticasone propionate can be decreased when used in combination with Loxapine.
Triamcinolone The therapeutic efficacy of Triamcinolone can be decreased when used in combination with Loxapine.
Zileuton The therapeutic efficacy of Zileuton can be decreased when used in combination with Loxapine.
Orciprenaline The therapeutic efficacy of Orciprenaline can be decreased when used in combination with Loxapine.
Terbutaline The therapeutic efficacy of Terbutaline can be decreased when used in combination with Loxapine.
Salmeterol The therapeutic efficacy of Salmeterol can be decreased when used in combination with Loxapine.
Formoterol The therapeutic efficacy of Formoterol can be decreased when used in combination with Loxapine.
Albuterol The therapeutic efficacy of Salbutamol can be decreased when used in combination with Loxapine.
Budesonide The therapeutic efficacy of Budesonide can be decreased when used in combination with Loxapine.
Arformoterol The therapeutic efficacy of Arformoterol can be decreased when used in combination with Loxapine.
Fenoterol The therapeutic efficacy of Fenoterol can be decreased when used in combination with Loxapine.
Pirbuterol The therapeutic efficacy of Pirbuterol can be decreased when used in combination with Loxapine.
Clenbuterol The therapeutic efficacy of Clenbuterol can be decreased when used in combination with Loxapine.
Bambuterol The therapeutic efficacy of Bambuterol can be decreased when used in combination with Loxapine.
Tiotropium The therapeutic efficacy of Tiotropium can be decreased when used in combination with Loxapine.
Ciclesonide The therapeutic efficacy of Ciclesonide can be decreased when used in combination with Loxapine.
Pranlukast The therapeutic efficacy of Pranlukast can be decreased when used in combination with Loxapine.
Roflumilast The therapeutic efficacy of Roflumilast can be decreased when used in combination with Loxapine.
Indacaterol The therapeutic efficacy of Indacaterol can be decreased when used in combination with Loxapine.
Protokylol The therapeutic efficacy of Protokylol can be decreased when used in combination with Loxapine.
Aclidinium The therapeutic efficacy of Aclidinium can be decreased when used in combination with Loxapine.
Fluticasone furoate The therapeutic efficacy of Fluticasone furoate can be decreased when used in combination with Loxapine.
Umeclidinium The therapeutic efficacy of Umeclidinium can be decreased when used in combination with Loxapine.
Olodaterol The therapeutic efficacy of Olodaterol can be decreased when used in combination with Loxapine.
Vilanterol The therapeutic efficacy of Vilanterol can be decreased when used in combination with Loxapine.
Tulobuterol The therapeutic efficacy of Tulobuterol can be decreased when used in combination with Loxapine.
Levosalbutamol The therapeutic efficacy of Levosalbutamol can be decreased when used in combination with Loxapine.
Afatinib The serum concentration of Afatinib can be increased when it is combined with Loxapine.
Bosutinib The serum concentration of Bosutinib can be increased when it is combined with Loxapine.
Brentuximab vedotin The serum concentration of Brentuximab vedotin can be increased when it is combined with Loxapine.
Colchicine The serum concentration of Colchicine can be increased when it is combined with Loxapine.
Edoxaban The serum concentration of Edoxaban can be increased when it is combined with Loxapine.
Ledipasvir The serum concentration of Ledipasvir can be increased when it is combined with Loxapine.
Naloxegol The serum concentration of Naloxegol can be increased when it is combined with Loxapine.
Pazopanib The serum concentration of Pazopanib can be increased when it is combined with Loxapine.
Prucalopride The serum concentration of Prucalopride can be increased when it is combined with Loxapine.
Ranolazine The serum concentration of Ranolazine can be increased when it is combined with Loxapine.
Silodosin The excretion of Silodosin can be decreased when combined with Loxapine.
Topotecan The serum concentration of Topotecan can be increased when it is combined with Loxapine.
Buprenorphine Loxapine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Loxapine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Loxapine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Loxapine.
Hydrocodone Loxapine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Loxapine.
Magnesium sulfate The therapeutic efficacy of Loxapine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Loxapine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Loxapine may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Loxapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Loxapine.
Orphenadrine Loxapine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Loxapine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Loxapine.
Rotigotine Loxapine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Loxapine.
Sodium oxybate Loxapine may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Loxapine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Loxapine.
Thalidomide Loxapine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Loxapine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Lorazepam The risk or severity of adverse effects can be increased when Loxapine is combined with Lorazepam.
Everolimus The serum concentration of Everolimus can be increased when it is combined with Loxapine.
Rifaximin The serum concentration of Rifaximin can be increased when it is combined with Loxapine.
Amisulpride Loxapine may increase the antipsychotic activities of Amisulpride.
Methylphenidate The risk or severity of adverse effects can be increased when Loxapine is combined with Methylphenidate.
Metoclopramide The risk or severity of adverse effects can be increased when Metoclopramide is combined with Loxapine.
Quinagolide The therapeutic efficacy of Quinagolide can be decreased when used in combination with Loxapine.
Sulpiride Loxapine may increase the antipsychotic activities of Sulpiride.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Loxapine.
Lithium citrate Lithium citrate may increase the neurotoxic activities of Loxapine.
Lithium hydroxide Lithium hydroxide may increase the neurotoxic activities of Loxapine.
Mequitazine Loxapine may increase the arrhythmogenic activities of Mequitazine.
Carbamazepine The serum concentration of the active metabolites of Carbamazepine can be increased when Carbamazepine is used in combination with Loxapine.
Linezolid The risk or severity of serotonin syndrome can be increased when Linezolid is combined with Loxapine.
Dicoumarol The risk or severity of adverse effects can be increased when Loxapine is combined with Dicoumarol.
Phenindione The risk or severity of adverse effects can be increased when Loxapine is combined with Phenindione.
Warfarin The risk or severity of adverse effects can be increased when Loxapine is combined with Warfarin.
Phenprocoumon The risk or severity of adverse effects can be increased when Loxapine is combined with Phenprocoumon.
Acenocoumarol The risk or severity of adverse effects can be increased when Loxapine is combined with Acenocoumarol.
4-hydroxycoumarin The risk or severity of adverse effects can be increased when Loxapine is combined with 4-hydroxycoumarin.
Coumarin The risk or severity of adverse effects can be increased when Loxapine is combined with Coumarin.
(R)-warfarin The risk or severity of adverse effects can be increased when Loxapine is combined with (R)-warfarin.
Ethyl biscoumacetate The risk or severity of adverse effects can be increased when Loxapine is combined with Ethyl biscoumacetate.
Fluindione The risk or severity of adverse effects can be increased when Loxapine is combined with Fluindione.
Clorindione The risk or severity of adverse effects can be increased when Loxapine is combined with Clorindione.
Diphenadione The risk or severity of adverse effects can be increased when Loxapine is combined with Diphenadione.
Tioclomarol The risk or severity of adverse effects can be increased when Loxapine is combined with Tioclomarol.
(S)-Warfarin The risk or severity of adverse effects can be increased when Loxapine is combined with (S)-Warfarin.
Mirtazapine Loxapine may increase the serotonergic activities of Mirtazapine.
Vincristine The excretion of Vincristine can be decreased when combined with Loxapine.
Ethanol Loxapine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Loxapine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Loxapine.
Zimelidine The risk or severity of adverse effects can be increased when Loxapine is combined with Zimelidine.

Target Protein

5-hydroxytryptamine receptor 2A HTR2A
D(2) dopamine receptor DRD2
5-hydroxytryptamine receptor 2C HTR2C
5-hydroxytryptamine receptor 1A HTR1A
5-hydroxytryptamine receptor 1B HTR1B
5-hydroxytryptamine receptor 1D HTR1D
5-hydroxytryptamine receptor 1E HTR1E
5-hydroxytryptamine receptor 3A HTR3A
5-hydroxytryptamine receptor 5A HTR5A
5-hydroxytryptamine receptor 6 HTR6
5-hydroxytryptamine receptor 7 HTR7
Alpha-1A adrenergic receptor ADRA1A
Alpha-1B adrenergic receptor ADRA1B
Alpha-2A adrenergic receptor ADRA2A
Alpha-2B adrenergic receptor ADRA2B
Alpha-2C adrenergic receptor ADRA2C
Beta-1 adrenergic receptor ADRB1
Muscarinic acetylcholine receptor M1 CHRM1
Muscarinic acetylcholine receptor M2 CHRM2
Muscarinic acetylcholine receptor M3 CHRM3
Muscarinic acetylcholine receptor M4 CHRM4
Muscarinic acetylcholine receptor M5 CHRM5
D(1) dopamine receptor DRD1
D(3) dopamine receptor DRD3
D(4) dopamine receptor DRD4
D(1B) dopamine receptor DRD5
Histamine H1 receptor HRH1
Histamine H2 receptor HRH2
Histamine H4 receptor HRH4
Sodium-dependent serotonin transporter SLC6A4
Sodium-dependent noradrenaline transporter SLC6A2
Sodium-dependent dopamine transporter SLC6A3
D(1A) dopamine receptor DRD1

Referensi & Sumber

Synthesis reference: U.S. Patents 3,412,193; 3,546,226.
Artikel (PubMed)
  • PMID: 10340686
    Glazer WM: Does loxapine have "atypical" properties? Clinical evidence. J Clin Psychiatry. 1999;60 Suppl 10:42-6.
  • PMID: 1860915
    Cheung SW, Tang SW, Remington G: Simultaneous quantitation of loxapine, amoxapine and their 7- and 8-hydroxy metabolites in plasma by high-performance liquid chromatography. J Chromatogr. 1991 Mar 8;564(1):213-21.

Contoh Produk & Brand

Produk: 134 • International brands: 5
Produk
  • Adasuve
    Aerosol, powder • 10 mg/1 • Respiratory (inhalation) • US • Approved
  • Adasuve
    Aerosol, powder • 10 mg/1 • Respiratory (inhalation) • US • Approved
  • Adasuve
    Aerosol, powder • 10 mg/1 • Respiratory (inhalation) • US • Approved
  • Adasuve
    Powder, metered • 4.5 mg • Respiratory (inhalation) • EU • Approved
  • Adasuve
    Powder, metered • 9.1 mg • Respiratory (inhalation) • EU • Approved
  • Adasuve
    Powder, metered • 4.5 mg • Respiratory (inhalation) • EU • Approved
  • Adasuve
    Powder, metered • 9.1 mg • Respiratory (inhalation) • EU • Approved
  • Apo-loxapine
    Tablet • 5 mg • Oral • Canada • Generic • Approved
Menampilkan 8 dari 134 produk.
International Brands
  • Cloxazepine
  • Lopac — Newai Chem
  • Losagen — Patron
  • Loxapac — Wyeth
  • Rosup — Swiss Pharm

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul