Peringatan Keamanan

No serious or unexpected toxicity has been observed with dydrogesterone. In acute toxicity studies, the LD50 doses in rats exceeded 4,640mg/kg for the oral route.

Dydrogesterone

DB00378

small molecule approved investigational withdrawn

Deskripsi

A synthetic progestational hormone with no androgenic or estrogenic properties. Unlike many other progestational compounds, dydrogesterone produces no increase in temperature and does not inhibit ovulation.

Struktur Molekul 2D

Berat 312.4458
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Dydrogesterone: 5-7 hours, 20-dihydrodydrogesterone (DHD) metabolite: 14-17 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Rapidly absorbed in the gastrointestinal tract with a bioavailability of 28%.

Metabolisme

Metabolism is complete to a 20-dihydrodydrogesterone (DHD) metabolite.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

206 Data
Ulipristal The therapeutic efficacy of Dydrogesterone can be decreased when used in combination with Ulipristal.
Lepirudin Dydrogesterone may decrease the anticoagulant activities of Lepirudin.
Bivalirudin Dydrogesterone may decrease the anticoagulant activities of Bivalirudin.
Alteplase Dydrogesterone may decrease the anticoagulant activities of Alteplase.
Urokinase Dydrogesterone may decrease the anticoagulant activities of Urokinase.
Reteplase Dydrogesterone may decrease the anticoagulant activities of Reteplase.
Anistreplase Dydrogesterone may decrease the anticoagulant activities of Anistreplase.
Tenecteplase Dydrogesterone may decrease the anticoagulant activities of Tenecteplase.
Abciximab Dydrogesterone may decrease the anticoagulant activities of Abciximab.
Drotrecogin alfa Dydrogesterone may decrease the anticoagulant activities of Drotrecogin alfa.
Streptokinase Dydrogesterone may decrease the anticoagulant activities of Streptokinase.
Dicoumarol Dydrogesterone may decrease the anticoagulant activities of Dicoumarol.
Ardeparin Dydrogesterone may decrease the anticoagulant activities of Ardeparin.
Phenindione Dydrogesterone may decrease the anticoagulant activities of Phenindione.
Fondaparinux Dydrogesterone may decrease the anticoagulant activities of Fondaparinux.
Pentosan polysulfate Dydrogesterone may decrease the anticoagulant activities of Pentosan polysulfate.
Dipyridamole Dydrogesterone may decrease the anticoagulant activities of Dipyridamole.
Heparin Dydrogesterone may decrease the anticoagulant activities of Heparin.
Enoxaparin Dydrogesterone may decrease the anticoagulant activities of Enoxaparin.
Epoprostenol Dydrogesterone may decrease the anticoagulant activities of Epoprostenol.
Coumarin Dydrogesterone may decrease the anticoagulant activities of Coumarin.
Ximelagatran Dydrogesterone may decrease the anticoagulant activities of Ximelagatran.
Desmoteplase Dydrogesterone may decrease the anticoagulant activities of Desmoteplase.
Defibrotide Dydrogesterone may decrease the anticoagulant activities of Defibrotide.
Ancrod Dydrogesterone may decrease the anticoagulant activities of Ancrod.
Beraprost Dydrogesterone may decrease the anticoagulant activities of Beraprost.
Prasugrel Dydrogesterone may decrease the anticoagulant activities of Prasugrel.
Sulodexide Dydrogesterone may decrease the anticoagulant activities of Sulodexide.
Semuloparin Dydrogesterone may decrease the anticoagulant activities of Semuloparin.
Idraparinux Dydrogesterone may decrease the anticoagulant activities of Idraparinux.
Cangrelor Dydrogesterone may decrease the anticoagulant activities of Cangrelor.
Astaxanthin Dydrogesterone may decrease the anticoagulant activities of Astaxanthin.
Apixaban Dydrogesterone may decrease the anticoagulant activities of Apixaban.
Otamixaban Dydrogesterone may decrease the anticoagulant activities of Otamixaban.
Amediplase Dydrogesterone may decrease the anticoagulant activities of Amediplase.
Dabigatran etexilate Dydrogesterone may decrease the anticoagulant activities of Dabigatran etexilate.
Danaparoid Dydrogesterone may decrease the anticoagulant activities of Danaparoid.
Dalteparin Dydrogesterone may decrease the anticoagulant activities of Dalteparin.
Tinzaparin Dydrogesterone may decrease the anticoagulant activities of Tinzaparin.
(R)-warfarin Dydrogesterone may decrease the anticoagulant activities of (R)-warfarin.
Nadroparin Dydrogesterone may decrease the anticoagulant activities of Nadroparin.
Triflusal Dydrogesterone may decrease the anticoagulant activities of Triflusal.
Ditazole Dydrogesterone may decrease the anticoagulant activities of Ditazole.
Vorapaxar Dydrogesterone may decrease the anticoagulant activities of Vorapaxar.
Edoxaban Dydrogesterone may decrease the anticoagulant activities of Edoxaban.
Sodium citrate Dydrogesterone may decrease the anticoagulant activities of Sodium citrate.
Dextran Dydrogesterone may decrease the anticoagulant activities of Dextran.
Bemiparin Dydrogesterone may decrease the anticoagulant activities of Bemiparin.
Parnaparin Dydrogesterone may decrease the anticoagulant activities of Parnaparin.
Desirudin Dydrogesterone may decrease the anticoagulant activities of Desirudin.
Antithrombin Alfa Dydrogesterone may decrease the anticoagulant activities of Antithrombin Alfa.
Protein C Dydrogesterone may decrease the anticoagulant activities of Protein C.
Antithrombin III human Dydrogesterone may decrease the anticoagulant activities of Antithrombin III human.
Letaxaban Dydrogesterone may decrease the anticoagulant activities of Letaxaban.
Darexaban Dydrogesterone may decrease the anticoagulant activities of Darexaban.
Betrixaban Dydrogesterone may decrease the anticoagulant activities of Betrixaban.
Nafamostat Dydrogesterone may decrease the anticoagulant activities of Nafamostat.
Monteplase Dydrogesterone may decrease the anticoagulant activities of Monteplase.
Gabexate Dydrogesterone may decrease the anticoagulant activities of Gabexate.
Protein S human Dydrogesterone may decrease the anticoagulant activities of Protein S human.
Brinase Dydrogesterone may decrease the anticoagulant activities of Brinase.
Tioclomarol Dydrogesterone may decrease the anticoagulant activities of Tioclomarol.
Melagatran Dydrogesterone may decrease the anticoagulant activities of Melagatran.
Saruplase Dydrogesterone may decrease the anticoagulant activities of Saruplase.
(S)-Warfarin Dydrogesterone may decrease the anticoagulant activities of (S)-Warfarin.
Tocopherylquinone Dydrogesterone may decrease the anticoagulant activities of Tocopherylquinone.
Dabigatran Dydrogesterone may decrease the anticoagulant activities of Dabigatran.
Argatroban Dydrogesterone may decrease the anticoagulant activities of Argatroban.
Warfarin Dydrogesterone may decrease the anticoagulant activities of Warfarin.
Phenprocoumon Dydrogesterone may decrease the anticoagulant activities of Phenprocoumon.
Acenocoumarol Dydrogesterone may decrease the anticoagulant activities of Acenocoumarol.
4-hydroxycoumarin Dydrogesterone may decrease the anticoagulant activities of 4-hydroxycoumarin.
Rivaroxaban Dydrogesterone may decrease the anticoagulant activities of Rivaroxaban.
Ethyl biscoumacetate Dydrogesterone may decrease the anticoagulant activities of Ethyl biscoumacetate.
Ticagrelor Dydrogesterone may decrease the anticoagulant activities of Ticagrelor.
Fluindione Dydrogesterone may decrease the anticoagulant activities of Fluindione.
Clorindione Dydrogesterone may decrease the anticoagulant activities of Clorindione.
Diphenadione Dydrogesterone may decrease the anticoagulant activities of Diphenadione.
Troxerutin Dydrogesterone may decrease the anticoagulant activities of Troxerutin.
Edetic acid Dydrogesterone may decrease the anticoagulant activities of Edetic acid.
Reviparin Dydrogesterone may decrease the anticoagulant activities of Reviparin.
Dermatan sulfate Dydrogesterone may decrease the anticoagulant activities of Dermatan sulfate.
SR-123781A Dydrogesterone may decrease the anticoagulant activities of SR-123781A.
Human C1-esterase inhibitor The risk or severity of thromboembolism can be increased when Dydrogesterone is combined with Human C1-esterase inhibitor.
Conestat alfa The risk or severity of thromboembolism can be increased when Dydrogesterone is combined with Conestat alfa.
Lymecycline The serum concentration of Dydrogesterone can be decreased when it is combined with Lymecycline.
Clomocycline The serum concentration of Dydrogesterone can be decreased when it is combined with Clomocycline.
Tigecycline The serum concentration of Dydrogesterone can be decreased when it is combined with Tigecycline.
Oxytetracycline The serum concentration of Dydrogesterone can be decreased when it is combined with Oxytetracycline.
Demeclocycline The serum concentration of Dydrogesterone can be decreased when it is combined with Demeclocycline.
Metacycline The serum concentration of Dydrogesterone can be decreased when it is combined with Metacycline.
Minocycline The serum concentration of Dydrogesterone can be decreased when it is combined with Minocycline.
Rolitetracycline The serum concentration of Dydrogesterone can be decreased when it is combined with Rolitetracycline.
Sarecycline The serum concentration of Dydrogesterone can be decreased when it is combined with Sarecycline.
Omadacycline The serum concentration of Dydrogesterone can be decreased when it is combined with Omadacycline.
Penimepicycline The serum concentration of Dydrogesterone can be decreased when it is combined with Penimepicycline.
Doxycycline The serum concentration of Dydrogesterone can be decreased when it is combined with Doxycycline.
Tetracycline The serum concentration of Dydrogesterone can be decreased when it is combined with Tetracycline.
Eravacycline The serum concentration of Dydrogesterone can be decreased when it is combined with Eravacycline.
Pitolisant The serum concentration of Dydrogesterone can be decreased when it is combined with Pitolisant.

Target Protein

Progesterone receptor PGR

Referensi & Sumber

Synthesis reference: Reerink, E.H., Westerhof, P. and Scholer, H.F.L.; U.S. Patent 3,198,792; assigned to North American Philips Company, Inc.
Link

Contoh Produk & Brand

Produk: 0 • International brands: 4
International Brands
  • Dabroston — Abbott
  • Dufaston — Abbott
  • Duphaston — Abbott
  • Terolut — Solvay

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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