Peringatan Keamanan

Manifestations of acute overdosage of TORECAN (thiethylperazine) can be expected to reflect the CNS effects of the drug and include extrapyramidal symptoms (E.P.S), confusion and convulsions with reduced or absent reflexes, respiratory depression and hypotension.

Thiethylperazine

DB00372

small molecule approved withdrawn

Deskripsi

A dopamine antagonist that is particularly useful in treating the nausea and vomiting associated with anesthesia, mildly emetic cancer chemotherapy agents, radiation therapy, and toxins. This piperazine phenothiazine does not prevent vertigo or motion sickness. (From AMA Drug Evaluations Annual, 1994, p457)

Struktur Molekul 2D

Berat 399.616
Wujud liquid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Thiethylperazine is eliminated in the urine.

Interaksi Makanan

1 Data
  • 1. Avoid excessive or chronic alcohol consumption. Additive CNS depression may occur if alcohol is consumed with thiethylperazine.

Interaksi Obat

1436 Data
Buprenorphine Thiethylperazine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Thiethylperazine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Thiethylperazine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Thiethylperazine.
Hydrocodone Thiethylperazine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Thiethylperazine.
Magnesium sulfate The therapeutic efficacy of Thiethylperazine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Thiethylperazine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Thiethylperazine.
Mirtazapine Thiethylperazine may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Thiethylperazine.
Orphenadrine Thiethylperazine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Thiethylperazine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Thiethylperazine.
Rotigotine Thiethylperazine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Thiethylperazine.
Sodium oxybate Thiethylperazine may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Thiethylperazine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Thiethylperazine.
Thalidomide Thiethylperazine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Thiethylperazine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Amisulpride Thiethylperazine may increase the antipsychotic activities of Amisulpride.
Methylphenidate The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Methylphenidate.
Dexmethylphenidate The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Dexmethylphenidate.
Metoclopramide The risk or severity of adverse effects can be increased when Metoclopramide is combined with Thiethylperazine.
Quinagolide The therapeutic efficacy of Quinagolide can be decreased when used in combination with Thiethylperazine.
Sulpiride Thiethylperazine may increase the antipsychotic activities of Sulpiride.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Thiethylperazine.
Lithium hydroxide Lithium hydroxide may increase the neurotoxic activities of Thiethylperazine.
Lithium citrate Lithium citrate may increase the neurotoxic activities of Thiethylperazine.
Mequitazine Thiethylperazine may increase the arrhythmogenic activities of Mequitazine.
Thiopental The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Thiopental.
Metyrosine The risk or severity of extrapyramidal symptoms and CNS depression can be increased when Metyrosine is combined with Thiethylperazine.
Ethanol Thiethylperazine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Thiethylperazine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Thiethylperazine.
Fluvoxamine The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Escitalopram.
Zimelidine The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Seproxetine.
Levomilnacipran The risk or severity of adverse effects can be increased when Levomilnacipran is combined with Thiethylperazine.
Indalpine The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Thiethylperazine is combined with Alaproclate.
Esmolol The serum concentration of Esmolol can be increased when it is combined with Thiethylperazine.
Betaxolol The serum concentration of Betaxolol can be increased when it is combined with Thiethylperazine.
Metoprolol The serum concentration of Metoprolol can be increased when it is combined with Thiethylperazine.
Atenolol The serum concentration of Atenolol can be increased when it is combined with Thiethylperazine.
Timolol The serum concentration of Timolol can be increased when it is combined with Thiethylperazine.
Sotalol The serum concentration of Sotalol can be increased when it is combined with Thiethylperazine.
Propranolol The serum concentration of Propranolol can be increased when it is combined with Thiethylperazine.
Labetalol The serum concentration of Labetalol can be increased when it is combined with Thiethylperazine.
Bisoprolol The serum concentration of Bisoprolol can be increased when it is combined with Thiethylperazine.
Alprenolol The serum concentration of Alprenolol can be increased when it is combined with Thiethylperazine.
Pindolol The serum concentration of Pindolol can be increased when it is combined with Thiethylperazine.
Carvedilol The serum concentration of Carvedilol can be increased when it is combined with Thiethylperazine.
Propafenone The serum concentration of Propafenone can be increased when it is combined with Thiethylperazine.
Acebutolol The serum concentration of Acebutolol can be increased when it is combined with Thiethylperazine.
Nadolol The serum concentration of Nadolol can be increased when it is combined with Thiethylperazine.
Bevantolol The serum concentration of Bevantolol can be increased when it is combined with Thiethylperazine.
Practolol The serum concentration of Practolol can be increased when it is combined with Thiethylperazine.
Penbutolol The serum concentration of Penbutolol can be increased when it is combined with Thiethylperazine.
Oxprenolol The serum concentration of Oxprenolol can be increased when it is combined with Thiethylperazine.
Dexpropranolol The serum concentration of Dexpropranolol can be increased when it is combined with Thiethylperazine.
Celiprolol The serum concentration of Celiprolol can be increased when it is combined with Thiethylperazine.
Nebivolol The serum concentration of Nebivolol can be increased when it is combined with Thiethylperazine.
Bufuralol The serum concentration of Bufuralol can be increased when it is combined with Thiethylperazine.
Bopindolol The serum concentration of Bopindolol can be increased when it is combined with Thiethylperazine.
Bupranolol The serum concentration of Bupranolol can be increased when it is combined with Thiethylperazine.
Indenolol The serum concentration of Indenolol can be increased when it is combined with Thiethylperazine.
Arotinolol The serum concentration of Arotinolol can be increased when it is combined with Thiethylperazine.
Levobetaxolol The serum concentration of Levobetaxolol can be increased when it is combined with Thiethylperazine.
Talinolol The serum concentration of Talinolol can be increased when it is combined with Thiethylperazine.
Anisodamine The serum concentration of Anisodamine can be increased when it is combined with Thiethylperazine.
Bucindolol The serum concentration of Bucindolol can be increased when it is combined with Thiethylperazine.
Esatenolol The serum concentration of Esatenolol can be increased when it is combined with Thiethylperazine.
Cloranolol The serum concentration of Cloranolol can be increased when it is combined with Thiethylperazine.
Mepindolol The serum concentration of Mepindolol can be increased when it is combined with Thiethylperazine.
Epanolol The serum concentration of Epanolol can be increased when it is combined with Thiethylperazine.
Tertatolol The serum concentration of Tertatolol can be increased when it is combined with Thiethylperazine.
Landiolol The serum concentration of Landiolol can be increased when it is combined with Thiethylperazine.
Morphine The risk or severity of hypotension and CNS depression can be increased when Thiethylperazine is combined with Morphine.
Hydromorphone The risk or severity of hypotension and CNS depression can be increased when Thiethylperazine is combined with Hydromorphone.
Oxycodone The risk or severity of hypotension and CNS depression can be increased when Thiethylperazine is combined with Oxycodone.
Butorphanol The risk or severity of hypotension and CNS depression can be increased when Thiethylperazine is combined with Butorphanol.
Dextropropoxyphene The risk or severity of hypotension and CNS depression can be increased when Thiethylperazine is combined with Dextropropoxyphene.
Pentazocine The risk or severity of hypotension and CNS depression can be increased when Thiethylperazine is combined with Pentazocine.
Naltrexone The risk or severity of hypotension and CNS depression can be increased when Thiethylperazine is combined with Naltrexone.
Sufentanil The risk or severity of hypotension and CNS depression can be increased when Thiethylperazine is combined with Sufentanil.
Alfentanil The risk or severity of hypotension and CNS depression can be increased when Thiethylperazine is combined with Alfentanil.

Target Protein

D(2) dopamine receptor DRD2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 2904251
    Maurer H, Pfleger K: Identification of phenothiazine antihistamines and their metabolites in urine. Arch Toxicol. 1988;62(2-3):185-91.

Contoh Produk & Brand

Produk: 2 • International brands: 0
Produk
  • Torecan
    Tablet • 10 mg/1 • Oral • US • Approved
  • Torecan
    Injection, solution • 10 mg/2mL • Intramuscular • US • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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