Peringatan Keamanan

Symptoms of overdose include coma, drowsiness, loss of muscle control, severely impaired breathing, shock, sluggishness, and unresponsiveness. There have been a case of death resulting from oral ingestion of 12 g of meprobamate. One case study reports the consumption of 40 g of meprobamate resulting in successful survival.

Meprobamate

DB00371

small molecule approved illicit

Deskripsi

A carbamate with hypnotic, sedative, and some muscle relaxant properties, although in therapeutic doses reduction of anxiety rather than a direct effect may be responsible for muscle relaxation. Meprobamate has been reported to have anticonvulsant actions against petit mal seizures, but not against grand mal seizures (which may be exacerbated). It is used in the treatment of anxiety disorders, and also for the short-term management of insomnia but has largely been superseded by the benzodiazepines. (From Martindale, The Extra Pharmacopoeia, 30th ed, p603) Meprobamate is a controlled substance in the U.S.

Struktur Molekul 2D

Berat 218.2502
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Plasma half-life is about 10 hours.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Well absorbed from the gastrointestinal tract.

Metabolisme

Meprobamate undergoes hepatic metabolism.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol.
  • 2. Take with or without food. Food does not significantly affect absorption.

Interaksi Obat

671 Data
Buprenorphine Meprobamate may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Meprobamate.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Meprobamate.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Meprobamate.
Hydrocodone Meprobamate may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Meprobamate.
Magnesium sulfate The therapeutic efficacy of Meprobamate can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Meprobamate may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Meprobamate may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Meprobamate.
Mirtazapine Meprobamate may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Meprobamate.
Orphenadrine Meprobamate may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Meprobamate may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Meprobamate.
Pramipexole Meprobamate may increase the sedative activities of Pramipexole.
Ropinirole Meprobamate may increase the sedative activities of Ropinirole.
Rotigotine Meprobamate may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Meprobamate.
Suvorexant Meprobamate may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Meprobamate.
Thalidomide Meprobamate may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Meprobamate may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Yohimbine The therapeutic efficacy of Meprobamate can be increased when used in combination with Yohimbine.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Meprobamate.
Sodium oxybate Meprobamate may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Ethanol Meprobamate may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Meprobamate may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Meprobamate.
Zimelidine The risk or severity of adverse effects can be increased when Meprobamate is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Meprobamate is combined with Dapoxetine.
Seproxetine The risk or severity of adverse effects can be increased when Meprobamate is combined with Seproxetine.
Fluvoxamine The risk or severity of adverse effects can be increased when Meprobamate is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Meprobamate is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Meprobamate is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Meprobamate is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Meprobamate is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Meprobamate is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Meprobamate is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Meprobamate is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Meprobamate is combined with Escitalopram.
Milnacipran The risk or severity of adverse effects can be increased when Meprobamate is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Meprobamate is combined with Desvenlafaxine.
Levomilnacipran The risk or severity of adverse effects can be increased when Meprobamate is combined with Levomilnacipran.
Indalpine The risk or severity of adverse effects can be increased when Meprobamate is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Meprobamate is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Meprobamate is combined with Alaproclate.
Cyproheptadine The risk or severity of CNS depression can be increased when Meprobamate is combined with Cyproheptadine.
Propiomazine The risk or severity of CNS depression can be increased when Meprobamate is combined with Propiomazine.
Zopiclone The risk or severity of adverse effects can be increased when Meprobamate is combined with Zopiclone.
Botulinum toxin type B The risk or severity of CNS depression can be increased when Botulinum toxin type B is combined with Meprobamate.
Botulinum toxin type A The risk or severity of CNS depression can be increased when Botulinum toxin type A is combined with Meprobamate.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of Meprobamate.
Ethchlorvynol The risk or severity of CNS depression can be increased when Ethchlorvynol is combined with Meprobamate.
Succinylcholine The risk or severity of CNS depression can be increased when Succinylcholine is combined with Meprobamate.
Eletriptan The risk or severity of CNS depression can be increased when Eletriptan is combined with Meprobamate.
Enflurane The risk or severity of CNS depression can be increased when Enflurane is combined with Meprobamate.
Butabarbital The risk or severity of CNS depression can be increased when Butabarbital is combined with Meprobamate.
Butalbital The risk or severity of CNS depression can be increased when Butalbital is combined with Meprobamate.
Methysergide The risk or severity of CNS depression can be increased when Methysergide is combined with Meprobamate.
Cabergoline The risk or severity of CNS depression can be increased when Cabergoline is combined with Meprobamate.
Phenytoin The risk or severity of CNS depression can be increased when Phenytoin is combined with Meprobamate.
Topiramate The risk or severity of CNS depression can be increased when Topiramate is combined with Meprobamate.
Clemastine The risk or severity of CNS depression can be increased when Clemastine is combined with Meprobamate.
Etomidate The risk or severity of CNS depression can be increased when Etomidate is combined with Meprobamate.
Morphine The risk or severity of CNS depression can be increased when Morphine is combined with Meprobamate.
Talbutal The risk or severity of CNS depression can be increased when Talbutal is combined with Meprobamate.
Pentobarbital The risk or severity of CNS depression can be increased when Pentobarbital is combined with Meprobamate.
Zolmitriptan The risk or severity of CNS depression can be increased when Zolmitriptan is combined with Meprobamate.
Dihydroergotamine The risk or severity of CNS depression can be increased when Dihydroergotamine is combined with Meprobamate.
Tolcapone The risk or severity of CNS depression can be increased when Tolcapone is combined with Meprobamate.
Hydromorphone The risk or severity of CNS depression can be increased when Hydromorphone is combined with Meprobamate.
Cetirizine The risk or severity of CNS depression can be increased when Cetirizine is combined with Meprobamate.
Trimethadione The risk or severity of CNS depression can be increased when Trimethadione is combined with Meprobamate.
Chlorzoxazone The risk or severity of CNS depression can be increased when Chlorzoxazone is combined with Meprobamate.
Thiethylperazine The risk or severity of CNS depression can be increased when Meprobamate is combined with Thiethylperazine.
Palonosetron The risk or severity of CNS depression can be increased when Meprobamate is combined with Palonosetron.
Dexbrompheniramine The risk or severity of CNS depression can be increased when Meprobamate is combined with Dexbrompheniramine.
Metocurine iodide The risk or severity of CNS depression can be increased when Meprobamate is combined with Metocurine iodide.
Secobarbital The risk or severity of CNS depression can be increased when Meprobamate is combined with Secobarbital.
Methocarbamol The risk or severity of CNS depression can be increased when Meprobamate is combined with Methocarbamol.
Triprolidine The risk or severity of CNS depression can be increased when Meprobamate is combined with Triprolidine.
Meperidine The risk or severity of CNS depression can be increased when Meprobamate is combined with Meperidine.
Metharbital The risk or severity of CNS depression can be increased when Meprobamate is combined with Metharbital.
Quinine The risk or severity of CNS depression can be increased when Meprobamate is combined with Quinine.
Methohexital The risk or severity of CNS depression can be increased when Meprobamate is combined with Methohexital.
Gallamine triethiodide The risk or severity of CNS depression can be increased when Meprobamate is combined with Gallamine triethiodide.
Entacapone The risk or severity of CNS depression can be increased when Meprobamate is combined with Entacapone.
Oxycodone The risk or severity of CNS depression can be increased when Meprobamate is combined with Oxycodone.
Dextromethorphan The risk or severity of CNS depression can be increased when Meprobamate is combined with Dextromethorphan.
Mephenytoin The risk or severity of CNS depression can be increased when Meprobamate is combined with Mephenytoin.
Cisatracurium The risk or severity of CNS depression can be increased when Meprobamate is combined with Cisatracurium.
Fenfluramine The risk or severity of CNS depression can be increased when Meprobamate is combined with Fenfluramine.
Mazindol The risk or severity of CNS depression can be increased when Meprobamate is combined with Mazindol.
Fluticasone propionate The risk or severity of CNS depression can be increased when Meprobamate is combined with Fluticasone propionate.
Lisuride The risk or severity of CNS depression can be increased when Meprobamate is combined with Lisuride.
Ethosuximide The risk or severity of CNS depression can be increased when Meprobamate is combined with Ethosuximide.
Thiopental The risk or severity of CNS depression can be increased when Meprobamate is combined with Thiopental.
Cisapride The risk or severity of CNS depression can be increased when Meprobamate is combined with Cisapride.
Butorphanol The risk or severity of CNS depression can be increased when Meprobamate is combined with Butorphanol.

Target Protein

Peptide deformylase, mitochondrial PDF
Protein kinase C epsilon type PRKCE
GABA(A) Receptor GABRA1
Gamma-aminobutyric acid receptor subunit alpha-1 GABRA1
Gamma-aminobutyric acid receptor subunit alpha-2 GABRA2
Gamma-aminobutyric acid receptor subunit alpha-3 GABRA3
Gamma-aminobutyric acid receptor subunit alpha-4 GABRA4
Gamma-aminobutyric acid receptor subunit alpha-5 GABRA5
Gamma-aminobutyric acid receptor subunit alpha-6 GABRA6

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 27 • International brands: 3
Produk
  • 282 Mep Tab
    Tablet • - • Oral • Canada • Approved
  • Apo Meprobamate Tab 400mg
    Tablet • 400 mg / tab • Oral • Canada • Generic • Approved
  • Equagesic
    Tablet • - • Oral • US • Approved
  • Equagesic Tablets
    Tablet • - • Oral • Canada • Approved
  • Equanil Tablets 400mg
    Tablet • 400 mg / tab • Oral • Canada • Approved
  • Meditran 400mg
    Tablet • 400 mg • Oral • Canada • Approved
  • Meprobamate
    Tablet • 200 mg/1 • Oral • US • Generic • Approved
  • Meprobamate
    Tablet • 400 mg/1 • Oral • US • Generic • Approved
Menampilkan 8 dari 27 produk.
International Brands
  • Equanil — Wyeth
  • Meprospan
  • Miltown — Wallace Laboratories

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul