Sapropterin

DB00360

small molecule approved investigational

Deskripsi

Sapropterin (tetrahydrobiopterin or BH4) is a cofactor in the synthesis of nitric oxide. It is also essential in the conversion of phenylalanine to tyrosine by the enzyme phenylalanine-4-hydroxylase; the conversion of tyrosine to L-dopa by the enzyme tyrosine hydroxylase; and conversion of tryptophan to 5-hydroxytryptophan via tryptophan hydroxylase.

Struktur Molekul 2D

Berat 241.2471
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Take at the same time every day.
  • 2. Take with food. Taking sapropterin with food increases oral absorption. Sapropterin may be dissolved in water, juice, or dispersed in applesauce.

Interaksi Obat

170 Data
Afatinib The serum concentration of Afatinib can be increased when it is combined with Sapropterin.
Bosutinib The serum concentration of Bosutinib can be increased when it is combined with Sapropterin.
Brentuximab vedotin The serum concentration of Brentuximab vedotin can be increased when it is combined with Sapropterin.
Colchicine The serum concentration of Colchicine can be increased when it is combined with Sapropterin.
Edoxaban The serum concentration of Edoxaban can be increased when it is combined with Sapropterin.
Ledipasvir The serum concentration of Ledipasvir can be increased when it is combined with Sapropterin.
Naloxegol The serum concentration of Naloxegol can be increased when it is combined with Sapropterin.
Pazopanib The serum concentration of Pazopanib can be increased when it is combined with Sapropterin.
Prucalopride The serum concentration of Prucalopride can be increased when it is combined with Sapropterin.
Ranolazine The serum concentration of Ranolazine can be increased when it is combined with Sapropterin.
Silodosin The excretion of Silodosin can be decreased when combined with Sapropterin.
Topotecan The serum concentration of Topotecan can be increased when it is combined with Sapropterin.
Everolimus The serum concentration of Everolimus can be increased when it is combined with Sapropterin.
Rifaximin The serum concentration of Rifaximin can be increased when it is combined with Sapropterin.
Levodopa The risk or severity of adverse effects can be increased when Sapropterin is combined with Levodopa.
Methotrexate The serum concentration of Sapropterin can be decreased when it is combined with Methotrexate.
Pralatrexate The serum concentration of Sapropterin can be decreased when it is combined with Pralatrexate.
Sildenafil Sapropterin may increase the hypotensive activities of Sildenafil.
Tadalafil Sapropterin may increase the hypotensive activities of Tadalafil.
Vardenafil Sapropterin may increase the hypotensive activities of Vardenafil.
Udenafil Sapropterin may increase the hypotensive activities of Udenafil.
Mirodenafil Sapropterin may increase the hypotensive activities of Mirodenafil.
Avanafil Sapropterin may increase the hypotensive activities of Avanafil.
Dipyridamole Sapropterin may increase the hypotensive activities of Dipyridamole.
Fostamatinib Sapropterin may increase the hypotensive activities of Fostamatinib.
Ibudilast Sapropterin may increase the hypotensive activities of Ibudilast.
Doxofylline Sapropterin may increase the hypotensive activities of Doxofylline.
Vincristine The excretion of Vincristine can be decreased when combined with Sapropterin.
Doxorubicin The serum concentration of Doxorubicin can be increased when it is combined with Sapropterin.
Betrixaban The serum concentration of Betrixaban can be increased when it is combined with Sapropterin.
Daptomycin The serum concentration of Daptomycin can be increased when it is combined with Sapropterin.
Pravastatin The serum concentration of Pravastatin can be increased when it is combined with Sapropterin.
Morphine The serum concentration of Morphine can be increased when it is combined with Sapropterin.
Tenofovir disoproxil The serum concentration of Tenofovir disoproxil can be increased when it is combined with Sapropterin.
Clobazam The serum concentration of Clobazam can be increased when it is combined with Sapropterin.
Mefloquine The serum concentration of Mefloquine can be increased when it is combined with Sapropterin.
Quinine The serum concentration of Quinine can be increased when it is combined with Sapropterin.
Toremifene The serum concentration of Toremifene can be increased when it is combined with Sapropterin.
Bisoprolol The serum concentration of Bisoprolol can be increased when it is combined with Sapropterin.
Simvastatin The serum concentration of Simvastatin can be increased when it is combined with Sapropterin.
Mannitol The serum concentration of Mannitol can be increased when it is combined with Sapropterin.
Loperamide The excretion of Loperamide can be decreased when combined with Sapropterin.
Clomifene The serum concentration of Clomifene can be increased when it is combined with Sapropterin.
Tipranavir The serum concentration of Tipranavir can be increased when it is combined with Sapropterin.
Fexofenadine The serum concentration of Fexofenadine can be increased when it is combined with Sapropterin.
Tegaserod The serum concentration of Tegaserod can be increased when it is combined with Sapropterin.
Saquinavir The serum concentration of Saquinavir can be increased when it is combined with Sapropterin.
Sitagliptin The serum concentration of Sitagliptin can be increased when it is combined with Sapropterin.
Posaconazole The serum concentration of Posaconazole can be increased when it is combined with Sapropterin.
Darunavir The serum concentration of Darunavir can be increased when it is combined with Sapropterin.
Paliperidone The serum concentration of Paliperidone can be increased when it is combined with Sapropterin.
Mibefradil The serum concentration of Mibefradil can be increased when it is combined with Sapropterin.
Belinostat The serum concentration of Belinostat can be increased when it is combined with Sapropterin.
Indacaterol The serum concentration of Indacaterol can be increased when it is combined with Sapropterin.
Telaprevir The serum concentration of Telaprevir can be increased when it is combined with Sapropterin.
Rivaroxaban The serum concentration of Rivaroxaban can be increased when it is combined with Sapropterin.
Simeprevir The serum concentration of Simeprevir can be increased when it is combined with Sapropterin.
Ambrisentan The serum concentration of Ambrisentan can be increased when it is combined with Sapropterin.
Cethromycin The serum concentration of Cethromycin can be increased when it is combined with Sapropterin.
Apixaban The serum concentration of Apixaban can be increased when it is combined with Sapropterin.
Odanacatib The serum concentration of Odanacatib can be increased when it is combined with Sapropterin.
Ticagrelor The serum concentration of Ticagrelor can be increased when it is combined with Sapropterin.
Linagliptin The serum concentration of Linagliptin can be increased when it is combined with Sapropterin.
Mirabegron The serum concentration of Mirabegron can be increased when it is combined with Sapropterin.
Canagliflozin The serum concentration of Canagliflozin can be increased when it is combined with Sapropterin.
Dolutegravir The serum concentration of Dolutegravir can be increased when it is combined with Sapropterin.
Sofosbuvir The serum concentration of Sofosbuvir can be increased when it is combined with Sapropterin.
Idelalisib The serum concentration of Idelalisib can be increased when it is combined with Sapropterin.
Umeclidinium The serum concentration of Umeclidinium can be increased when it is combined with Sapropterin.
Lenvatinib The serum concentration of Lenvatinib can be increased when it is combined with Sapropterin.
Nintedanib The serum concentration of Nintedanib can be increased when it is combined with Sapropterin.
Technetium Tc-99m sestamibi The serum concentration of Technetium Tc-99m sestamibi can be increased when it is combined with Sapropterin.
Dasabuvir The serum concentration of Dasabuvir can be increased when it is combined with Sapropterin.
Methylene blue The serum concentration of Methylene blue can be increased when it is combined with Sapropterin.
Ombitasvir The serum concentration of Ombitasvir can be increased when it is combined with Sapropterin.
Paritaprevir The serum concentration of Paritaprevir can be increased when it is combined with Sapropterin.
Selexipag The serum concentration of Selexipag can be increased when it is combined with Sapropterin.
Elbasvir The serum concentration of Elbasvir can be increased when it is combined with Sapropterin.
Grazoprevir The serum concentration of Grazoprevir can be increased when it is combined with Sapropterin.
Velpatasvir The serum concentration of Velpatasvir can be increased when it is combined with Sapropterin.
Tucatinib The serum concentration of Tucatinib can be increased when it is combined with Sapropterin.
Selumetinib The serum concentration of Selumetinib can be increased when it is combined with Sapropterin.
Voclosporin The serum concentration of Voclosporin can be increased when it is combined with Sapropterin.
Tezacaftor The serum concentration of Tezacaftor can be increased when it is combined with Sapropterin.
Lasmiditan The serum concentration of Lasmiditan can be increased when it is combined with Sapropterin.
Talinolol The serum concentration of Talinolol can be increased when it is combined with Sapropterin.
Fostemsavir The serum concentration of Fostemsavir can be increased when it is combined with Sapropterin.
Revefenacin The serum concentration of Revefenacin can be increased when it is combined with Sapropterin.
Valspodar The serum concentration of Valspodar can be increased when it is combined with Sapropterin.
Lemborexant The serum concentration of Lemborexant can be increased when it is combined with Sapropterin.
Duvelisib The serum concentration of Duvelisib can be increased when it is combined with Sapropterin.
Glasdegib The serum concentration of Glasdegib can be increased when it is combined with Sapropterin.
Elagolix The serum concentration of Elagolix can be increased when it is combined with Sapropterin.
Voxilaprevir The serum concentration of Voxilaprevir can be increased when it is combined with Sapropterin.
Gilteritinib The serum concentration of Gilteritinib can be increased when it is combined with Sapropterin.
Omadacycline The serum concentration of Omadacycline can be increased when it is combined with Sapropterin.
Fedratinib The serum concentration of Fedratinib can be increased when it is combined with Sapropterin.
Grapiprant The serum concentration of Grapiprant can be increased when it is combined with Sapropterin.
Tazemetostat The serum concentration of Tazemetostat can be increased when it is combined with Sapropterin.
Darolutamide The serum concentration of Darolutamide can be increased when it is combined with Sapropterin.

Target Protein

Phenylalanine-4-hydroxylase PAH
Nitric oxide synthase 3 NOS3
Tyrosine 3-monooxygenase TH
Tryptophan 5-hydroxylase 1 TPH1

Referensi & Sumber

Synthesis reference: Steven S. Gross, "Blocking utilization of tetrahydrobiopterin to block induction of nitric oxide synthesis." U.S. Patent US5502050, issued October, 1984.
Artikel (PubMed)
  • PMID: 10727395
    Thony B, Auerbach G, Blau N: Tetrahydrobiopterin biosynthesis, regeneration and functions. Biochem J. 2000 Apr 1;347 Pt 1:1-16.

Contoh Produk & Brand

Produk: 32 • International brands: 2
Produk
  • Javygtor
    Powder, for solution • 100 mg/1 • Oral • US • Generic • Approved
  • Javygtor
    Tablet • 100 mg/1 • Oral • US • Generic • Approved
  • Javygtor
    Powder, for solution • 500 mg/1 • Oral • US • Generic • Approved
  • Kuvan
    Tablet • 100 mg/1 • Oral • US • Approved
  • Kuvan
    Powder, for solution • 100 mg/1 • Oral • US • Approved
  • Kuvan
    Powder, for solution • 500 mg/1 • Oral • US • Approved
  • Kuvan
    Tablet • 100 mg • Oral • Canada • Approved
  • Kuvan
    Powder • 100 mg / sachet • Oral • Canada • Approved
Menampilkan 8 dari 32 produk.
International Brands
  • BH4 — Excelsior
  • Biopten — Daiichi Sankyo

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul