Peringatan Keamanan

Side effects include anxiety, blood disorders, confusion, decreased libido, dizziness, flushing, headache, impotence, insomnia, low blood pressure, nightmares, rapid or irregular heartbeat, rash, seizures, sensitivity to sunlight, stomach and intestinal discomfort, sedation, hypotension, blurred vision, dry mouth, constipation, urinary retention, postural hypotension, tachycardia, hypertension, ECG changes, heart failure, impaired memory and delirium, and precipitation of hypomanic or manic episodes in bipolar depression. Withdrawal symptoms include gastrointestinal disturbances, anxiety, and insomnia.

Protriptyline

DB00344

small molecule approved

Deskripsi

Protriptyline hydrochloride is a dibenzocycloheptene-derivative tricyclic antidepressant (TCA). TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-depressed individuals, protriptyline does not affect mood or arousal, but may cause sedation. In depressed individuals, protriptyline exerts a positive effect on mood. TCAs are potent inhibitors of serotonin and norepinephrine reuptake. In addition, TCAs down-regulate cerebral cortical β-adrenergic receptors and sensitize post-synaptic serotonergic receptors with chronic use. The antidepressant effects of TCAs are thought to be due to an overall increase in serotonergic neurotransmission. TCAs also block histamine H1 receptors, alpha1-adrenergic receptors and muscarinic receptors, which accounts for their sedative, hypotensive and anticholinergic effects (e.g. blurred vision, dry mouth, constipation, urinary retention), respectively. See toxicity section below for a complete listing of side effects. Protriptyline may be used for the treatment of depression.

Struktur Molekul 2D

Berat 263.3767
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Protriptyline is reported to undergo cumulative urinary excretion during 16 days, which accounts for approximately 50% of the total drug administered. The fecal excretion pathway seems to play a minimal role in drug elimination.

Interaksi Obat

1558 Data
Valsartan Protriptyline may decrease the antihypertensive activities of Valsartan.
Ramipril Protriptyline may decrease the antihypertensive activities of Ramipril.
Remikiren Protriptyline may decrease the antihypertensive activities of Remikiren.
Torasemide Protriptyline may decrease the antihypertensive activities of Torasemide.
Guanadrel Protriptyline may decrease the antihypertensive activities of Guanadrel.
Olmesartan Protriptyline may decrease the antihypertensive activities of Olmesartan.
Chlorthalidone Protriptyline may decrease the antihypertensive activities of Chlorthalidone.
Nitroprusside Protriptyline may decrease the antihypertensive activities of Nitroprusside.
Minoxidil Protriptyline may decrease the antihypertensive activities of Minoxidil.
Nisoldipine Protriptyline may decrease the antihypertensive activities of Nisoldipine.
Bendroflumethiazide Protriptyline may decrease the antihypertensive activities of Bendroflumethiazide.
Fosinopril Protriptyline may decrease the antihypertensive activities of Fosinopril.
Trandolapril Protriptyline may decrease the antihypertensive activities of Trandolapril.
Metolazone Protriptyline may decrease the antihypertensive activities of Metolazone.
Benazepril Protriptyline may decrease the antihypertensive activities of Benazepril.
Bosentan Protriptyline may decrease the antihypertensive activities of Bosentan.
Enalapril Protriptyline may decrease the antihypertensive activities of Enalapril.
Cyclothiazide Protriptyline may decrease the antihypertensive activities of Cyclothiazide.
Candoxatril Protriptyline may decrease the antihypertensive activities of Candoxatril.
Eplerenone Protriptyline may decrease the antihypertensive activities of Eplerenone.
Lisinopril Protriptyline may decrease the antihypertensive activities of Lisinopril.
Nitroglycerin Protriptyline may decrease the antihypertensive activities of Nitroglycerin.
Hydroflumethiazide Protriptyline may decrease the antihypertensive activities of Hydroflumethiazide.
Cryptenamine Protriptyline may decrease the antihypertensive activities of Cryptenamine.
Perindopril Protriptyline may decrease the antihypertensive activities of Perindopril.
Candesartan cilexetil Protriptyline may decrease the antihypertensive activities of Candesartan cilexetil.
Fenoldopam Protriptyline may decrease the antihypertensive activities of Fenoldopam.
Tadalafil Protriptyline may decrease the antihypertensive activities of Tadalafil.
Eprosartan Protriptyline may decrease the antihypertensive activities of Eprosartan.
Chlorothiazide Protriptyline may decrease the antihypertensive activities of Chlorothiazide.
Quinapril Protriptyline may decrease the antihypertensive activities of Quinapril.
Telmisartan Protriptyline may decrease the antihypertensive activities of Telmisartan.
Trichlormethiazide Protriptyline may decrease the antihypertensive activities of Trichlormethiazide.
Irbesartan Protriptyline may decrease the antihypertensive activities of Irbesartan.
Deserpidine Protriptyline may decrease the antihypertensive activities of Deserpidine.
Diazoxide Protriptyline may decrease the antihypertensive activities of Diazoxide.
Terazosin Protriptyline may decrease the antihypertensive activities of Terazosin.
Guanethidine Protriptyline may decrease the antihypertensive activities of Guanethidine.
Epoprostenol Protriptyline may decrease the antihypertensive activities of Epoprostenol.
Hydralazine Protriptyline may decrease the antihypertensive activities of Hydralazine.
Polythiazide Protriptyline may decrease the antihypertensive activities of Polythiazide.
Cilazapril Protriptyline may decrease the antihypertensive activities of Cilazapril.
Saprisartan Protriptyline may decrease the antihypertensive activities of Saprisartan.
Spirapril Protriptyline may decrease the antihypertensive activities of Spirapril.
Dexpropranolol Protriptyline may decrease the antihypertensive activities of Dexpropranolol.
Tienilic acid Protriptyline may decrease the antihypertensive activities of Tienilic acid.
Sitaxentan Protriptyline may decrease the antihypertensive activities of Sitaxentan.
Diethylnorspermine Protriptyline may decrease the antihypertensive activities of Diethylnorspermine.
Pinacidil Protriptyline may decrease the antihypertensive activities of Pinacidil.
Temocapril Protriptyline may decrease the antihypertensive activities of Temocapril.
Riociguat Protriptyline may decrease the antihypertensive activities of Riociguat.
Macitentan Protriptyline may decrease the antihypertensive activities of Macitentan.
Aliskiren Protriptyline may decrease the antihypertensive activities of Aliskiren.
Trimazosin Protriptyline may decrease the antihypertensive activities of Trimazosin.
Rauwolfia serpentina root Protriptyline may decrease the antihypertensive activities of Rauwolfia serpentina root.
Enalaprilat Protriptyline may decrease the antihypertensive activities of Enalaprilat.
Angiotensin 1-7 Protriptyline may decrease the antihypertensive activities of Angiotensin 1-7.
Imidapril Protriptyline may decrease the antihypertensive activities of Imidapril.
BQ-123 Protriptyline may decrease the antihypertensive activities of BQ-123.
Dihydralazine Protriptyline may decrease the antihypertensive activities of Dihydralazine.
Zofenopril Protriptyline may decrease the antihypertensive activities of Zofenopril.
Guanoxan Protriptyline may decrease the antihypertensive activities of Guanoxan.
Delapril Protriptyline may decrease the antihypertensive activities of Delapril.
Vincamine Protriptyline may decrease the antihypertensive activities of Vincamine.
Linsidomine Protriptyline may decrease the antihypertensive activities of Linsidomine.
Guanoxabenz Protriptyline may decrease the antihypertensive activities of Guanoxabenz.
Tolonidine Protriptyline may decrease the antihypertensive activities of Tolonidine.
Endralazine Protriptyline may decrease the antihypertensive activities of Endralazine.
Cadralazine Protriptyline may decrease the antihypertensive activities of Cadralazine.
Cyclopenthiazide Protriptyline may decrease the antihypertensive activities of Cyclopenthiazide.
Bietaserpine Protriptyline may decrease the antihypertensive activities of Bietaserpine.
Guanazodine Protriptyline may decrease the antihypertensive activities of Guanazodine.
Methoserpidine Protriptyline may decrease the antihypertensive activities of Methoserpidine.
Guanoclor Protriptyline may decrease the antihypertensive activities of Guanoclor.
Muzolimine Protriptyline may decrease the antihypertensive activities of Muzolimine.
Xipamide Protriptyline may decrease the antihypertensive activities of Xipamide.
Candesartan Protriptyline may decrease the antihypertensive activities of Candesartan.
Dexniguldipine Protriptyline may decrease the antihypertensive activities of Dexniguldipine.
Tocopherylquinone Protriptyline may decrease the antihypertensive activities of Tocopherylquinone.
Benazeprilat Protriptyline may decrease the antihypertensive activities of Benazeprilat.
Fosinoprilat Protriptyline may decrease the antihypertensive activities of Fosinoprilat.
Ramiprilat Protriptyline may decrease the antihypertensive activities of Ramiprilat.
Perindoprilat Protriptyline may decrease the antihypertensive activities of Perindoprilat.
Quinaprilat Protriptyline may decrease the antihypertensive activities of Quinaprilat.
Furosemide Protriptyline may decrease the antihypertensive activities of Furosemide.
Captopril Protriptyline may decrease the antihypertensive activities of Captopril.
Prazosin Protriptyline may decrease the antihypertensive activities of Prazosin.
Bisoprolol Protriptyline may decrease the antihypertensive activities of Bisoprolol.
Ambrisentan Protriptyline may decrease the antihypertensive activities of Ambrisentan.
Selexipag Protriptyline may decrease the antihypertensive activities of Selexipag.
Atenolol Protriptyline may decrease the antihypertensive activities of Atenolol.
Amlodipine Protriptyline may decrease the antihypertensive activities of Amlodipine.
Doxazosin Protriptyline may decrease the antihypertensive activities of Doxazosin.
Carvedilol Protriptyline may decrease the antihypertensive activities of Carvedilol.
Nadolol Protriptyline may decrease the antihypertensive activities of Nadolol.
Bevantolol Protriptyline may decrease the antihypertensive activities of Bevantolol.
Practolol Protriptyline may decrease the antihypertensive activities of Practolol.
Debrisoquine Protriptyline may decrease the antihypertensive activities of Debrisoquine.
Landiolol Protriptyline may decrease the antihypertensive activities of Landiolol.
Esatenolol Protriptyline may decrease the antihypertensive activities of Esatenolol.

Target Protein

Sodium-dependent noradrenaline transporter SLC6A2
Sodium-dependent serotonin transporter SLC6A4

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 16 • International brands: 1
Produk
  • Protriptyline Hydrochloride
    Tablet, film coated • 5 mg/1 • Oral • US • Generic • Approved
  • Protriptyline Hydrochloride
    Tablet, film coated • 10 mg/1 • Oral • US • Generic • Approved
  • Protriptyline Hydrochloride
    Tablet • 5 mg/1 • Oral • US • Generic • Approved
  • Protriptyline Hydrochloride
    Tablet • 10 mg/1 • Oral • US • Generic • Approved
  • Protriptyline hydrochloride
    Tablet, film coated • 5 mg/1 • Oral • US • Generic • Approved
  • Protriptyline hydrochloride
    Tablet, film coated • 10 mg/1 • Oral • US • Generic • Approved
  • Protriptyline Hydrochloride
    Tablet, film coated • 5 mg/1 • Oral • US • Generic • Approved
  • Protriptyline Hydrochloride
    Tablet, film coated • 10 mg/1 • Oral • US • Generic • Approved
Menampilkan 8 dari 16 produk.
International Brands
  • Triptil

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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