Peringatan Keamanan

Symptoms of an overdose typically include sluggishness, incoordination, difficulty in thinking, slowness of speech, faulty judgment, drowsiness or coma, shallow breathing, staggering, and in severe cases coma and death.

Pentobarbital

DB00312

small molecule approved investigational vet_approved

Deskripsi

A short-acting barbiturate that is effective as a sedative and hypnotic (but not as an anti-anxiety) agent and is usually given orally. It is prescribed more frequently for sleep induction than for sedation but, like similar agents, may lose its effectiveness by the second week of continued administration. (From AMA Drug Evaluations Annual, 1994, p236)

Struktur Molekul 2D

Berat 226.2722
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 5 to 50 hours (dose dependent)
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Barbiturates are absorbed in varying degrees following oral, rectal, or parenteral administration.

Metabolisme

by hepatic microsomal enzyme system

Rute Eliminasi

Barbiturates are metabolized primarily by the hepatic microsomal enzyme system, and the metabolic products are excreted in the urine, and less commonly, in the feces. Approximately 25 to 50 percent of a dose of aprobarbital or phenobarbital is eliminated unchanged in the urine, whereas the amount of other barbiturates excreted unchanged in the urine is negligible.

Interaksi Obat

2134 Data
Aripiprazole The metabolism of Aripiprazole can be increased when combined with Pentobarbital.
Buprenorphine Pentobarbital may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Pentobarbital.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Pentobarbital.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Pentobarbital.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Pentobarbital.
Magnesium sulfate The therapeutic efficacy of Pentobarbital can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Pentobarbital may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Pentobarbital may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Pentobarbital.
Mirtazapine Pentobarbital may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Pentobarbital.
Orphenadrine Pentobarbital may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Pentobarbital may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Pramipexole Pentobarbital may increase the sedative activities of Pramipexole.
Ropinirole Pentobarbital may increase the sedative activities of Ropinirole.
Rotigotine Pentobarbital may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Pentobarbital.
Suvorexant Pentobarbital may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Pentobarbital.
Thalidomide Pentobarbital may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Pentobarbital may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Dabrafenib The serum concentration of Pentobarbital can be decreased when it is combined with Dabrafenib.
Secretin porcine The therapeutic efficacy of Secretin porcine can be decreased when used in combination with Pentobarbital.
Luliconazole The serum concentration of Pentobarbital can be increased when it is combined with Luliconazole.
Mefloquine The therapeutic efficacy of Pentobarbital can be decreased when used in combination with Mefloquine.
Orlistat Orlistat can cause a decrease in the absorption of Pentobarbital resulting in a reduced serum concentration and potentially a decrease in efficacy.
Chloramphenicol The metabolism of Pentobarbital can be decreased when combined with Chloramphenicol.
Doxycycline The serum concentration of Doxycycline can be decreased when it is combined with Pentobarbital.
Felbamate The serum concentration of Pentobarbital can be increased when it is combined with Felbamate.
Griseofulvin The serum concentration of Griseofulvin can be decreased when it is combined with Pentobarbital.
Lamotrigine The serum concentration of Lamotrigine can be decreased when it is combined with Pentobarbital.
Mianserin The therapeutic efficacy of Pentobarbital can be decreased when used in combination with Mianserin.
Primidone The risk or severity of adverse effects can be increased when Primidone is combined with Pentobarbital.
Methylphenobarbital The risk or severity of adverse effects can be increased when Methylphenobarbital is combined with Pentobarbital.
Phenobarbital The risk or severity of adverse effects can be increased when Phenobarbital is combined with Pentobarbital.
Pyridoxine The metabolism of Pentobarbital can be increased when combined with Pyridoxine.
Teniposide The serum concentration of Teniposide can be decreased when it is combined with Pentobarbital.
Voriconazole The serum concentration of Voriconazole can be decreased when it is combined with Pentobarbital.
Topotecan Pentobarbital may increase the excretion rate of Topotecan which could result in a lower serum level and potentially a reduction in efficacy.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Pentobarbital.
Sodium oxybate Pentobarbital may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Ifosfamide The metabolism of Ifosfamide can be increased when combined with Pentobarbital.
Perampanel The metabolism of Perampanel can be increased when combined with Pentobarbital.
Warfarin The metabolism of Warfarin can be increased when combined with Pentobarbital.
Acenocoumarol The metabolism of Acenocoumarol can be increased when combined with Pentobarbital.
(R)-warfarin The metabolism of (R)-warfarin can be increased when combined with Pentobarbital.
R,S-Warfarin alcohol The metabolism of R,S-Warfarin alcohol can be increased when combined with Pentobarbital.
S,R-Warfarin alcohol The metabolism of S,R-Warfarin alcohol can be increased when combined with Pentobarbital.
(S)-Warfarin The metabolism of (S)-Warfarin can be increased when combined with Pentobarbital.
Tetracosactide The risk or severity of liver damage can be increased when Tetracosactide is combined with Pentobarbital.
Aminophylline The therapeutic efficacy of Pentobarbital can be decreased when used in combination with Aminophylline.
Botulinum toxin type A The risk or severity of adverse effects can be increased when Pentobarbital is combined with Botulinum toxin type A.
Botulinum toxin type B The risk or severity of adverse effects can be increased when Pentobarbital is combined with Botulinum toxin type B.
Meperidine Pentobarbital may increase the hypotensive and central nervous system depressant (CNS depressant) activities of Meperidine.
Somatostatin The risk or severity of adverse effects can be increased when Somatostatin is combined with Pentobarbital.
Ethanol Pentobarbital may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Pentobarbital may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Pentobarbital.
Zimelidine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Zimelidine.
Seproxetine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Seproxetine.
Ritanserin The risk or severity of adverse effects can be increased when Pentobarbital is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Pentobarbital is combined with Alaproclate.
Duloxetine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Duloxetine.
Naltrexone The risk or severity of adverse effects can be increased when Pentobarbital is combined with Naltrexone.
Bezitramide The risk or severity of adverse effects can be increased when Pentobarbital is combined with Bezitramide.
Butorphanol The risk or severity of adverse effects can be increased when Pentobarbital is combined with Butorphanol.
Pentazocine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Pentazocine.
Nalbuphine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Nalbuphine.
Levorphanol The risk or severity of adverse effects can be increased when Pentobarbital is combined with Levorphanol.
Remifentanil The risk or severity of adverse effects can be increased when Pentobarbital is combined with Remifentanil.
Diphenoxylate The risk or severity of adverse effects can be increased when Pentobarbital is combined with Diphenoxylate.
Dezocine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Dezocine.
Methadyl acetate The risk or severity of adverse effects can be increased when Pentobarbital is combined with Methadyl acetate.
Dihydroetorphine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Dihydroetorphine.
Diamorphine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Diamorphine.
Etorphine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Etorphine.
Dextromoramide The risk or severity of adverse effects can be increased when Pentobarbital is combined with Dextromoramide.
Desomorphine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Desomorphine.
Carfentanil The risk or severity of adverse effects can be increased when Pentobarbital is combined with Carfentanil.
Alphacetylmethadol The risk or severity of adverse effects can be increased when Pentobarbital is combined with Alphacetylmethadol.
Dihydromorphine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Dihydromorphine.
DPDPE The risk or severity of adverse effects can be increased when Pentobarbital is combined with DPDPE.
Lofentanil The risk or severity of adverse effects can be increased when Pentobarbital is combined with Lofentanil.
Normethadone The risk or severity of adverse effects can be increased when Pentobarbital is combined with Normethadone.
Piritramide The risk or severity of adverse effects can be increased when Pentobarbital is combined with Piritramide.
Alphaprodine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Alphaprodine.
Nicomorphine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Nicomorphine.
Meptazinol The risk or severity of adverse effects can be increased when Pentobarbital is combined with Meptazinol.
Phenoperidine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Phenoperidine.
Phenazocine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Phenazocine.
Tilidine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Tilidine.
Carfentanil, C-11 The risk or severity of adverse effects can be increased when Pentobarbital is combined with Carfentanil, C-11.
Alfentanil The risk or severity of adverse effects can be increased when Pentobarbital is combined with Alfentanil.
Fentanyl The risk or severity of adverse effects can be increased when Pentobarbital is combined with Fentanyl.
Levacetylmethadol The risk or severity of adverse effects can be increased when Pentobarbital is combined with Levacetylmethadol.
Benzhydrocodone The risk or severity of adverse effects can be increased when Pentobarbital is combined with Benzhydrocodone.
Hydromorphone The risk or severity of adverse effects can be increased when Pentobarbital is combined with Hydromorphone.
Morphine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Morphine.
Codeine The risk or severity of adverse effects can be increased when Pentobarbital is combined with Codeine.

Target Protein

Gamma-aminobutyric acid receptor subunit alpha-1 GABRA1
Gamma-aminobutyric acid receptor subunit alpha-2 GABRA2
Gamma-aminobutyric acid receptor subunit alpha-3 GABRA3
Gamma-aminobutyric acid receptor subunit alpha-4 GABRA4
Gamma-aminobutyric acid receptor subunit alpha-5 GABRA5
Gamma-aminobutyric acid receptor subunit alpha-6 GABRA6
GABA(A) Receptor GABRA1
Neuronal acetylcholine receptor subunit alpha-4 CHRNA4
Neuronal acetylcholine receptor subunit alpha-7 CHRNA7
Glutamate receptor 2 GRIA2
Glutamate receptor ionotropic, kainate 2 GRIK2
NMDA receptor GRIN1
Nuclear receptor subfamily 1 group I member 2 NR1I2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 6777235
    Knodell RG, Spector MH, Brooks DA, Keller FX, Kyner WT: Alterations in pentobarbital pharmacokinetics in response to parenteral and enteral alimentation in the rat. Gastroenterology. 1980 Dec;79(6):1211-6.

Contoh Produk & Brand

Produk: 14 • International brands: 1
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Menampilkan 8 dari 14 produk.
International Brands
  • Nembutal — Lundbeck

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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