Ethoxzolamide

DB00311

small molecule withdrawn

Deskripsi

Ethoxzolamide is a sulfonamide used as diuretic and in glaucoma. It inhibits carbonic anhydrase activity in proximal renal tubules to decrease reabsorption of water, sodium, potassium, bicarbonate. Its pharmacological activity thus confers the risk for hypokalemia.

Struktur Molekul 2D

Berat 258.317
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 2.5-5.5 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Rapidly absorbed with 65% bioavailability

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

788 Data
Nicotine The risk or severity of adverse effects can be increased when Ethoxzolamide is combined with Nicotine.
Mecamylamine The risk or severity of adverse effects can be increased when Ethoxzolamide is combined with Mecamylamine.
Pentolinium The risk or severity of adverse effects can be increased when Ethoxzolamide is combined with Pentolinium.
Trimethaphan The risk or severity of adverse effects can be increased when Ethoxzolamide is combined with Trimethaphan.
Hexamethonium The risk or severity of adverse effects can be increased when Ethoxzolamide is combined with Hexamethonium.
Cyclopentamine The risk or severity of adverse effects can be increased when Ethoxzolamide is combined with Cyclopentamine.
Flecainide The excretion of Flecainide can be decreased when combined with Ethoxzolamide.
Memantine The excretion of Memantine can be decreased when combined with Ethoxzolamide.
Quinine The excretion of Quinine can be decreased when combined with Ethoxzolamide.
Quinidine The excretion of Quinidine can be decreased when combined with Ethoxzolamide.
Methotrexate The protein binding of Methotrexate can be increased when combined with Ethoxzolamide.
Lithium hydroxide The excretion of Lithium hydroxide can be increased when combined with Ethoxzolamide.
Lithium citrate The excretion of Lithium citrate can be increased when combined with Ethoxzolamide.
Metformin The risk or severity of lactic acidosis can be increased when Ethoxzolamide is combined with Metformin.
Dexketoprofen The risk or severity of adverse effects can be increased when Dexketoprofen is combined with Ethoxzolamide.
Ketoprofen The risk or severity of adverse effects can be increased when Ketoprofen is combined with Ethoxzolamide.
Methenamine The serum concentration of the active metabolites of Methenamine can be reduced when Methenamine is used in combination with Ethoxzolamide resulting in a loss in efficacy.
Cyclosporine The risk or severity of renal failure can be increased when Ethoxzolamide is combined with Cyclosporine.
Triethylenetetramine The excretion of Triethylenetetramine can be increased when combined with Ethoxzolamide.
Aminosalicylic acid The risk or severity of adverse effects can be increased when Aminosalicylic acid is combined with Ethoxzolamide.
Mesalazine The risk or severity of adverse effects can be increased when Mesalazine is combined with Ethoxzolamide.
Sulfasalazine The risk or severity of adverse effects can be increased when Sulfasalazine is combined with Ethoxzolamide.
Diflunisal The risk or severity of adverse effects can be increased when Diflunisal is combined with Ethoxzolamide.
Salicylic acid The risk or severity of adverse effects can be increased when Salicylic acid is combined with Ethoxzolamide.
Balsalazide The risk or severity of adverse effects can be increased when Balsalazide is combined with Ethoxzolamide.
Olsalazine The risk or severity of adverse effects can be increased when Olsalazine is combined with Ethoxzolamide.
Bismuth subsalicylate The risk or severity of adverse effects can be increased when Bismuth subsalicylate is combined with Ethoxzolamide.
Dersalazine The risk or severity of adverse effects can be increased when Dersalazine is combined with Ethoxzolamide.
Phenyl aminosalicylate The risk or severity of adverse effects can be increased when Phenyl aminosalicylate is combined with Ethoxzolamide.
Methyl salicylate The risk or severity of adverse effects can be increased when Methyl salicylate is combined with Ethoxzolamide.
Nitroaspirin The risk or severity of adverse effects can be increased when Nitroaspirin is combined with Ethoxzolamide.
Aloxiprin The risk or severity of adverse effects can be increased when Aloxiprin is combined with Ethoxzolamide.
Guacetisal The risk or severity of adverse effects can be increased when Guacetisal is combined with Ethoxzolamide.
Carbaspirin calcium The risk or severity of adverse effects can be increased when Carbaspirin calcium is combined with Ethoxzolamide.
Choline salicylate The risk or severity of adverse effects can be increased when Choline salicylate is combined with Ethoxzolamide.
Thiosalicylic acid The risk or severity of adverse effects can be increased when Thiosalicylic acid is combined with Ethoxzolamide.
Phenytoin The risk or severity of osteomalacia can be increased when Ethoxzolamide is combined with Phenytoin.
Fosphenytoin The risk or severity of osteomalacia can be increased when Ethoxzolamide is combined with Fosphenytoin.
Methazolamide The risk or severity of adverse effects can be increased when Ethoxzolamide is combined with Methazolamide.
Acetazolamide The risk or severity of adverse effects can be increased when Ethoxzolamide is combined with Acetazolamide.
Zonisamide The risk or severity of adverse effects can be increased when Ethoxzolamide is combined with Zonisamide.
Diclofenamide The risk or severity of adverse effects can be increased when Ethoxzolamide is combined with Diclofenamide.
Amphetamine Ethoxzolamide may decrease the excretion rate of Amphetamine which could result in a higher serum level.
Phentermine Ethoxzolamide may decrease the excretion rate of Phentermine which could result in a higher serum level.
Pseudoephedrine Ethoxzolamide may decrease the excretion rate of Pseudoephedrine which could result in a higher serum level.
Benzphetamine Ethoxzolamide may decrease the excretion rate of Benzphetamine which could result in a higher serum level.
Diethylpropion Ethoxzolamide may decrease the excretion rate of Diethylpropion which could result in a higher serum level.
Lisdexamfetamine Ethoxzolamide may decrease the excretion rate of Lisdexamfetamine which could result in a higher serum level.
Mephentermine Ethoxzolamide may decrease the excretion rate of Mephentermine which could result in a higher serum level.
MMDA Ethoxzolamide may decrease the excretion rate of MMDA which could result in a higher serum level.
Midomafetamine Ethoxzolamide may decrease the excretion rate of Midomafetamine which could result in a higher serum level.
2,5-Dimethoxy-4-ethylamphetamine Ethoxzolamide may decrease the excretion rate of 2,5-Dimethoxy-4-ethylamphetamine which could result in a higher serum level.
4-Bromo-2,5-dimethoxyamphetamine Ethoxzolamide may decrease the excretion rate of 4-Bromo-2,5-dimethoxyamphetamine which could result in a higher serum level.
Tenamfetamine Ethoxzolamide may decrease the excretion rate of Tenamfetamine which could result in a higher serum level.
Chlorphentermine Ethoxzolamide may decrease the excretion rate of Chlorphentermine which could result in a higher serum level.
Methylenedioxyethamphetamine Ethoxzolamide may decrease the excretion rate of Methylenedioxyethamphetamine which could result in a higher serum level.
Dextroamphetamine Ethoxzolamide may decrease the excretion rate of Dextroamphetamine which could result in a higher serum level.
Metamfetamine Ethoxzolamide may decrease the excretion rate of Metamfetamine which could result in a higher serum level.
Iofetamine I-123 Ethoxzolamide may decrease the excretion rate of Iofetamine I-123 which could result in a higher serum level.
Ritobegron Ethoxzolamide may decrease the excretion rate of Ritobegron which could result in a higher serum level.
Mephedrone Ethoxzolamide may decrease the excretion rate of Mephedrone which could result in a higher serum level.
Methoxyphenamine Ethoxzolamide may decrease the excretion rate of Methoxyphenamine which could result in a higher serum level.
Gepefrine Ethoxzolamide may decrease the excretion rate of Gepefrine which could result in a higher serum level.
2,5-Dimethoxy-4-ethylthioamphetamine Ethoxzolamide may decrease the excretion rate of 2,5-Dimethoxy-4-ethylthioamphetamine which could result in a higher serum level.
Phendimetrazine Ethoxzolamide may decrease the excretion rate of Phendimetrazine which could result in a higher serum level.
Sodium phosphate, monobasic Ethoxzolamide may increase the nephrotoxic activities of Sodium phosphate, monobasic.
Acemetacin The therapeutic efficacy of Ethoxzolamide can be decreased when used in combination with Acemetacin.
Lactulose The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Lactulose.
Magnesium sulfate The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Magnesium sulfate.
Mannitol The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Mannitol.
Lubiprostone The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Lubiprostone.
Tegaserod The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Tegaserod.
Magnesium oxide The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Magnesium oxide.
Magnesium cation The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Magnesium cation.
Sorbitol The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Sorbitol.
Dantron The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Dantron.
Oxyphenisatin The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Oxyphenisatin.
Phenolphthalein The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Phenolphthalein.
Prucalopride The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Prucalopride.
Emodin The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Emodin.
Linaclotide The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Linaclotide.
Bisacodyl The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Bisacodyl.
Magnesium hydroxide The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Magnesium hydroxide.
Bisoxatin The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Bisoxatin.
Picosulfuric acid The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Picosulfuric acid.
Magnesium trisilicate The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Magnesium trisilicate.
Polyethylene glycol The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Polyethylene glycol.
Polycarbophil The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Polycarbophil.
Magnesium acetate tetrahydrate The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Magnesium acetate tetrahydrate.
Monopotassium phosphate The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Monopotassium phosphate.
Dipotassium phosphate The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Dipotassium phosphate.
Glycerin The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Glycerin.
Sodium sulfate The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Sodium sulfate.
Magnesium carbonate The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Magnesium carbonate.
Potassium lactate The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Potassium lactate.
Sodium fluorophosphate The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Sodium fluorophosphate.
Mineral oil The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Mineral oil.
Carboxymethylcellulose The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Carboxymethylcellulose.
Docusate The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Docusate.
Plantago seed The risk or severity of dehydration can be increased when Ethoxzolamide is combined with Plantago seed.

Target Protein

Carbonic anhydrase 2 CA2
Carbonic anhydrase 4 CA4
Carbonic anhydrase 7 CA7
Carbonic anhydrase 1 CA1
Carbonic anhydrase 3 CA3

Referensi & Sumber

Synthesis reference: Korman, J.; U.S. Patent 2,868,800; January 13, 1959; assigned to The Upjohn Company.

Contoh Produk & Brand

Produk: 0 • International brands: 2
International Brands
  • Cardrase — PHARMACIA AND UPJOHN
  • Ethamide — ALLERGAN

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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