Peringatan Keamanan

Acute overdose in animals results in CNS toxicity; notably, CNS depression, rapid gasping breathing, and convulsions. The intravenous median lethal dose in the rat was more than 50 mg/kg which is, on a mg/m2 basis, at least 250 times the maximum recommended human dose.

Ibutilide

DB00308

small molecule approved

Deskripsi

Ibutilide is a Class III antiarrhythmic agent available in intravenous formulations. It is indicated for the conversion of acute atrial flutter and recent onset atrial fibrillation to normal sinus rhythm (NSR).

Struktur Molekul 2D

Berat 384.576
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 6 hours (ranges from 2-12 hours)
Volume Distribusi * 11 L/kg
Klirens (Clearance) * 29 mL/min/kg

Absorpsi

Rapid after intravenous injection

Metabolisme

Primarily hepatic. Eight metabolites of ibutilide were detected in metabolic profiling of urine. These metabolites are thought to be formed primarily by o-oxidation followed by sequential b-oxidation of the heptyl side chain of ibutilide. Of the eight metabolites, only the o-hydroxy metabolite possesses class III electrophysiologic properties similar to that of ibutilide in an in vitro isolated rabbit myocardium model.

Rute Eliminasi

In healthy male volunteers, about 82% of a 0.01 mg/kg dose of 14C ibutilide fumarate was excreted in the urine (about 7% of the dose as unchanged ibutilide) and the remainder (about 19%) was recovered in the feces.

Interaksi Obat

1090 Data
Fingolimod Fingolimod may increase the arrhythmogenic activities of Ibutilide.
Lidocaine Lidocaine may increase the arrhythmogenic activities of Ibutilide.
Atenolol Ibutilide may increase the arrhythmogenic activities of Atenolol.
Mexiletine Ibutilide may increase the arrhythmogenic activities of Mexiletine.
Acetyldigitoxin Ibutilide may increase the arrhythmogenic activities of Acetyldigitoxin.
Carteolol Ibutilide may increase the arrhythmogenic activities of Carteolol.
Lercanidipine Ibutilide may increase the arrhythmogenic activities of Lercanidipine.
Magnesium sulfate Ibutilide may increase the arrhythmogenic activities of Magnesium sulfate.
Alprenolol Ibutilide may increase the arrhythmogenic activities of Alprenolol.
Tocainide Ibutilide may increase the arrhythmogenic activities of Tocainide.
Deslanoside Ibutilide may increase the arrhythmogenic activities of Deslanoside.
Carvedilol Ibutilide may increase the arrhythmogenic activities of Carvedilol.
Metipranolol Ibutilide may increase the arrhythmogenic activities of Metipranolol.
Practolol Ibutilide may increase the arrhythmogenic activities of Practolol.
Aprindine Ibutilide may increase the arrhythmogenic activities of Aprindine.
Dexpropranolol Ibutilide may increase the arrhythmogenic activities of Dexpropranolol.
Cyclandelate Ibutilide may increase the arrhythmogenic activities of Cyclandelate.
Flunarizine Ibutilide may increase the arrhythmogenic activities of Flunarizine.
Nebivolol Ibutilide may increase the arrhythmogenic activities of Nebivolol.
Seletracetam Ibutilide may increase the arrhythmogenic activities of Seletracetam.
Nylidrin Ibutilide may increase the arrhythmogenic activities of Nylidrin.
Dotarizine Ibutilide may increase the arrhythmogenic activities of Dotarizine.
Xylometazoline Ibutilide may increase the arrhythmogenic activities of Xylometazoline.
Sparteine Ibutilide may increase the arrhythmogenic activities of Sparteine.
Tranilast Ibutilide may increase the arrhythmogenic activities of Tranilast.
Fasudil Ibutilide may increase the arrhythmogenic activities of Fasudil.
Agmatine Ibutilide may increase the arrhythmogenic activities of Agmatine.
Barnidipine Ibutilide may increase the arrhythmogenic activities of Barnidipine.
Azelnidipine Ibutilide may increase the arrhythmogenic activities of Azelnidipine.
Cilnidipine Ibutilide may increase the arrhythmogenic activities of Cilnidipine.
Darodipine Ibutilide may increase the arrhythmogenic activities of Darodipine.
Manidipine Ibutilide may increase the arrhythmogenic activities of Manidipine.
Niludipine Ibutilide may increase the arrhythmogenic activities of Niludipine.
Carboxyamidotriazole Ibutilide may increase the arrhythmogenic activities of Carboxyamidotriazole.
Naftopidil Ibutilide may increase the arrhythmogenic activities of Naftopidil.
Vinpocetine Ibutilide may increase the arrhythmogenic activities of Vinpocetine.
Landiolol Ibutilide may increase the arrhythmogenic activities of Landiolol.
Cymarin Ibutilide may increase the arrhythmogenic activities of Cymarin.
Metildigoxin Ibutilide may increase the arrhythmogenic activities of Metildigoxin.
Tiracizine Ibutilide may increase the arrhythmogenic activities of Tiracizine.
Ethacizine Ibutilide may increase the arrhythmogenic activities of Ethacizine.
Hydroquinine Ibutilide may increase the arrhythmogenic activities of Hydroquinine.
Bioallethrin Ibutilide may increase the arrhythmogenic activities of Bioallethrin.
Tertatolol Ibutilide may increase the arrhythmogenic activities of Tertatolol.
Caroverine Ibutilide may increase the arrhythmogenic activities of Caroverine.
Fosfructose Ibutilide may increase the arrhythmogenic activities of Fosfructose.
WIN 55212-2 Ibutilide may increase the arrhythmogenic activities of WIN 55212-2.
Fish oil Ibutilide may increase the arrhythmogenic activities of Fish oil.
Emopamil Ibutilide may increase the arrhythmogenic activities of Emopamil.
Lomerizine Ibutilide may increase the arrhythmogenic activities of Lomerizine.
Tetrandrine Ibutilide may increase the arrhythmogenic activities of Tetrandrine.
Dexniguldipine Ibutilide may increase the arrhythmogenic activities of Dexniguldipine.
Fosinoprilat Ibutilide may increase the arrhythmogenic activities of Fosinoprilat.
Hydroquinidine Ibutilide may increase the arrhythmogenic activities of Hydroquinidine.
SOR-C13 Ibutilide may increase the arrhythmogenic activities of SOR-C13.
Betaxolol Betaxolol may increase the arrhythmogenic activities of Ibutilide.
Diltiazem Ibutilide may increase the arrhythmogenic activities of Diltiazem.
Nimodipine Ibutilide may increase the arrhythmogenic activities of Nimodipine.
Cinnarizine Ibutilide may increase the arrhythmogenic activities of Cinnarizine.
Propranolol Ibutilide may increase the arrhythmogenic activities of Propranolol.
Atropine Ibutilide may increase the arrhythmogenic activities of Atropine.
Adenosine Ibutilide may increase the arrhythmogenic activities of Adenosine.
Loperamide Ibutilide may increase the arrhythmogenic activities of Loperamide.
Levosimendan Ibutilide may increase the arrhythmogenic activities of Levosimendan.
Nifedipine Ibutilide may increase the arrhythmogenic activities of Nifedipine.
Propafenone Ibutilide may increase the arrhythmogenic activities of Propafenone.
Acebutolol Ibutilide may increase the arrhythmogenic activities of Acebutolol.
Flecainide Ibutilide may increase the arrhythmogenic activities of Flecainide.
Mibefradil Ibutilide may increase the arrhythmogenic activities of Mibefradil.
Oxprenolol Ibutilide may increase the arrhythmogenic activities of Oxprenolol.
Prenylamine Ibutilide may increase the arrhythmogenic activities of Prenylamine.
Fluspirilene Ibutilide may increase the arrhythmogenic activities of Fluspirilene.
Azimilide Ibutilide may increase the arrhythmogenic activities of Azimilide.
Tedisamil Ibutilide may increase the arrhythmogenic activities of Tedisamil.
Nilvadipine Ibutilide may increase the arrhythmogenic activities of Nilvadipine.
Fendiline Ibutilide may increase the arrhythmogenic activities of Fendiline.
Eperisone Ibutilide may increase the arrhythmogenic activities of Eperisone.
Melperone Ibutilide may increase the arrhythmogenic activities of Melperone.
Benidipine Ibutilide may increase the arrhythmogenic activities of Benidipine.
Simendan Ibutilide may increase the arrhythmogenic activities of Simendan.
Otilonium Ibutilide may increase the arrhythmogenic activities of Otilonium.
Nizofenone Ibutilide may increase the arrhythmogenic activities of Nizofenone.
Bunaftine Ibutilide may increase the arrhythmogenic activities of Bunaftine.
Lorcainide Ibutilide may increase the arrhythmogenic activities of Lorcainide.
Penfluridol Ibutilide may increase the arrhythmogenic activities of Penfluridol.
Dexverapamil Ibutilide may increase the arrhythmogenic activities of Dexverapamil.
Esmolol Esmolol may increase the arrhythmogenic activities of Ibutilide.
Isradipine Isradipine may increase the arrhythmogenic activities of Ibutilide.
Trimethadione Ibutilide may increase the arrhythmogenic activities of Trimethadione.
Timolol Ibutilide may increase the arrhythmogenic activities of Timolol.
Amlodipine Ibutilide may increase the arrhythmogenic activities of Amlodipine.
Digoxin Ibutilide may increase the arrhythmogenic activities of Digoxin.
Hyoscyamine Ibutilide may increase the arrhythmogenic activities of Hyoscyamine.
Lamotrigine Ibutilide may increase the arrhythmogenic activities of Lamotrigine.
Ethosuximide Ibutilide may increase the arrhythmogenic activities of Ethosuximide.
Nicardipine Ibutilide may increase the arrhythmogenic activities of Nicardipine.
Verapamil Ibutilide may increase the arrhythmogenic activities of Verapamil.
Losartan Ibutilide may increase the arrhythmogenic activities of Losartan.
Moricizine Ibutilide may increase the arrhythmogenic activities of Moricizine.
Levomenthol Ibutilide may increase the arrhythmogenic activities of Levomenthol.

Target Protein

Voltage-dependent L-type calcium channel subunit alpha-1C CACNA1C
Voltage-dependent L-type calcium channel subunit beta-1 CACNB1
Voltage-gated inwardly rectifying potassium channel KCNH2 KCNH2
Voltage-dependent calcium channel subunit alpha-2/delta-1 CACNA2D1
Voltage-dependent calcium channel gamma-1 subunit CACNG1
Potassium channel subfamily K member 1 KCNK1
Potassium channel subfamily K member 6 KCNK6
Voltage-gated inwardly rectifying potassium channel KCNH6 KCNH6
Voltage-gated inwardly rectifying potassium channel KCNH7 KCNH7
ATP-sensitive inward rectifier potassium channel 11 KCNJ11

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 6 • International brands: 0
Produk
  • Corvert
    Injection, solution • 0.1 mg/1mL • Intravenous • US • Approved
  • Corvert
    Solution • 0.1 mg / mL • Intravenous • Canada • Approved
  • Ibutilide Fumarate
    Injection, solution • 0.1 mg/1mL • Intravenous • US • Generic • Approved
  • Ibutilide Fumarate
    Injection, solution • 0.1 mg/1mL • Intravenous • US • Generic • Approved
  • Ibutilide Fumarate
    Injection, solution • 0.1 mg/1mL • Intravenous • US • Generic • Approved
  • Ibutilide Fumarate
    Injection, solution • 1 mg/10mL • Intravenous • US • Generic • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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