Peringatan Keamanan

Oral, mouse: LD50 = 23 mg/kg; Oral, rat: LD50 = 30 mg/kg. Symptoms of overdose include nausea and vomiting.

Mitomycin

DB00305

small molecule approved

Deskripsi

Mitomycin is an antineoplastic antibiotic first isolated by Japanese microbiologists in the 1950s from cultures of Streptomyces caespitosus.L12867,A193419 It is an alkylating agent that inhibits DNA synthesis (and, at higher concentrations, RNA and protein synthesis) by cross-linking the complementary strands of the DNA double helix.A193419 Few other antibiotics have been discovered that work via this alkylating mechanism, making mitomycin relatively unique in the space of microbiota-derived therapies.A193419

Mitomycin's cross-linking activity has resulted in its approval for the treatment of a variety of cancers - the most recent of which is an April 2020 approval for its use in low-grade Upper Tract Urothelial Cancer (LG-UTUC)L12867 - as well as adjunctly to ab externo glaucoma surgeries.

Struktur Molekul 2D

Berat 334.3272
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 8-48 min
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Erratic.

Metabolisme

Primarily hepatic, some in various other tissues.

Rute Eliminasi

Approximately 10% of a dose of mitomycin is excreted unchanged in the urine.

Interaksi Obat

549 Data
Denosumab The risk or severity of adverse effects can be increased when Denosumab is combined with Mitomycin.
Etanercept The risk or severity of adverse effects can be increased when Etanercept is combined with Mitomycin.
Peginterferon alfa-2a The risk or severity of adverse effects can be increased when Peginterferon alfa-2a is combined with Mitomycin.
Interferon alfa-n1 The risk or severity of adverse effects can be increased when Interferon alfa-n1 is combined with Mitomycin.
Interferon alfa-n3 The risk or severity of adverse effects can be increased when Interferon alfa-n3 is combined with Mitomycin.
Peginterferon alfa-2b The risk or severity of adverse effects can be increased when Peginterferon alfa-2b is combined with Mitomycin.
Anakinra The risk or severity of adverse effects can be increased when Anakinra is combined with Mitomycin.
Interferon gamma-1b The risk or severity of adverse effects can be increased when Interferon gamma-1b is combined with Mitomycin.
Interferon alfa-2a The risk or severity of adverse effects can be increased when Interferon alfa-2a is combined with Mitomycin.
Aldesleukin The risk or severity of adverse effects can be increased when Aldesleukin is combined with Mitomycin.
Adalimumab The risk or severity of adverse effects can be increased when Adalimumab is combined with Mitomycin.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Mitomycin.
Pegaspargase The risk or severity of adverse effects can be increased when Pegaspargase is combined with Mitomycin.
Infliximab The risk or severity of adverse effects can be increased when Infliximab is combined with Mitomycin.
Interferon beta-1b The risk or severity of adverse effects can be increased when Interferon beta-1b is combined with Mitomycin.
Interferon alfacon-1 The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Mitomycin.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Mitomycin.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Mitomycin.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Mitomycin.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Mitomycin.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Mitomycin.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Mitomycin.
Alefacept The risk or severity of adverse effects can be increased when Alefacept is combined with Mitomycin.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Mitomycin.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Mitomycin.
Interferon alfa-2b The risk or severity of adverse effects can be increased when Interferon alfa-2b is combined with Mitomycin.
Daclizumab The risk or severity of adverse effects can be increased when Daclizumab is combined with Mitomycin.
Phenylalanine The risk or severity of adverse effects can be increased when Phenylalanine is combined with Mitomycin.
Flunisolide The risk or severity of adverse effects can be increased when Flunisolide is combined with Mitomycin.
Bortezomib The risk or severity of adverse effects can be increased when Bortezomib is combined with Mitomycin.
Cladribine Mitomycin may increase the immunosuppressive activities of Cladribine.
Carmustine The risk or severity of adverse effects can be increased when Carmustine is combined with Mitomycin.
Amsacrine The risk or severity of adverse effects can be increased when Amsacrine is combined with Mitomycin.
Bleomycin The risk or severity of adverse effects can be increased when Bleomycin is combined with Mitomycin.
Chlorambucil The risk or severity of adverse effects can be increased when Chlorambucil is combined with Mitomycin.
Raltitrexed The risk or severity of adverse effects can be increased when Raltitrexed is combined with Mitomycin.
Bexarotene The risk or severity of adverse effects can be increased when Mitomycin is combined with Bexarotene.
Floxuridine The risk or severity of adverse effects can be increased when Mitomycin is combined with Floxuridine.
Indomethacin The risk or severity of adverse effects can be increased when Mitomycin is combined with Indomethacin.
Tioguanine The risk or severity of adverse effects can be increased when Mitomycin is combined with Tioguanine.
Dexrazoxane The risk or severity of adverse effects can be increased when Mitomycin is combined with Dexrazoxane.
Beclomethasone dipropionate The risk or severity of adverse effects can be increased when Mitomycin is combined with Beclomethasone dipropionate.
Sorafenib The risk or severity of adverse effects can be increased when Mitomycin is combined with Sorafenib.
Streptozocin The risk or severity of adverse effects can be increased when Mitomycin is combined with Streptozocin.
Trifluridine The risk or severity of adverse effects can be increased when Mitomycin is combined with Trifluridine.
Gemcitabine The risk or severity of adverse effects can be increased when Mitomycin is combined with Gemcitabine.
Betamethasone The risk or severity of adverse effects can be increased when Mitomycin is combined with Betamethasone.
Teniposide The risk or severity of adverse effects can be increased when Mitomycin is combined with Teniposide.
Epirubicin The risk or severity of adverse effects can be increased when Mitomycin is combined with Epirubicin.
Chloramphenicol The risk or severity of adverse effects can be increased when Mitomycin is combined with Chloramphenicol.
Lenalidomide The risk or severity of adverse effects can be increased when Mitomycin is combined with Lenalidomide.
Altretamine The risk or severity of adverse effects can be increased when Mitomycin is combined with Altretamine.
Zidovudine The risk or severity of adverse effects can be increased when Mitomycin is combined with Zidovudine.
Cisplatin The risk or severity of adverse effects can be increased when Mitomycin is combined with Cisplatin.
Oxaliplatin The risk or severity of adverse effects can be increased when Mitomycin is combined with Oxaliplatin.
Cyclophosphamide The risk or severity of adverse effects can be increased when Mitomycin is combined with Cyclophosphamide.
Fluorouracil The risk or severity of adverse effects can be increased when Mitomycin is combined with Fluorouracil.
Propylthiouracil The risk or severity of adverse effects can be increased when Mitomycin is combined with Propylthiouracil.
Pentostatin The risk or severity of adverse effects can be increased when Mitomycin is combined with Pentostatin.
Methotrexate The risk or severity of adverse effects can be increased when Mitomycin is combined with Methotrexate.
Carbamazepine The risk or severity of adverse effects can be increased when Mitomycin is combined with Carbamazepine.
Fluticasone propionate The risk or severity of adverse effects can be increased when Mitomycin is combined with Fluticasone propionate.
Fluocinolone acetonide The risk or severity of adverse effects can be increased when Mitomycin is combined with Fluocinolone acetonide.
Linezolid The risk or severity of adverse effects can be increased when Mitomycin is combined with Linezolid.
Imatinib The risk or severity of adverse effects can be increased when Mitomycin is combined with Imatinib.
Triamcinolone The risk or severity of adverse effects can be increased when Mitomycin is combined with Triamcinolone.
Clofarabine The risk or severity of adverse effects can be increased when Mitomycin is combined with Clofarabine.
Prednisone The risk or severity of adverse effects can be increased when Mitomycin is combined with Prednisone.
Pemetrexed The risk or severity of adverse effects can be increased when Mitomycin is combined with Pemetrexed.
Fludrocortisone The risk or severity of adverse effects can be increased when Mitomycin is combined with Fludrocortisone.
Mycophenolate mofetil The risk or severity of adverse effects can be increased when Mitomycin is combined with Mycophenolate mofetil.
Daunorubicin The risk or severity of adverse effects can be increased when Mitomycin is combined with Daunorubicin.
Tretinoin The risk or severity of cardiotoxicity can be increased when Mitomycin is combined with Tretinoin.
Irinotecan The risk or severity of adverse effects can be increased when Mitomycin is combined with Irinotecan.
Methimazole The risk or severity of adverse effects can be increased when Mitomycin is combined with Methimazole.
Etoposide The risk or severity of adverse effects can be increased when Mitomycin is combined with Etoposide.
Sulfasalazine The risk or severity of adverse effects can be increased when Mitomycin is combined with Sulfasalazine.
Dacarbazine The risk or severity of adverse effects can be increased when Mitomycin is combined with Dacarbazine.
Temozolomide The risk or severity of adverse effects can be increased when Mitomycin is combined with Temozolomide.
Penicillamine The risk or severity of adverse effects can be increased when Mitomycin is combined with Penicillamine.
Prednisolone The risk or severity of adverse effects can be increased when Mitomycin is combined with Prednisolone.
Sirolimus The risk or severity of adverse effects can be increased when Mitomycin is combined with Sirolimus.
Mechlorethamine The risk or severity of adverse effects can be increased when Mitomycin is combined with Mechlorethamine.
Azacitidine The risk or severity of adverse effects can be increased when Mitomycin is combined with Azacitidine.
Carboplatin The risk or severity of adverse effects can be increased when Mitomycin is combined with Carboplatin.
Methylprednisolone The risk or severity of adverse effects can be increased when Mitomycin is combined with Methylprednisolone.
Dactinomycin The risk or severity of adverse effects can be increased when Mitomycin is combined with Dactinomycin.
Cytarabine The risk or severity of adverse effects can be increased when Mitomycin is combined with Cytarabine.
Azathioprine The risk or severity of adverse effects can be increased when Mitomycin is combined with Azathioprine.
Doxorubicin The risk or severity of adverse effects can be increased when Mitomycin is combined with Doxorubicin.
Hydroxyurea The risk or severity of adverse effects can be increased when Mitomycin is combined with Hydroxyurea.
Busulfan The risk or severity of adverse effects can be increased when Mitomycin is combined with Busulfan.
Mycophenolic acid The risk or severity of adverse effects can be increased when Mitomycin is combined with Mycophenolic acid.
Topotecan The risk or severity of adverse effects can be increased when Mitomycin is combined with Topotecan.
Mercaptopurine The risk or severity of adverse effects can be increased when Mitomycin is combined with Mercaptopurine.
Thalidomide The risk or severity of adverse effects can be increased when Mitomycin is combined with Thalidomide.
Melphalan The risk or severity of adverse effects can be increased when Mitomycin is combined with Melphalan.
Fludarabine The risk or severity of adverse effects can be increased when Mitomycin is combined with Fludarabine.
Flucytosine The risk or severity of adverse effects can be increased when Mitomycin is combined with Flucytosine.
Capecitabine The risk or severity of adverse effects can be increased when Mitomycin is combined with Capecitabine.

Target Protein

DNA

Referensi & Sumber

Synthesis reference: Leslie Jimenez, Zheng Wang, "Synthesis of mitomycin and its analogs." U.S. Patent US5523411, issued June, 1972.
Artikel (PubMed)
  • PMID: 9383461
    Tomasz M: Mitomycin C: small, fast and deadly (but very selective). Chem Biol. 1995 Sep;2(9):575-9. doi: 10.1016/1074-5521(95)90120-5.

Contoh Produk & Brand

Produk: 63 • International brands: 1
Produk
  • Jelmyto
    Kit; Powder, for solution • 40 mg/1 • Ureteral • US • Approved
  • Jelmyto
    Kit; Powder, for solution • 40 mg/1 • Ureteral • US • Approved
  • Mitomycin
    Injection, powder, lyophilized, for solution • 0.5 mg/1mL • Intravenous • US • Generic • Approved
  • Mitomycin
    Injection, powder, lyophilized, for solution • 0.5 mg/1mL • Intravenous • US • Generic • Approved
  • Mitomycin
    Injection, powder, lyophilized, for solution • 0.5 mg/1mL • Intravenous • US • Generic • Approved
  • Mitomycin
    Injection, powder, lyophilized, for solution • 5 mg/10mL • Intravenous • US • Generic • Approved
  • Mitomycin
    Injection, powder, lyophilized, for solution • 20 mg/40mL • Intravenous • US • Generic • Approved
  • Mitomycin
    Injection, powder, lyophilized, for solution • 40 mg/80mL • Intravenous • US • Generic • Approved
Menampilkan 8 dari 63 produk.
International Brands
  • Mitozytrex

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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