Peringatan Keamanan

Oral LD50 in rats is 3,204 mg/kg. With other b-lactam antibiotics, adverse effects following overdosage have included nausea, vomiting, epigastric distress, diarrhea, and convulsions.

Cefmetazole

DB00274

small molecule approved investigational

Deskripsi

A semisynthetic cephamycin antibiotic with a broad spectrum of activity against both gram-positive and gram-negative microorganisms. It has a high rate of efficacy in many types of infection and to date no severe side effects have been noted.

Struktur Molekul 2D

Berat 471.534
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 1.50 ±0.14 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Bioavailability is approximately 100% following intramuscular injection.

Metabolisme

No appreciable metabolism.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

795 Data
Probenecid The serum concentration of Cefmetazole can be increased when it is combined with Probenecid.
Foscarnet The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Foscarnet.
Mannitol The risk or severity of nephrotoxicity can be increased when Mannitol is combined with Cefmetazole.
Tenofovir disoproxil Cefmetazole may increase the nephrotoxic activities of Tenofovir disoproxil.
Tenofovir alafenamide Cefmetazole may increase the nephrotoxic activities of Tenofovir alafenamide.
Tenofovir Cefmetazole may increase the nephrotoxic activities of Tenofovir.
Cyclosporine The risk or severity of nephrotoxicity can be increased when Cyclosporine is combined with Cefmetazole.
Icosapent The risk or severity of nephrotoxicity can be increased when Icosapent is combined with Cefmetazole.
Cefotiam The risk or severity of nephrotoxicity can be increased when Cefotiam is combined with Cefmetazole.
Mesalazine The risk or severity of nephrotoxicity can be increased when Mesalazine is combined with Cefmetazole.
Cefmenoxime The risk or severity of nephrotoxicity can be increased when Cefmenoxime is combined with Cefmetazole.
Indomethacin The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Indomethacin.
Triamterene The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Triamterene.
Cefpiramide The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefpiramide.
Loracarbef The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Loracarbef.
Cefalotin The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefalotin.
Nabumetone The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Nabumetone.
Ketorolac The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Ketorolac.
Tenoxicam The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Tenoxicam.
Celecoxib The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Celecoxib.
Cefotaxime The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefotaxime.
Tolmetin The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Tolmetin.
Rofecoxib The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Rofecoxib.
Fenoprofen The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Fenoprofen.
Valdecoxib The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Valdecoxib.
Diclofenac The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Diclofenac.
Sulindac The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Sulindac.
Bacitracin The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Bacitracin.
Amphotericin B The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Amphotericin B.
Cephaloglycin The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cephaloglycin.
Adefovir dipivoxil The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Adefovir dipivoxil.
Pentamidine The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Pentamidine.
Mefenamic acid The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Mefenamic acid.
Naproxen The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Naproxen.
Sulfasalazine The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Sulfasalazine.
Phenylbutazone The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Phenylbutazone.
Meloxicam The risk or severity of methemoglobinemia can be increased when Cefmetazole is combined with Meloxicam.
Carprofen The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Carprofen.
Tacrolimus The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Tacrolimus.
Etacrynic acid The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Etacrynic acid.
Ceforanide The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Ceforanide.
Salicylic acid The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Salicylic acid.
Acetylsalicylic acid The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Acetylsalicylic acid.
Hydrochlorothiazide The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Hydrochlorothiazide.
Balsalazide The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Balsalazide.
Cefditoren The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefditoren.
Atazanavir The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Atazanavir.
Colistimethate The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Colistimethate.
Cefuroxime The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefuroxime.
Cefapirin The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefapirin.
Cefprozil The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefprozil.
Olsalazine The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Olsalazine.
Lumiracoxib The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Lumiracoxib.
Cefamandole The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefamandole.
Cefazolin The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefazolin.
Cefonicid The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefonicid.
Cefoperazone The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefoperazone.
Cefoxitin The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefoxitin.
Ceftizoxime The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Ceftizoxime.
Magnesium salicylate The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Magnesium salicylate.
Salsalate The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Salsalate.
Choline magnesium trisalicylate The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Choline magnesium trisalicylate.
Cefepime The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefepime.
Cefacetrile The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefacetrile.
Cefpodoxime The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefpodoxime.
Antrafenine The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Antrafenine.
Aminophenazone The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Aminophenazone.
Antipyrine The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Antipyrine.
Tiaprofenic acid The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Tiaprofenic acid.
Lopinavir The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Lopinavir.
Etoricoxib The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Etoricoxib.
Hydrolyzed Cephalothin The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Hydrolyzed Cephalothin.
Cephalothin Group The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cephalothin Group.
Oxyphenbutazone The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Oxyphenbutazone.
Latamoxef The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Latamoxef.
Nimesulide The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Nimesulide.
Benoxaprofen The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Benoxaprofen.
Metamizole The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Metamizole.
Zomepirac The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Zomepirac.
Ceftobiprole The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Ceftobiprole.
Cimicoxib The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cimicoxib.
Ceftaroline fosamil The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Ceftaroline fosamil.
Lornoxicam The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Lornoxicam.
Zaltoprofen The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Zaltoprofen.
Azapropazone The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Azapropazone.
Parecoxib The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Parecoxib.
Salicylamide The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Salicylamide.
Kebuzone The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Kebuzone.
Isoxicam The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Isoxicam.
Indoprofen The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Indoprofen.
Ibuproxam The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Ibuproxam.
Floctafenine The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Floctafenine.
Fenbufen The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Fenbufen.
Etofenamate The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Etofenamate.
Epirizole The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Epirizole.
Cefaloridine The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefaloridine.
Cefminox The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefminox.
Dexibuprofen The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Dexibuprofen.
Droxicam The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Droxicam.
Tolfenamic acid The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Tolfenamic acid.

Target Protein

Penicillin binding protein 2a mecA
Penicillin-binding protein 1A mrcA
Penicillin-binding protein 1B mrcB
Peptidoglycan synthase FtsI ftsI
D-alanyl-D-alanine carboxypeptidase DacA dacA
D-alanyl-D-alanine carboxypeptidase DacC dacC

Referensi & Sumber

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Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Zefazone

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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