Peringatan Keamanan

Overdosage might be expected to produce nasal congestion, syncope, or hallucinations. Measures to support blood pressure should be taken if necessary.

Dapsone

DB00250

small molecule approved investigational

Deskripsi

A sulfone active against a wide range of bacteria but mainly employed for its actions against mycobacterium leprae. Its mechanism of action is probably similar to that of the sulfonamides which involves inhibition of folic acid synthesis in susceptible organisms. It is also used with pyrimethamine in the treatment of malaria. (From Martindale, The Extra Pharmacopoeia, 30th ed, p157-8)

Struktur Molekul 2D

Berat 248.301
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 28 hours (range 10-50 hours)
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Bioavailability is 70 to 80% following oral administration.

Metabolisme

Hepatic, mostly CYP2E1-mediated.

Rute Eliminasi

Renal

Interaksi Makanan

1 Data
  • 1. Take with or without food. The absorption is unaffected by food.

Interaksi Obat

710 Data
Artemether The risk or severity of QTc prolongation can be increased when Dapsone is combined with Artemether.
Lumefantrine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Lumefantrine.
Probenecid Probenecid may decrease the excretion rate of Dapsone which could result in a higher serum level.
Trimethoprim The serum concentration of Dapsone can be increased when it is combined with Trimethoprim.
Mifepristone The serum concentration of Dapsone can be increased when it is combined with Mifepristone.
Tetrahydrofolic acid The therapeutic efficacy of Dapsone can be decreased when used in combination with Tetrahydrofolic acid.
Folic acid The therapeutic efficacy of Dapsone can be decreased when used in combination with Folic acid.
Leucovorin The therapeutic efficacy of Dapsone can be decreased when used in combination with Leucovorin.
(6S)-5,6,7,8-tetrahydrofolic acid The therapeutic efficacy of Dapsone can be decreased when used in combination with (6S)-5,6,7,8-tetrahydrofolic acid.
Triglu-5-formyl-tetrahydrofolate The therapeutic efficacy of Dapsone can be decreased when used in combination with Triglu-5-formyl-tetrahydrofolate.
Levoleucovorin The therapeutic efficacy of Dapsone can be decreased when used in combination with Levoleucovorin.
5-methyltetrahydrofolic acid The therapeutic efficacy of Dapsone can be decreased when used in combination with 5-methyltetrahydrofolic acid.
Picosulfuric acid The therapeutic efficacy of Picosulfuric acid can be decreased when used in combination with Dapsone.
Thiethylperazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Thiethylperazine.
Promazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Promazine.
Prochlorperazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Prochlorperazine.
Chlorpromazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Chlorpromazine.
Triflupromazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Triflupromazine.
Fluphenazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Fluphenazine.
Thioridazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Thioridazine.
Moricizine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Moricizine.
Trifluoperazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Trifluoperazine.
Perphenazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Perphenazine.
Mesoridazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Mesoridazine.
Acetophenazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Acetophenazine.
Promethazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Promethazine.
Alimemazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Alimemazine.
Methotrimeprazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Methotrimeprazine.
Periciazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Periciazine.
Acepromazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Acepromazine.
Aceprometazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Aceprometazine.
Pipotiazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Pipotiazine.
Thioproperazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Thioproperazine.
BL-1020 The risk or severity of QTc prolongation can be increased when Dapsone is combined with BL-1020.
Cyamemazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Cyamemazine.
Methylene blue The risk or severity of QTc prolongation can be increased when Dapsone is combined with Methylene blue.
Propiopromazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Propiopromazine.
Perazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Perazine.
Butaperazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Butaperazine.
Chlorproethazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Chlorproethazine.
Thiazinam The risk or severity of QTc prolongation can be increased when Dapsone is combined with Thiazinam.
Dixyrazine The risk or severity of QTc prolongation can be increased when Dapsone is combined with Dixyrazine.
Perphenazine enanthate The risk or severity of QTc prolongation can be increased when Dapsone is combined with Perphenazine enanthate.
Pyrimethamine The risk or severity of adverse effects can be increased when Pyrimethamine is combined with Dapsone.
Amodiaquine The risk or severity of adverse effects can be increased when Amodiaquine is combined with Dapsone.
Quinidine The risk or severity of adverse effects can be increased when Quinidine is combined with Dapsone.
Quinacrine The risk or severity of adverse effects can be increased when Quinacrine is combined with Dapsone.
Atovaquone The risk or severity of adverse effects can be increased when Atovaquone is combined with Dapsone.
Proguanil The risk or severity of adverse effects can be increased when Proguanil is combined with Dapsone.
Halofantrine The risk or severity of adverse effects can be increased when Halofantrine is combined with Dapsone.
Sulfadoxine The risk or severity of adverse effects can be increased when Sulfadoxine is combined with Dapsone.
Hydroxychloroquine The risk or severity of adverse effects can be increased when Hydroxychloroquine is combined with Dapsone.
Tafenoquine The risk or severity of adverse effects can be increased when Tafenoquine is combined with Dapsone.
Artesunate The risk or severity of adverse effects can be increased when Artesunate is combined with Dapsone.
Artenimol The risk or severity of adverse effects can be increased when Artenimol is combined with Dapsone.
Artefenomel The risk or severity of adverse effects can be increased when Artefenomel is combined with Dapsone.
Chlorproguanil The risk or severity of adverse effects can be increased when Chlorproguanil is combined with Dapsone.
Mizoribine The risk or severity of adverse effects can be increased when Mizoribine is combined with Dapsone.
Pyronaridine The risk or severity of adverse effects can be increased when Pyronaridine is combined with Dapsone.
Artemisinin The risk or severity of adverse effects can be increased when Artemisinin is combined with Dapsone.
Artemotil The risk or severity of adverse effects can be increased when Artemotil is combined with Dapsone.
Piperaquine The risk or severity of adverse effects can be increased when Piperaquine is combined with Dapsone.
Tetrandrine The risk or severity of adverse effects can be increased when Tetrandrine is combined with Dapsone.
Cycloguanil The risk or severity of adverse effects can be increased when Cycloguanil is combined with Dapsone.
Butalbital The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Butalbital.
Phenytoin The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Phenytoin.
Lidocaine The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Lidocaine.
Acetaminophen The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Acetaminophen.
Nitroprusside The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Nitroprusside.
Sulfadiazine The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Sulfadiazine.
Nitric Oxide The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Nitric Oxide.
Quinine The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Quinine.
Celecoxib The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Celecoxib.
Flutamide The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Flutamide.
Chloroquine The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Chloroquine.
Nitrofurantoin The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Nitrofurantoin.
Nitroglycerin The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Nitroglycerin.
Prilocaine The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Prilocaine.
Isosorbide dinitrate The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Isosorbide dinitrate.
Sulfamethoxazole The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Sulfamethoxazole.
Isosorbide mononitrate The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Isosorbide mononitrate.
Benzocaine The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Benzocaine.
Primaquine The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Primaquine.
Phenobarbital The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Phenobarbital.
Zopiclone The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Zopiclone.
Metoclopramide The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Metoclopramide.
Antipyrine The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Antipyrine.
Phenazopyridine The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Phenazopyridine.
Amyl Nitrite The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Amyl Nitrite.
Isometheptene The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Isometheptene.
Mafenide The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Mafenide.
Nitrous oxide The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Nitrous oxide.
Cyclophosphamide The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Cyclophosphamide.
Ifosfamide The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Ifosfamide.
Sulfasalazine The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Sulfasalazine.
Sulfanilamide The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Sulfanilamide.
Sulfapyridine The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Sulfapyridine.
Valproic acid The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Valproic acid.
Rasburicase The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Rasburicase.
Aminosalicylic acid The risk or severity of methemoglobinemia can be increased when Dapsone is combined with Aminosalicylic acid.

Target Protein

Inactive dihydropteroate synthase 2 folP2
Dihydropteroate synthase folP1

Referensi & Sumber

Synthesis reference: Weijiard, J.and Messerly, J.P.; U.S. Patent 2,385,899; October 2,1945; assigned to Merck & Co., Inc.

Contoh Produk & Brand

Produk: 79 • International brands: 0
Produk
  • 011503 Dapsone 6% / Niacinamide 2% / Spironolactone 5%
    Gel • - • Topical • US
  • 011504 Dapsone 8.5% / Niacinamide 4%
    Gel • - • Topical • US
  • Aczone
    Gel • 50 mg/1g • Topical • US • Approved
  • Aczone
    Gel • 75 mg/1g • Topical • US • Approved
  • Aczone
    Gel • 50 mg/1g • Topical • US • Approved
  • Aczone
    Gel • 5 % w/w • Topical • Canada • Approved
  • Aczone
    Gel • 50 mg/1g • Topical • US • Approved
  • Aczone 7.5
    Gel • 75 mg/1g • Topical • US • Approved
Menampilkan 8 dari 79 produk.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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