Peringatan Keamanan

Few cases of acute methysergide intoxication have been reported. The possible symptom complex is therefore not fully known. The following symptoms are based on these few case reports. Euphoria, hyperactivity, tachycardia, dilated pupils, and dizziness have been reported in a child with a dose of 20-24 mg of methysergide. In adults, peripheral vasospasm, with diminished or absent pulses, coldness, mottling and cyanosis, has been observed at a dose of 200 mg. Ischemic tissue damage has not been reported in acute overdosage with methysergide.

Methysergide

DB00247

small molecule approved

Deskripsi

An ergot derivative that is a congener of lysergic acid diethylamide. It antagonizes the effects of serotonin in blood vessels and gastrointestinal smooth muscle, but has few of the properties of other ergot alkaloids. Methysergide is used prophylactically in migraine and other vascular headaches and to antagonize serotonin in the carcinoid syndrome.

Struktur Molekul 2D

Berat 353.458
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Rapid

Metabolisme

Hepatic

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

1 Data
  • 1. Take with food. Food reduces irritation.

Interaksi Obat

1468 Data
Phenytoin The metabolism of Methysergide can be increased when combined with Phenytoin.
Fosphenytoin The metabolism of Methysergide can be increased when combined with Fosphenytoin.
Valsartan Methysergide may decrease the antihypertensive activities of Valsartan.
Ramipril Methysergide may decrease the antihypertensive activities of Ramipril.
Remikiren Methysergide may decrease the antihypertensive activities of Remikiren.
Torasemide Methysergide may decrease the antihypertensive activities of Torasemide.
Guanadrel Methysergide may decrease the antihypertensive activities of Guanadrel.
Olmesartan Methysergide may decrease the antihypertensive activities of Olmesartan.
Chlorthalidone Methysergide may decrease the antihypertensive activities of Chlorthalidone.
Nitroprusside Methysergide may decrease the antihypertensive activities of Nitroprusside.
Minoxidil Methysergide may decrease the antihypertensive activities of Minoxidil.
Treprostinil Methysergide may decrease the antihypertensive activities of Treprostinil.
Bendroflumethiazide Methysergide may decrease the antihypertensive activities of Bendroflumethiazide.
Prazosin Methysergide may decrease the antihypertensive activities of Prazosin.
Fosinopril Methysergide may decrease the antihypertensive activities of Fosinopril.
Trandolapril Methysergide may decrease the antihypertensive activities of Trandolapril.
Metolazone Methysergide may decrease the antihypertensive activities of Metolazone.
Benazepril Methysergide may decrease the antihypertensive activities of Benazepril.
Cyclothiazide Methysergide may decrease the antihypertensive activities of Cyclothiazide.
Candoxatril Methysergide may decrease the antihypertensive activities of Candoxatril.
Mecamylamine Methysergide may decrease the antihypertensive activities of Mecamylamine.
Moexipril Methysergide may decrease the antihypertensive activities of Moexipril.
Lisinopril Methysergide may decrease the antihypertensive activities of Lisinopril.
Hydroflumethiazide Methysergide may decrease the antihypertensive activities of Hydroflumethiazide.
Cryptenamine Methysergide may decrease the antihypertensive activities of Cryptenamine.
Perindopril Methysergide may decrease the antihypertensive activities of Perindopril.
Candesartan cilexetil Methysergide may decrease the antihypertensive activities of Candesartan cilexetil.
Fenoldopam Methysergide may decrease the antihypertensive activities of Fenoldopam.
Eprosartan Methysergide may decrease the antihypertensive activities of Eprosartan.
Chlorothiazide Methysergide may decrease the antihypertensive activities of Chlorothiazide.
Quinapril Methysergide may decrease the antihypertensive activities of Quinapril.
Telmisartan Methysergide may decrease the antihypertensive activities of Telmisartan.
Hydrochlorothiazide Methysergide may decrease the antihypertensive activities of Hydrochlorothiazide.
Trichlormethiazide Methysergide may decrease the antihypertensive activities of Trichlormethiazide.
Deserpidine Methysergide may decrease the antihypertensive activities of Deserpidine.
Pentolinium Methysergide may decrease the antihypertensive activities of Pentolinium.
Trimethaphan Methysergide may decrease the antihypertensive activities of Trimethaphan.
Diazoxide Methysergide may decrease the antihypertensive activities of Diazoxide.
Bretylium Methysergide may decrease the antihypertensive activities of Bretylium.
Terazosin Methysergide may decrease the antihypertensive activities of Terazosin.
Captopril Methysergide may decrease the antihypertensive activities of Captopril.
Epoprostenol Methysergide may decrease the antihypertensive activities of Epoprostenol.
Polythiazide Methysergide may decrease the antihypertensive activities of Polythiazide.
Cilazapril Methysergide may decrease the antihypertensive activities of Cilazapril.
Saprisartan Methysergide may decrease the antihypertensive activities of Saprisartan.
Spirapril Methysergide may decrease the antihypertensive activities of Spirapril.
Tienilic acid Methysergide may decrease the antihypertensive activities of Tienilic acid.
Debrisoquine Methysergide may decrease the antihypertensive activities of Debrisoquine.
Diethylnorspermine Methysergide may decrease the antihypertensive activities of Diethylnorspermine.
Temocapril Methysergide may decrease the antihypertensive activities of Temocapril.
Trimazosin Methysergide may decrease the antihypertensive activities of Trimazosin.
Nicorandil Methysergide may decrease the antihypertensive activities of Nicorandil.
Rauwolfia serpentina root Methysergide may decrease the antihypertensive activities of Rauwolfia serpentina root.
Enalaprilat Methysergide may decrease the antihypertensive activities of Enalaprilat.
Angiotensin 1-7 Methysergide may decrease the antihypertensive activities of Angiotensin 1-7.
Imidapril Methysergide may decrease the antihypertensive activities of Imidapril.
BQ-123 Methysergide may decrease the antihypertensive activities of BQ-123.
Cicletanine Methysergide may decrease the antihypertensive activities of Cicletanine.
Dihydralazine Methysergide may decrease the antihypertensive activities of Dihydralazine.
Zofenopril Methysergide may decrease the antihypertensive activities of Zofenopril.
Guanoxan Methysergide may decrease the antihypertensive activities of Guanoxan.
Delapril Methysergide may decrease the antihypertensive activities of Delapril.
Vincamine Methysergide may decrease the antihypertensive activities of Vincamine.
Linsidomine Methysergide may decrease the antihypertensive activities of Linsidomine.
Guanoxabenz Methysergide may decrease the antihypertensive activities of Guanoxabenz.
Tolonidine Methysergide may decrease the antihypertensive activities of Tolonidine.
Endralazine Methysergide may decrease the antihypertensive activities of Endralazine.
Cadralazine Methysergide may decrease the antihypertensive activities of Cadralazine.
Cyclopenthiazide Methysergide may decrease the antihypertensive activities of Cyclopenthiazide.
Bietaserpine Methysergide may decrease the antihypertensive activities of Bietaserpine.
Guanazodine Methysergide may decrease the antihypertensive activities of Guanazodine.
Methoserpidine Methysergide may decrease the antihypertensive activities of Methoserpidine.
Guanoclor Methysergide may decrease the antihypertensive activities of Guanoclor.
Muzolimine Methysergide may decrease the antihypertensive activities of Muzolimine.
Xipamide Methysergide may decrease the antihypertensive activities of Xipamide.
Candesartan Methysergide may decrease the antihypertensive activities of Candesartan.
Tocopherylquinone Methysergide may decrease the antihypertensive activities of Tocopherylquinone.
Benazeprilat Methysergide may decrease the antihypertensive activities of Benazeprilat.
Fosinoprilat Methysergide may decrease the antihypertensive activities of Fosinoprilat.
Ramiprilat Methysergide may decrease the antihypertensive activities of Ramiprilat.
Perindoprilat Methysergide may decrease the antihypertensive activities of Perindoprilat.
Quinaprilat Methysergide may decrease the antihypertensive activities of Quinaprilat.
Furosemide Methysergide may decrease the antihypertensive activities of Furosemide.
Enalapril Methysergide may decrease the antihypertensive activities of Enalapril.
Amlodipine Methysergide may decrease the antihypertensive activities of Amlodipine.
Nimodipine Methysergide may decrease the antihypertensive activities of Nimodipine.
Lercanidipine Methysergide may decrease the antihypertensive activities of Lercanidipine.
Indapamide Methysergide may decrease the antihypertensive activities of Indapamide.
Nitrendipine Methysergide may decrease the antihypertensive activities of Nitrendipine.
Guanethidine Methysergide may decrease the antihypertensive activities of Guanethidine.
Bepridil Methysergide may decrease the antihypertensive activities of Bepridil.
Ambrisentan Methysergide may decrease the antihypertensive activities of Ambrisentan.
Pinacidil Methysergide may decrease the antihypertensive activities of Pinacidil.
Riociguat Methysergide may decrease the antihypertensive activities of Riociguat.
Macitentan Methysergide may decrease the antihypertensive activities of Macitentan.
Aliskiren Methysergide may decrease the antihypertensive activities of Aliskiren.
Lacidipine Methysergide may decrease the antihypertensive activities of Lacidipine.
Niguldipine Methysergide may decrease the antihypertensive activities of Niguldipine.
Selexipag Methysergide may decrease the antihypertensive activities of Selexipag.
Naftopidil Methysergide may decrease the antihypertensive activities of Naftopidil.

Target Protein

5-hydroxytryptamine receptor 2B HTR2B
5-hydroxytryptamine receptor 2C HTR2C
5-hydroxytryptamine receptor 2A HTR2A
5-hydroxytryptamine receptor 1A HTR1A
5-hydroxytryptamine receptor 7 HTR7
5-hydroxytryptamine receptor 1B HTR1B
5-hydroxytryptamine receptor 1F HTR1F
5-hydroxytryptamine receptor 1E HTR1E

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 2 • International brands: 2
Produk
  • Sansert
    Tablet, coated • 2 mg/1 • Oral • US • Approved
  • Sansert
    Tablet • 2 mg • Oral • Canada • Approved
International Brands
  • Deseril
  • Desernil

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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