Cevimeline

DB00185

small molecule approved

Deskripsi

Cevimeline is a parasympathomimetic agent that act as an agonist at the muscarinic acetylcholine receptors M1 and M3. It is indicated by the Food and Drug Administration for the treatment of dry mouth associated with Sjögren's syndrome.

Struktur Molekul 2D

Berat 199.313
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 5 ± 1 hours
Volume Distribusi * 6 L/kg
Klirens (Clearance) -

Absorpsi

Rapidly absorbed with peak concentration after 1.5 to 2 hours

Metabolisme

Primarily hepatic, isozymes CYP2D6 and CYP3A4 are responsible for the metabolism of cevimeline. Approximately 44.5% of the drug is converted to cis and trans-sulfoxide, 22.3% to glucuronic acid conjugate, and 4% to N-oxide of cevimeline. Approximately 8% of the trans-sulfoxide metabolite is then converted into the corresponding glucuronic acid conjugate.

Rute Eliminasi

After 24 hours, 84% of a 30 mg dose of cevimeline was excreted in urine.

Interaksi Obat

1105 Data
Mirabegron The serum concentration of Cevimeline can be increased when it is combined with Mirabegron.
Esmolol The risk or severity of adverse effects can be increased when Esmolol is combined with Cevimeline.
Betaxolol The risk or severity of adverse effects can be increased when Betaxolol is combined with Cevimeline.
Atenolol The risk or severity of adverse effects can be increased when Atenolol is combined with Cevimeline.
Alprenolol The risk or severity of adverse effects can be increased when Alprenolol is combined with Cevimeline.
Bevantolol The risk or severity of adverse effects can be increased when Bevantolol is combined with Cevimeline.
Practolol The risk or severity of adverse effects can be increased when Practolol is combined with Cevimeline.
Dexpropranolol The risk or severity of adverse effects can be increased when Dexpropranolol is combined with Cevimeline.
Celiprolol The risk or severity of adverse effects can be increased when Celiprolol is combined with Cevimeline.
Bufuralol The risk or severity of adverse effects can be increased when Bufuralol is combined with Cevimeline.
Bopindolol The risk or severity of adverse effects can be increased when Bopindolol is combined with Cevimeline.
Bupranolol The risk or severity of adverse effects can be increased when Bupranolol is combined with Cevimeline.
Indenolol The risk or severity of adverse effects can be increased when Indenolol is combined with Cevimeline.
Levobetaxolol The risk or severity of adverse effects can be increased when Levobetaxolol is combined with Cevimeline.
Talinolol The risk or severity of adverse effects can be increased when Talinolol is combined with Cevimeline.
Anisodamine The risk or severity of adverse effects can be increased when Anisodamine is combined with Cevimeline.
Bucindolol The risk or severity of adverse effects can be increased when Bucindolol is combined with Cevimeline.
Esatenolol The risk or severity of adverse effects can be increased when Esatenolol is combined with Cevimeline.
Cloranolol The risk or severity of adverse effects can be increased when Cloranolol is combined with Cevimeline.
Mepindolol The risk or severity of adverse effects can be increased when Mepindolol is combined with Cevimeline.
Epanolol The risk or severity of adverse effects can be increased when Epanolol is combined with Cevimeline.
Tertatolol The risk or severity of adverse effects can be increased when Tertatolol is combined with Cevimeline.
Timolol The risk or severity of adverse effects can be increased when Timolol is combined with Cevimeline.
Propranolol The risk or severity of adverse effects can be increased when Propranolol is combined with Cevimeline.
Bisoprolol The risk or severity of adverse effects can be increased when Bisoprolol is combined with Cevimeline.
Pindolol The risk or severity of adverse effects can be increased when Pindolol is combined with Cevimeline.
Nadolol The risk or severity of adverse effects can be increased when Nadolol is combined with Cevimeline.
Penbutolol The risk or severity of adverse effects can be increased when Penbutolol is combined with Cevimeline.
Arotinolol The risk or severity of adverse effects can be increased when Arotinolol is combined with Cevimeline.
Carvedilol The risk or severity of adverse effects can be increased when Carvedilol is combined with Cevimeline.
Nebivolol The risk or severity of adverse effects can be increased when Nebivolol is combined with Cevimeline.
Landiolol The risk or severity of adverse effects can be increased when Landiolol is combined with Cevimeline.
Cimetropium Cevimeline may decrease the anticholinergic activities of Cimetropium.
Tacrine The risk or severity of adverse effects can be increased when Tacrine is combined with Cevimeline.
Sulpiride The risk or severity of adverse effects can be increased when Sulpiride is combined with Cevimeline.
Profenamine The risk or severity of adverse effects can be increased when Profenamine is combined with Cevimeline.
Gallamine triethiodide The risk or severity of adverse effects can be increased when Gallamine triethiodide is combined with Cevimeline.
Triflupromazine The risk or severity of adverse effects can be increased when Triflupromazine is combined with Cevimeline.
Cinchocaine The risk or severity of adverse effects can be increased when Cinchocaine is combined with Cevimeline.
Nizatidine The risk or severity of adverse effects can be increased when Nizatidine is combined with Cevimeline.
Isoflurophate The risk or severity of adverse effects can be increased when Isoflurophate is combined with Cevimeline.
Diethylcarbamazine The risk or severity of adverse effects can be increased when Diethylcarbamazine is combined with Cevimeline.
Procaine The risk or severity of adverse effects can be increased when Procaine is combined with Cevimeline.
Mechlorethamine The risk or severity of adverse effects can be increased when Mechlorethamine is combined with Cevimeline.
Hexafluronium The risk or severity of adverse effects can be increased when Hexafluronium is combined with Cevimeline.
Demecarium The risk or severity of adverse effects can be increased when Demecarium is combined with Cevimeline.
Physostigmine The risk or severity of adverse effects can be increased when Physostigmine is combined with Cevimeline.
Ambenonium The risk or severity of adverse effects can be increased when Ambenonium is combined with Cevimeline.
Tubocurarine The risk or severity of adverse effects can be increased when Tubocurarine is combined with Cevimeline.
Decamethonium The risk or severity of adverse effects can be increased when Decamethonium is combined with Cevimeline.
Pancuronium The risk or severity of adverse effects can be increased when Pancuronium is combined with Cevimeline.
Pipecuronium The risk or severity of adverse effects can be increased when Pipecuronium is combined with Cevimeline.
Ginkgo biloba The risk or severity of adverse effects can be increased when Ginkgo biloba is combined with Cevimeline.
Neostigmine The risk or severity of adverse effects can be increased when Neostigmine is combined with Cevimeline.
Bambuterol The risk or severity of adverse effects can be increased when Bambuterol is combined with Cevimeline.
1,10-Phenanthroline The risk or severity of adverse effects can be increased when 1,10-Phenanthroline is combined with Cevimeline.
Huperzine A The risk or severity of adverse effects can be increased when Huperzine A is combined with Cevimeline.
Phenserine The risk or severity of adverse effects can be increased when Phenserine is combined with Cevimeline.
Regramostim The risk or severity of adverse effects can be increased when Regramostim is combined with Cevimeline.
Aprotinin The risk or severity of adverse effects can be increased when Aprotinin is combined with Cevimeline.
Betaine The risk or severity of adverse effects can be increased when Betaine is combined with Cevimeline.
Coumaphos The risk or severity of adverse effects can be increased when Coumaphos is combined with Cevimeline.
Dichlorvos The risk or severity of adverse effects can be increased when Dichlorvos is combined with Cevimeline.
Fenthion The risk or severity of adverse effects can be increased when Fenthion is combined with Cevimeline.
Metrifonate The risk or severity of adverse effects can be increased when Metrifonate is combined with Cevimeline.
Acotiamide The risk or severity of adverse effects can be increased when Acotiamide is combined with Cevimeline.
Methanesulfonyl Fluoride The risk or severity of adverse effects can be increased when Methanesulfonyl Fluoride is combined with Cevimeline.
Paraoxon The risk or severity of adverse effects can be increased when Paraoxon is combined with Cevimeline.
Tyrothricin The risk or severity of adverse effects can be increased when Tyrothricin is combined with Cevimeline.
Ipidacrine The risk or severity of adverse effects can be increased when Ipidacrine is combined with Cevimeline.
Distigmine The risk or severity of adverse effects can be increased when Distigmine is combined with Cevimeline.
Tretamine The risk or severity of adverse effects can be increased when Tretamine is combined with Cevimeline.
Posiphen The risk or severity of adverse effects can be increased when Posiphen is combined with Cevimeline.
Pyridostigmine The risk or severity of adverse effects can be increased when Pyridostigmine is combined with Cevimeline.
Rivastigmine The risk or severity of adverse effects can be increased when Rivastigmine is combined with Cevimeline.
Methylphosphinic Acid The risk or severity of adverse effects can be increased when Methylphosphinic Acid is combined with Cevimeline.
Pegvisomant The risk or severity of adverse effects can be increased when Pegvisomant is combined with Cevimeline.
Mefloquine The risk or severity of adverse effects can be increased when Mefloquine is combined with Cevimeline.
Thiotepa The risk or severity of adverse effects can be increased when Thiotepa is combined with Cevimeline.
Capsaicin The risk or severity of adverse effects can be increased when Capsaicin is combined with Cevimeline.
Celecoxib The metabolism of Cevimeline can be decreased when combined with Celecoxib.
Fluvoxamine The metabolism of Cevimeline can be decreased when combined with Fluvoxamine.
Metoprolol The metabolism of Cevimeline can be decreased when combined with Metoprolol.
Venlafaxine Cevimeline may decrease the excretion rate of Venlafaxine which could result in a higher serum level.
Clobazam The serum concentration of Cevimeline can be increased when it is combined with Clobazam.
Clozapine The serum concentration of Cevimeline can be increased when it is combined with Clozapine.
Duloxetine The metabolism of Cevimeline can be decreased when combined with Duloxetine.
Chlorpromazine The metabolism of Cevimeline can be decreased when combined with Chlorpromazine.
Cimetidine Cevimeline may decrease the excretion rate of Cimetidine which could result in a higher serum level.
Chloroquine The metabolism of Cevimeline can be decreased when combined with Chloroquine.
Nicardipine The metabolism of Cevimeline can be decreased when combined with Nicardipine.
Primaquine The metabolism of Cevimeline can be decreased when combined with Primaquine.
Fusidic acid The metabolism of Cevimeline can be decreased when combined with Fusidic acid.
Cholecalciferol The metabolism of Cevimeline can be decreased when combined with Cholecalciferol.
Tranylcypromine The metabolism of Cevimeline can be decreased when combined with Tranylcypromine.
Perhexiline The metabolism of Cevimeline can be decreased when combined with Perhexiline.
Tegaserod The metabolism of Cevimeline can be decreased when combined with Tegaserod.
Abiraterone The metabolism of Cevimeline can be decreased when combined with Abiraterone.
Panobinostat The metabolism of Cevimeline can be decreased when combined with Panobinostat.
Vilazodone The metabolism of Cevimeline can be decreased when combined with Vilazodone.

Target Protein

Muscarinic acetylcholine receptor M3 CHRM3
Muscarinic acetylcholine receptor M1 CHRM1

Contoh Produk & Brand

Produk: 19 • International brands: 1
Produk
  • Cevimeline
    Capsule • 30 mg/1 • Oral • US • Approved
  • Cevimeline
    Capsule • 30 mg/1 • Oral • US • Generic • Approved
  • Cevimeline Hydrochloride
    Capsule • 30 mg/1 • Oral • US • Generic • Approved
  • Cevimeline Hydrochloride
    Capsule • 30 mg/1 • Oral • US • Approved
  • Cevimeline Hydrochloride
    Capsule • 30 mg/1 • Oral • US • Generic • Approved
  • Cevimeline Hydrochloride
    Capsule • 30 mg/1 • Oral • US • Generic • Approved
  • Cevimeline Hydrochloride
    Capsule • 30 mg/1 • Oral • US • Generic • Approved
  • Cevimeline Hydrochloride
    Capsule • 30 mg/1 • Oral • US • Generic • Approved
Menampilkan 8 dari 19 produk.
International Brands
  • Saligren

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul