Peringatan Keamanan

Menadione (vitamin K3), which is not used as a nutritional supplemental form of vitamin K for humans, has been reported to cause adverse reactions, including hemolytic anemia. Large doses have also been reported to cause brain damage.

Menadione

DB00170

small molecule approved nutraceutical

Deskripsi

A synthetic naphthoquinone without the isoprenoid side chain and biological activity, but can be converted to active vitamin K2, menaquinone, after alkylation in vivo.

Struktur Molekul 2D

Berat 172.18
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Variable and ranges from 10% to 80%

Metabolisme

Hepatic

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

57 Data
Orlistat Orlistat can cause a decrease in the absorption of Menadione resulting in a reduced serum concentration and potentially a decrease in efficacy.
Alpha-1-proteinase inhibitor Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Menadione.
Tranexamic acid Menadione may increase the thrombogenic activities of Tranexamic acid.
Aminocaproic acid Menadione may increase the thrombogenic activities of Aminocaproic acid.
Aprotinin Menadione may increase the thrombogenic activities of Aprotinin.
Hydrogen peroxide Menadione may increase the thrombogenic activities of Hydrogen peroxide.
Aminomethylbenzoic acid Menadione may increase the thrombogenic activities of Aminomethylbenzoic acid.
Camostat Menadione may increase the thrombogenic activities of Camostat.
Menadione bisulfite Menadione may increase the thrombogenic activities of Menadione bisulfite.
Fibrinogen human The therapeutic efficacy of Fibrinogen human can be increased when used in combination with Menadione.
Tretinoin The risk or severity of Thrombosis can be increased when Menadione is combined with Tretinoin.
Antihemophilic factor, human recombinant Menadione may increase the thrombogenic activities of Antihemophilic factor, human recombinant.
Coagulation factor VIIa Recombinant Human Menadione may increase the thrombogenic activities of Coagulation factor VIIa Recombinant Human.
Coagulation Factor IX (Recombinant) Menadione may increase the thrombogenic activities of Coagulation Factor IX (Recombinant).
Calcium Menadione may increase the thrombogenic activities of Calcium.
Pantothenic acid Menadione may increase the thrombogenic activities of Pantothenic acid.
Formic acid Menadione may increase the thrombogenic activities of Formic acid.
Platelet Activating Factor Menadione may increase the thrombogenic activities of Platelet Activating Factor.
Turoctocog alfa Menadione may increase the thrombogenic activities of Turoctocog alfa.
Catridecacog Menadione may increase the thrombogenic activities of Catridecacog.
Antihemophilic factor (recombinant), PEGylated Menadione may increase the thrombogenic activities of Antihemophilic factor (recombinant), PEGylated.
Prothrombin Menadione may increase the thrombogenic activities of Prothrombin.
Factor IX Complex (Human) Menadione may increase the thrombogenic activities of Factor IX Complex (Human).
Susoctocog alfa Menadione may increase the thrombogenic activities of Susoctocog alfa.
Eftrenonacog alfa Menadione may increase the thrombogenic activities of Eftrenonacog alfa.
Rusalatide acetate Menadione may increase the thrombogenic activities of Rusalatide acetate.
Vatreptacog alfa Menadione may increase the thrombogenic activities of Vatreptacog alfa.
Factor XIII (human) Menadione may increase the thrombogenic activities of Factor XIII (human).
Von Willebrand factor human Menadione may increase the thrombogenic activities of Von Willebrand factor human.
Coagulation factor X human Menadione may increase the thrombogenic activities of Coagulation factor X human.
Coagulation factor VII human Menadione may increase the thrombogenic activities of Coagulation factor VII human.
Anti-inhibitor coagulant complex Menadione may increase the thrombogenic activities of Anti-inhibitor coagulant complex.
Coagulation Factor IX Human Menadione may increase the thrombogenic activities of Coagulation Factor IX Human.
Antihemophilic factor human Menadione may increase the thrombogenic activities of Antihemophilic factor human.
Kallidinogenase Menadione may increase the thrombogenic activities of Kallidinogenase.
Trenonacog alfa Menadione may increase the thrombogenic activities of Trenonacog alfa.
Albutrepenonacog alfa Menadione may increase the thrombogenic activities of Albutrepenonacog alfa.
Emicizumab Menadione may increase the thrombogenic activities of Emicizumab.
Nonacog beta pegol Menadione may increase the thrombogenic activities of Nonacog beta pegol.
Moroctocog alfa Menadione may increase the thrombogenic activities of Moroctocog alfa.
Beroctocog alfa Menadione may increase the thrombogenic activities of Beroctocog alfa.
Andexanet alfa Menadione may increase the thrombogenic activities of Andexanet alfa.
Calcium cation Menadione may increase the thrombogenic activities of Calcium cation.
Damoctocog alfa pegol Menadione may increase the thrombogenic activities of Damoctocog alfa pegol.
Turoctocog alfa pegol Menadione may increase the thrombogenic activities of Turoctocog alfa pegol.
Alteplase The therapeutic efficacy of Menadione can be decreased when used in combination with Alteplase.
Urokinase The therapeutic efficacy of Menadione can be decreased when used in combination with Urokinase.
Reteplase The therapeutic efficacy of Menadione can be decreased when used in combination with Reteplase.
Anistreplase The therapeutic efficacy of Menadione can be decreased when used in combination with Anistreplase.
Tenecteplase The therapeutic efficacy of Menadione can be decreased when used in combination with Tenecteplase.
Streptokinase The therapeutic efficacy of Menadione can be decreased when used in combination with Streptokinase.
Lanoteplase The therapeutic efficacy of Menadione can be decreased when used in combination with Lanoteplase.
Amediplase The therapeutic efficacy of Menadione can be decreased when used in combination with Amediplase.
Saruplase The therapeutic efficacy of Menadione can be decreased when used in combination with Saruplase.
Protein S human Menadione may increase the thrombogenic activities of Protein S human.
Rurioctocog alfa pegol Menadione may increase the thrombogenic activities of Rurioctocog alfa pegol.
Etranacogene dezaparvovec Menadione may increase the thrombogenic activities of Etranacogene dezaparvovec.

Target Protein

Aldehyde oxidase AOX1
Vitamin K-dependent gamma-carboxylase GGCX
Vitamin K epoxide reductase complex subunit 1 VKORC1
Vitamin K epoxide reductase complex subunit 1-like protein 1 VKORC1L1
Prothrombin F2
Coagulation factor IX F9
Vitamin K-dependent protein C PROC
Vitamin K-dependent protein S PROS1
Ribosyldihydronicotinamide dehydrogenase [quinone] NQO2
NAD(P)H dehydrogenase [quinone] 1 NQO1
Osteocalcin BGLAP

Referensi & Sumber

Synthesis reference: Joachim U. Schneider, Hans Kiefer, "Menadione choline bisulfite adduct, its preparation and antihemorrhagic compositions." U.S. Patent US4735969, issued January, 1980.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Synkavite

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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