Peringatan Keamanan

Thiamine toxicity is uncommon; as excesses are readily excreted, although long-term supplementation of amounts larger than 3 gram have been known to cause toxicity. Oral mouse LD50 = 8224 mg/kg, oral rat LD50 = 3710 mg/kg.

Thiamine

DB00152

small molecule approved investigational nutraceutical vet_approved

Deskripsi

Thiamine or thiamin, also known as vitamin B1, is a colorless compound with the chemical formula C12H17N4OS. It is soluble in water and insoluble in alcohol. Thiamine decomposes if heated. Thiamine was first discovered by Umetaro Suzuki in Japan when researching how rice bran cured patients of Beriberi. Thiamine plays a key role in intracellular glucose metabolism and it is thought that thiamine inhibits the effect of glucose and insulin on arterial smooth muscle cell proliferation. Thiamine plays an important role in helping the body convert carbohydrates and fat into energy. It is essential for normal growth and development and helps to maintain proper functioning of the heart and the nervous and digestive systems. Thiamine cannot be stored in the body; however, once absorbed, the vitamin is concentrated in muscle tissue.

Struktur Molekul 2D

Berat 265.355
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Absorbed mainly from duodenum, by both active and passive processes

Metabolisme

Hepatic

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

68 Data
Tipiracil The excretion of Tipiracil can be decreased when combined with Thiamine.
Varenicline The excretion of Varenicline can be decreased when combined with Thiamine.
Prazosin The serum concentration of Prazosin can be increased when it is combined with Thiamine.
Solriamfetol The serum concentration of Solriamfetol can be increased when it is combined with Thiamine.
Ranitidine The serum concentration of Ranitidine can be increased when it is combined with Thiamine.
Linagliptin The serum concentration of Linagliptin can be increased when it is combined with Thiamine.
Choline salicylate The serum concentration of Choline salicylate can be increased when it is combined with Thiamine.
Metformin The serum concentration of Metformin can be increased when it is combined with Thiamine.
Norepinephrine The serum concentration of Norepinephrine can be increased when it is combined with Thiamine.
Reserpine The serum concentration of Reserpine can be increased when it is combined with Thiamine.
Pramipexole The serum concentration of Pramipexole can be increased when it is combined with Thiamine.
Cimetidine The risk or severity of adverse effects can be increased when Cimetidine is combined with Thiamine.
Epinephrine The serum concentration of Epinephrine can be increased when it is combined with Thiamine.
Lamivudine The serum concentration of Lamivudine can be increased when it is combined with Thiamine.
Amantadine The serum concentration of Amantadine can be increased when it is combined with Thiamine.
Dopamine The serum concentration of Dopamine can be increased when it is combined with Thiamine.
Memantine The serum concentration of Memantine can be increased when it is combined with Thiamine.
Histamine The serum concentration of Histamine can be increased when it is combined with Thiamine.
Agmatine The serum concentration of Agmatine can be increased when it is combined with Thiamine.
Nafamostat The serum concentration of Nafamostat can be increased when it is combined with Thiamine.
Nicotine The risk or severity of adverse effects can be increased when Nicotine is combined with Thiamine.
Nelfinavir The risk or severity of adverse effects can be increased when Nelfinavir is combined with Thiamine.
Indinavir The risk or severity of adverse effects can be increased when Indinavir is combined with Thiamine.
Nevirapine The risk or severity of adverse effects can be increased when Nevirapine is combined with Thiamine.
Disopyramide The risk or severity of adverse effects can be increased when Disopyramide is combined with Thiamine.
Codeine The risk or severity of adverse effects can be increased when Codeine is combined with Thiamine.
Progesterone The risk or severity of adverse effects can be increased when Progesterone is combined with Thiamine.
Quinine The risk or severity of adverse effects can be increased when Quinine is combined with Thiamine.
Guanidine The risk or severity of adverse effects can be increased when Guanidine is combined with Thiamine.
Doxazosin The risk or severity of adverse effects can be increased when Doxazosin is combined with Thiamine.
Efavirenz The risk or severity of adverse effects can be increased when Efavirenz is combined with Thiamine.
Verapamil The risk or severity of adverse effects can be increased when Verapamil is combined with Thiamine.
Rocuronium The risk or severity of adverse effects can be increased when Rocuronium is combined with Thiamine.
Clopidogrel The risk or severity of adverse effects can be increased when Clopidogrel is combined with Thiamine.
Acyclovir The risk or severity of adverse effects can be increased when Acyclovir is combined with Thiamine.
Quinidine The risk or severity of adverse effects can be increased when Quinidine is combined with Thiamine.
Phenformin The risk or severity of adverse effects can be increased when Phenformin is combined with Thiamine.
Dinoprostone The risk or severity of adverse effects can be increased when Dinoprostone is combined with Thiamine.
Phenoxybenzamine The risk or severity of adverse effects can be increased when Phenoxybenzamine is combined with Thiamine.
Ganciclovir The risk or severity of adverse effects can be increased when Ganciclovir is combined with Thiamine.
Probenecid The risk or severity of adverse effects can be increased when Probenecid is combined with Thiamine.
Chlorpheniramine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Thiamine.
Desipramine The risk or severity of adverse effects can be increased when Desipramine is combined with Thiamine.
Saquinavir The risk or severity of adverse effects can be increased when Saquinavir is combined with Thiamine.
Pancuronium The risk or severity of adverse effects can be increased when Pancuronium is combined with Thiamine.
Palbociclib The risk or severity of adverse effects can be increased when Palbociclib is combined with Thiamine.
Dexchlorpheniramine maleate The risk or severity of adverse effects can be increased when Dexchlorpheniramine maleate is combined with Thiamine.
Pitolisant The risk or severity of adverse effects can be increased when Pitolisant is combined with Thiamine.
Dacomitinib The risk or severity of adverse effects can be increased when Dacomitinib is combined with Thiamine.
Gilteritinib The risk or severity of adverse effects can be increased when Gilteritinib is combined with Thiamine.
Estradiol acetate The risk or severity of adverse effects can be increased when Estradiol acetate is combined with Thiamine.
Estradiol benzoate The risk or severity of adverse effects can be increased when Estradiol benzoate is combined with Thiamine.
Estradiol cypionate The risk or severity of adverse effects can be increased when Estradiol cypionate is combined with Thiamine.
Estradiol dienanthate The risk or severity of adverse effects can be increased when Estradiol dienanthate is combined with Thiamine.
Estradiol valerate The risk or severity of adverse effects can be increased when Estradiol valerate is combined with Thiamine.
Dronedarone The risk or severity of adverse effects can be increased when Dronedarone is combined with Thiamine.
Formoterol The risk or severity of adverse effects can be increased when Formoterol is combined with Thiamine.
Guanfacine The risk or severity of adverse effects can be increased when Guanfacine is combined with Thiamine.
Salmeterol The risk or severity of adverse effects can be increased when Salmeterol is combined with Thiamine.
Dofetilide The serum concentration of Dofetilide can be increased when it is combined with Thiamine.
Cisplatin The serum concentration of Cisplatin can be increased when it is combined with Thiamine.
Oxaliplatin The serum concentration of Oxaliplatin can be increased when it is combined with Thiamine.
Procainamide The serum concentration of Procainamide can be increased when it is combined with Thiamine.
Dalfampridine The serum concentration of Dalfampridine can be increased when it is combined with Thiamine.
Clofarabine The serum concentration of Clofarabine can be increased when it is combined with Thiamine.
Gentamicin The serum concentration of Gentamicin can be increased when it is combined with Thiamine.
Pacritinib The serum concentration of Thiamine can be increased when it is combined with Pacritinib.
Patiromer Patiromer can cause a decrease in the absorption of Thiamine resulting in a reduced serum concentration and potentially a decrease in efficacy.

Target Protein

Thiamine pyrophosphokinase 1 TPK1
Pyruvate dehydrogenase E1 component aceE

Referensi & Sumber

Synthesis reference: Nobuyuki Kitamori, Masaya Maeno, Seiji Izuhara, "Granules of thiamine salt and the production thereof." U.S. Patent US4702919, issued July, 1974.
Artikel (PubMed)

Contoh Produk & Brand

Produk: 1327 • International brands: 2
Produk
  • 24 Multivitamins + Minerals
    Tablet • - • Oral • Canada • OTC • Approved
  • 50 Plus
    Tablet • - • Oral • Canada • OTC • Approved
  • 50 Plus Multiple Vitamins & Minerals
    Tablet • - • Oral • Canada • OTC • Approved
  • Abavite
    Tablet • - • Oral • US
  • Acti-MN + B1 + C Caplet
    Tablet • - • Oral • Canada • OTC • Approved
  • Acti-thiamine Caplet 100mg
    Tablet • 100 mg • Oral • Canada • OTC • Approved
  • Active FE
    Tablet • - • Oral • US
  • Active FE
    Tablet • - • Oral • US
Menampilkan 8 dari 1327 produk.
International Brands
  • Betalin S — Eli Lilly
  • Biamine

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul