Daclizumab

DB00111

biotech investigational withdrawn

Deskripsi

Humanized IgG1 Mab that binds to the human interleukin-2 receptor (anti-Tac or anti-CD25). Daclizumab is a composite of human (90%) and murine (10%) antibody sequences. The human sequences were derived from the constant domains of human IgG1 and the variable framework regions of the Eu myeloma antibody. The murine sequences were derived from the complementarity-determining regions of a murine anti-Tac antibody.

On 22 April 2008, Roche Registration Limited chose to voluntarily withdraw the marketing authorization for their product Zenapax (daclizumab), as indicated for the prophylaxis of acute organ rejection in de novo allogeneic renal transplantation and used concomitantly with an immunosuppressive regimen like cyclosporine and corticosteroids in patients who are not hight immunized, for commercial reasons and confirmed that this decision was not related to any safety concerns associated with the use of Zenapax (daclizumab) L1744. Regardless of the withdrawal of Zenapax, Biogen and Abbvie's Zinbryta (daclizumab), as indicated for the treatment of adult patients with relapsing forms of multiple sclerosis, was approved for use by the FDA in 2016 L1746.

Despite being approved for use, Zinbryta (daclizumab)'s complex pre-existing safety profile consisting of its restricted availability through a Risk Evaluation and Mitigation Strategy program L1738 and its black box warning for possible hepatic injury, autoimmune hepatitis, and other immune mediated disorders L1738 meant its therapeutic usage, adverse effects, and prescribing information was subject to continuous monitoring and updating.

Although Zinbryta (daclizumab) was available for patients as needed until 30 April 2018, Biogen and Abbvie announced a voluntary withdrawal of their product Zinbryta (daclizumab) from the global market on 2 March 2018 L1738. This withdrawal was concurrent to the European Medicines Agency announcement of a recall owing to 12 worldwide reports of serious inflammatory brain disorders associated with the use of Zinbryta (daclizumab) L1738.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 11-38 days
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Most likely removed by opsonization via the reticuloendothelial system when bound to lymphocytes.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

670 Data
Denosumab The risk or severity of adverse effects can be increased when Denosumab is combined with Daclizumab.
Etanercept The risk or severity of adverse effects can be increased when Etanercept is combined with Daclizumab.
Peginterferon alfa-2a The risk or severity of adverse effects can be increased when Peginterferon alfa-2a is combined with Daclizumab.
Interferon alfa-n1 The risk or severity of adverse effects can be increased when Interferon alfa-n1 is combined with Daclizumab.
Interferon alfa-n3 The risk or severity of adverse effects can be increased when Interferon alfa-n3 is combined with Daclizumab.
Peginterferon alfa-2b The risk or severity of adverse effects can be increased when Peginterferon alfa-2b is combined with Daclizumab.
Anakinra The risk or severity of adverse effects can be increased when Anakinra is combined with Daclizumab.
Interferon gamma-1b The risk or severity of adverse effects can be increased when Interferon gamma-1b is combined with Daclizumab.
Interferon alfa-2a The risk or severity of adverse effects can be increased when Interferon alfa-2a is combined with Daclizumab.
Aldesleukin The risk or severity of adverse effects can be increased when Aldesleukin is combined with Daclizumab.
Adalimumab The risk or severity of adverse effects can be increased when Adalimumab is combined with Daclizumab.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Daclizumab.
Pegaspargase The risk or severity of adverse effects can be increased when Pegaspargase is combined with Daclizumab.
Infliximab The risk or severity of adverse effects can be increased when Infliximab is combined with Daclizumab.
Interferon beta-1b The risk or severity of adverse effects can be increased when Interferon beta-1b is combined with Daclizumab.
Interferon alfacon-1 The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Daclizumab.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Daclizumab.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Daclizumab.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Daclizumab.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Daclizumab.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Daclizumab.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Daclizumab.
Alefacept The risk or severity of adverse effects can be increased when Alefacept is combined with Daclizumab.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Daclizumab.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Daclizumab.
Interferon alfa-2b The risk or severity of adverse effects can be increased when Interferon alfa-2b is combined with Daclizumab.
Phenylalanine The risk or severity of adverse effects can be increased when Daclizumab is combined with Phenylalanine.
Flunisolide The risk or severity of adverse effects can be increased when Daclizumab is combined with Flunisolide.
Bortezomib The risk or severity of adverse effects can be increased when Daclizumab is combined with Bortezomib.
Cladribine Daclizumab may increase the immunosuppressive activities of Cladribine.
Carmustine The risk or severity of adverse effects can be increased when Daclizumab is combined with Carmustine.
Amsacrine The risk or severity of adverse effects can be increased when Daclizumab is combined with Amsacrine.
Bleomycin The risk or severity of adverse effects can be increased when Daclizumab is combined with Bleomycin.
Chlorambucil The risk or severity of adverse effects can be increased when Daclizumab is combined with Chlorambucil.
Raltitrexed The risk or severity of adverse effects can be increased when Daclizumab is combined with Raltitrexed.
Mitomycin The risk or severity of adverse effects can be increased when Daclizumab is combined with Mitomycin.
Bexarotene The risk or severity of adverse effects can be increased when Daclizumab is combined with Bexarotene.
Vindesine The risk or severity of adverse effects can be increased when Daclizumab is combined with Vindesine.
Floxuridine The risk or severity of adverse effects can be increased when Daclizumab is combined with Floxuridine.
Indomethacin The risk or severity of adverse effects can be increased when Daclizumab is combined with Indomethacin.
Tioguanine The risk or severity of adverse effects can be increased when Daclizumab is combined with Tioguanine.
Vinorelbine The risk or severity of adverse effects can be increased when Daclizumab is combined with Vinorelbine.
Dexrazoxane The risk or severity of adverse effects can be increased when Daclizumab is combined with Dexrazoxane.
Beclomethasone dipropionate The risk or severity of adverse effects can be increased when Daclizumab is combined with Beclomethasone dipropionate.
Sorafenib The risk or severity of adverse effects can be increased when Daclizumab is combined with Sorafenib.
Streptozocin The risk or severity of adverse effects can be increased when Daclizumab is combined with Streptozocin.
Trifluridine The risk or severity of adverse effects can be increased when Daclizumab is combined with Trifluridine.
Gemcitabine The risk or severity of adverse effects can be increased when Daclizumab is combined with Gemcitabine.
Betamethasone The risk or severity of adverse effects can be increased when Daclizumab is combined with Betamethasone.
Teniposide The risk or severity of adverse effects can be increased when Daclizumab is combined with Teniposide.
Epirubicin The risk or severity of adverse effects can be increased when Daclizumab is combined with Epirubicin.
Chloramphenicol The risk or severity of adverse effects can be increased when Daclizumab is combined with Chloramphenicol.
Lenalidomide The risk or severity of adverse effects can be increased when Daclizumab is combined with Lenalidomide.
Altretamine The risk or severity of adverse effects can be increased when Daclizumab is combined with Altretamine.
Zidovudine The risk or severity of adverse effects can be increased when Daclizumab is combined with Zidovudine.
Cisplatin The risk or severity of adverse effects can be increased when Daclizumab is combined with Cisplatin.
Oxaliplatin The risk or severity of adverse effects can be increased when Daclizumab is combined with Oxaliplatin.
Cyclophosphamide The risk or severity of adverse effects can be increased when Daclizumab is combined with Cyclophosphamide.
Vincristine The risk or severity of adverse effects can be increased when Daclizumab is combined with Vincristine.
Fluorouracil The risk or severity of adverse effects can be increased when Daclizumab is combined with Fluorouracil.
Propylthiouracil The risk or severity of adverse effects can be increased when Daclizumab is combined with Propylthiouracil.
Pentostatin The risk or severity of adverse effects can be increased when Daclizumab is combined with Pentostatin.
Methotrexate The risk or severity of adverse effects can be increased when Daclizumab is combined with Methotrexate.
Carbamazepine The risk or severity of adverse effects can be increased when Daclizumab is combined with Carbamazepine.
Vinblastine The risk or severity of adverse effects can be increased when Daclizumab is combined with Vinblastine.
Fluticasone propionate The risk or severity of adverse effects can be increased when Daclizumab is combined with Fluticasone propionate.
Fluocinolone acetonide The risk or severity of adverse effects can be increased when Daclizumab is combined with Fluocinolone acetonide.
Linezolid The risk or severity of adverse effects can be increased when Daclizumab is combined with Linezolid.
Imatinib The risk or severity of adverse effects can be increased when Daclizumab is combined with Imatinib.
Triamcinolone The risk or severity of adverse effects can be increased when Daclizumab is combined with Triamcinolone.
Clofarabine The risk or severity of adverse effects can be increased when Daclizumab is combined with Clofarabine.
Prednisone The risk or severity of adverse effects can be increased when Daclizumab is combined with Prednisone.
Pemetrexed The risk or severity of adverse effects can be increased when Daclizumab is combined with Pemetrexed.
Fludrocortisone The risk or severity of adverse effects can be increased when Daclizumab is combined with Fludrocortisone.
Mycophenolate mofetil The risk or severity of adverse effects can be increased when Daclizumab is combined with Mycophenolate mofetil.
Daunorubicin The risk or severity of adverse effects can be increased when Daclizumab is combined with Daunorubicin.
Irinotecan The risk or severity of adverse effects can be increased when Daclizumab is combined with Irinotecan.
Methimazole The risk or severity of adverse effects can be increased when Daclizumab is combined with Methimazole.
Etoposide The risk or severity of adverse effects can be increased when Daclizumab is combined with Etoposide.
Sulfasalazine The risk or severity of adverse effects can be increased when Daclizumab is combined with Sulfasalazine.
Dacarbazine The risk or severity of adverse effects can be increased when Daclizumab is combined with Dacarbazine.
Temozolomide The risk or severity of adverse effects can be increased when Daclizumab is combined with Temozolomide.
Penicillamine The risk or severity of adverse effects can be increased when Daclizumab is combined with Penicillamine.
Prednisolone The risk or severity of adverse effects can be increased when Daclizumab is combined with Prednisolone.
Sirolimus The risk or severity of adverse effects can be increased when Daclizumab is combined with Sirolimus.
Mechlorethamine The risk or severity of adverse effects can be increased when Daclizumab is combined with Mechlorethamine.
Azacitidine The risk or severity of adverse effects can be increased when Daclizumab is combined with Azacitidine.
Carboplatin The risk or severity of adverse effects can be increased when Daclizumab is combined with Carboplatin.
Methylprednisolone The risk or severity of adverse effects can be increased when Daclizumab is combined with Methylprednisolone.
Dactinomycin The risk or severity of adverse effects can be increased when Daclizumab is combined with Dactinomycin.
Cytarabine The risk or severity of adverse effects can be increased when Daclizumab is combined with Cytarabine.
Azathioprine The risk or severity of adverse effects can be increased when Daclizumab is combined with Azathioprine.
Doxorubicin The risk or severity of adverse effects can be increased when Daclizumab is combined with Doxorubicin.
Hydroxyurea The risk or severity of adverse effects can be increased when Daclizumab is combined with Hydroxyurea.
Busulfan The risk or severity of adverse effects can be increased when Daclizumab is combined with Busulfan.
Mycophenolic acid The risk or severity of adverse effects can be increased when Daclizumab is combined with Mycophenolic acid.
Topotecan The risk or severity of adverse effects can be increased when Daclizumab is combined with Topotecan.
Mercaptopurine The risk or severity of adverse effects can be increased when Daclizumab is combined with Mercaptopurine.
Thalidomide The risk or severity of adverse effects can be increased when Daclizumab is combined with Thalidomide.
Melphalan The risk or severity of adverse effects can be increased when Daclizumab is combined with Melphalan.

Target Protein

Interleukin-2 receptor subunit alpha IL2RA
Interleukin-2 receptor subunit beta IL2RB
Low affinity immunoglobulin gamma Fc region receptor III-B FCGR3B
Complement C1r subcomponent C1R
Complement C1q subcomponent subunit A C1QA
Complement C1q subcomponent subunit B C1QB
Complement C1q subcomponent subunit C C1QC
Low affinity immunoglobulin gamma Fc region receptor III-A FCGR3A
High affinity immunoglobulin gamma Fc receptor I FCGR1A
Low affinity immunoglobulin gamma Fc region receptor II-a FCGR2A
Low affinity immunoglobulin gamma Fc region receptor II-b FCGR2B
Low affinity immunoglobulin gamma Fc region receptor II-c FCGR2C

Contoh Produk & Brand

Produk: 8 • International brands: 0
Produk
  • Zenapax
    Injection, solution, concentrate • 25 mg/5mL • Intravenous • US • Approved
  • Zenapax
    Injection, solution, concentrate • 25 mg • Intravenous • EU
  • Zenapax
    Injection, solution, concentrate • 25 mg • Intravenous • EU
  • Zenapax 5mg/ml
    Liquid • 5 mg / mL • Intravenous • Canada • Approved
  • Zinbryta
    Injection, solution • 150 mg/1mL • Subcutaneous • US • Approved
  • Zinbryta
    Solution • 150 mg / mL • Subcutaneous • Canada • Approved
  • Zinbryta
    Solution • 150 mg / mL • Subcutaneous • Canada • Approved
  • Zinbryta Pen
    Injection, solution • 150 mg/1mL • Subcutaneous • US • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul