Peringatan Keamanan

Reproductive toxicity studies in pregnant rhesus monkeys and golden Syrian hamsters demonstrated an increase in fetal loss in hamsters treated with Interferon alfacon-1 at doses of > 150 mcg/kg/day, and in rhesus monkeys at doses of 3 and 10 mcg/kg/day. The Interferon alfacon-1 toxicity profile described is consistent with the known toxicity profile of other alpha interferons.

Interferon alfacon-1

DB00069

biotech approved investigational

Deskripsi

Interferon alfacon-1 is a recombinant non-naturally occurring type-I interferon. The 166-amino acid sequence of Interferon alfacon-1 was derived by scanning the sequences of several natural interferon alpha subtypes and assigning the most frequently observed amino acid in each corresponding position. Four additional amino acid changes were made to facilitate the molecular construction, and a corresponding synthetic DNA sequence was constructed using chemical synthesis methodology. Interferon alfacon-1 differs from interferon alfa-2b at 20/166 amino acids (88% homology), and comparison with interferon-beta shows identity at over 30% of the amino acid positions. Interferon alfacon-1 is produced in Escherichia coli (E. coli) cells that have been genetically altered by insertion of a synthetically constructed sequence that codes for Interferon alfacon-1. Prior to final purification, Interferon alfacon-1 is allowed to oxidize to its native state, and its final purity is achieved by sequential passage over a series of chromatography columns. This protein has a molecular weight of 19,434 daltons.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The terminal half-life following subcutaneous dosing was 1.3 hours in golden Syrian hamsters and 3.4 hours in rhesus monkeys.
Volume Distribusi -
Klirens (Clearance) Clearance, averaging 1.99 mL/minute/kg in golden Syrian hamsters and 0.71 to 0.92 mL/minute/kg in rhesus monkeys

Absorpsi

Subcutaneous bioavailability averages 99% in golden Syrian hamsters and 83% to 104% in rhesus monkeys.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Due predominantly to catabolism and excretion by the kidneys.

Interaksi Obat

658 Data
Denosumab The risk or severity of adverse effects can be increased when Denosumab is combined with Interferon alfacon-1.
Etanercept The risk or severity of adverse effects can be increased when Etanercept is combined with Interferon alfacon-1.
Peginterferon alfa-2a The risk or severity of adverse effects can be increased when Peginterferon alfa-2a is combined with Interferon alfacon-1.
Interferon alfa-n1 The risk or severity of adverse effects can be increased when Interferon alfa-n1 is combined with Interferon alfacon-1.
Interferon alfa-n3 The risk or severity of adverse effects can be increased when Interferon alfa-n3 is combined with Interferon alfacon-1.
Peginterferon alfa-2b The risk or severity of adverse effects can be increased when Peginterferon alfa-2b is combined with Interferon alfacon-1.
Anakinra The risk or severity of adverse effects can be increased when Anakinra is combined with Interferon alfacon-1.
Interferon gamma-1b The risk or severity of adverse effects can be increased when Interferon gamma-1b is combined with Interferon alfacon-1.
Interferon alfa-2a The risk or severity of adverse effects can be increased when Interferon alfa-2a is combined with Interferon alfacon-1.
Adalimumab The risk or severity of adverse effects can be increased when Adalimumab is combined with Interferon alfacon-1.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Interferon alfacon-1.
Pegaspargase The risk or severity of adverse effects can be increased when Pegaspargase is combined with Interferon alfacon-1.
Infliximab The risk or severity of adverse effects can be increased when Infliximab is combined with Interferon alfacon-1.
Interferon beta-1b The risk or severity of adverse effects can be increased when Interferon beta-1b is combined with Interferon alfacon-1.
Rituximab The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Rituximab.
Basiliximab The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Basiliximab.
Muromonab The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Muromonab.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Ibritumomab tiuxetan.
Tositumomab The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Tositumomab.
Alemtuzumab The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Alemtuzumab.
Alefacept The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Alefacept.
Efalizumab The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Efalizumab.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Antithymocyte immunoglobulin (rabbit).
Interferon alfa-2b The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Interferon alfa-2b.
Daclizumab The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Daclizumab.
Phenylalanine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Phenylalanine.
Flunisolide The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Flunisolide.
Bortezomib The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Bortezomib.
Cladribine Interferon alfacon-1 may increase the immunosuppressive activities of Cladribine.
Carmustine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Carmustine.
Amsacrine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Amsacrine.
Bleomycin The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Bleomycin.
Chlorambucil The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Chlorambucil.
Raltitrexed The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Raltitrexed.
Mitomycin The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Mitomycin.
Bexarotene The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Bexarotene.
Vindesine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Vindesine.
Floxuridine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Floxuridine.
Indomethacin The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Indomethacin.
Tioguanine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Tioguanine.
Vinorelbine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Vinorelbine.
Dexrazoxane The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Dexrazoxane.
Beclomethasone dipropionate The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Beclomethasone dipropionate.
Sorafenib The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Sorafenib.
Streptozocin The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Streptozocin.
Trifluridine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Trifluridine.
Gemcitabine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Gemcitabine.
Betamethasone The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Betamethasone.
Teniposide The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Teniposide.
Epirubicin The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Epirubicin.
Chloramphenicol The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Chloramphenicol.
Lenalidomide The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Lenalidomide.
Altretamine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Altretamine.
Zidovudine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Zidovudine.
Cisplatin The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Cisplatin.
Oxaliplatin The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Oxaliplatin.
Cyclophosphamide The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Cyclophosphamide.
Vincristine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Vincristine.
Fluorouracil The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Fluorouracil.
Propylthiouracil The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Propylthiouracil.
Pentostatin The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Pentostatin.
Methotrexate The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Methotrexate.
Carbamazepine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Carbamazepine.
Vinblastine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Vinblastine.
Fluticasone propionate The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Fluticasone propionate.
Fluocinolone acetonide The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Fluocinolone acetonide.
Linezolid The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Linezolid.
Imatinib The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Imatinib.
Triamcinolone The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Triamcinolone.
Clofarabine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Clofarabine.
Prednisone The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Prednisone.
Pemetrexed The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Pemetrexed.
Fludrocortisone The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Fludrocortisone.
Mycophenolate mofetil The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Mycophenolate mofetil.
Daunorubicin The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Daunorubicin.
Irinotecan The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Irinotecan.
Methimazole The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Methimazole.
Etoposide The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Etoposide.
Sulfasalazine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Sulfasalazine.
Dacarbazine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Dacarbazine.
Temozolomide The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Temozolomide.
Penicillamine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Penicillamine.
Prednisolone The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Prednisolone.
Sirolimus The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Sirolimus.
Mechlorethamine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Mechlorethamine.
Azacitidine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Azacitidine.
Carboplatin The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Carboplatin.
Methylprednisolone The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Methylprednisolone.
Dactinomycin The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Dactinomycin.
Cytarabine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Cytarabine.
Azathioprine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Azathioprine.
Doxorubicin The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Doxorubicin.
Hydroxyurea The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Hydroxyurea.
Busulfan The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Busulfan.
Mycophenolic acid The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Mycophenolic acid.
Topotecan The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Topotecan.
Mercaptopurine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Mercaptopurine.
Thalidomide The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Thalidomide.
Melphalan The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Melphalan.
Fludarabine The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Fludarabine.

Target Protein

Interferon alpha/beta receptor 1 IFNAR1
Interferon alpha/beta receptor 2 IFNAR2

Referensi & Sumber

Synthesis reference: Lin Wang, " NEW TYPE OF CONSENSUS INTERFERON AND PREPARATION METHOD THEREOF." U.S. Patent US20100266536, issued October 21, 2010.
Artikel (PubMed)
  • PMID: 8836913
    Blatt LM, Davis JM, Klein SB, Taylor MW: The biologic activity and molecular characterization of a novel synthetic interferon-alpha species, consensus interferon. J Interferon Cytokine Res. 1996 Jul;16(7):489-99.
Link

Contoh Produk & Brand

Produk: 4 • International brands: 1
Produk
  • Infergen
    Injection • 0.03 mg/1mL • Subcutaneous • US • Approved
  • Infergen
    Injection • 0.03 mg/1mL • Subcutaneous • US • Approved
  • Infergen
    Injection • 0.03 mg/1mL • Subcutaneous • US • Approved
  • Infergen
    Solution • 0.03 mg / mL • Subcutaneous • Canada • Approved
International Brands
  • Advaferon

Sekuens Gen/Protein (FASTA)

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