Alpha-1-proteinase inhibitor

DB00058

biotech approved

Deskripsi

Human alpha-1 proteinase inhibitor or alpha-1-antitrypsin, prepared from human plasma via Cohn alcohol fractionation followed by PEG and zinc chloride fractionation.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi * 5632 ± 2006 mL [ARALAST NP] * 5618 ± 1618 mL [Aralast]
Klirens (Clearance) * 940 +/- 275 mL/day [Patients with congenital ?1-PI deficiency with single IV infusion of 60 mg/kg]

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

55 Data
Menadione Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Menadione.
Tranexamic acid Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Tranexamic acid.
Aminocaproic acid Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Aminocaproic acid.
Aprotinin Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Aprotinin.
Hydrogen peroxide Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Hydrogen peroxide.
Aminomethylbenzoic acid Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Aminomethylbenzoic acid.
Camostat Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Camostat.
Menadione bisulfite Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Menadione bisulfite.
Fibrinogen human The therapeutic efficacy of Fibrinogen human can be increased when used in combination with Alpha-1-proteinase inhibitor.
Antihemophilic factor, human recombinant Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Antihemophilic factor, human recombinant.
Coagulation factor VIIa Recombinant Human Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Coagulation factor VIIa Recombinant Human.
Coagulation Factor IX (Recombinant) Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Coagulation Factor IX (Recombinant).
Calcium Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Calcium.
Pantothenic acid Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Pantothenic acid.
Formic acid Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Formic acid.
Platelet Activating Factor Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Platelet Activating Factor.
Turoctocog alfa Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Turoctocog alfa.
Catridecacog Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Catridecacog.
Antihemophilic factor (recombinant), PEGylated Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Antihemophilic factor (recombinant), PEGylated.
Prothrombin Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Prothrombin.
Factor IX Complex (Human) Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Factor IX Complex (Human).
Susoctocog alfa Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Susoctocog alfa.
Eftrenonacog alfa Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Eftrenonacog alfa.
Rusalatide acetate Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Rusalatide acetate.
Vatreptacog alfa Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Vatreptacog alfa.
Factor XIII (human) Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Factor XIII (human).
Von Willebrand factor human Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Von Willebrand factor human.
Coagulation factor X human Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Coagulation factor X human.
Coagulation factor VII human Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Coagulation factor VII human.
Anti-inhibitor coagulant complex Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Anti-inhibitor coagulant complex.
Coagulation Factor IX Human Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Coagulation Factor IX Human.
Antihemophilic factor human Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Antihemophilic factor human.
Kallidinogenase Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Kallidinogenase.
Trenonacog alfa Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Trenonacog alfa.
Albutrepenonacog alfa Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Albutrepenonacog alfa.
Emicizumab Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Emicizumab.
Nonacog beta pegol Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Nonacog beta pegol.
Moroctocog alfa Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Moroctocog alfa.
Beroctocog alfa Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Beroctocog alfa.
Andexanet alfa Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Andexanet alfa.
Calcium cation Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Calcium cation.
Damoctocog alfa pegol Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Damoctocog alfa pegol.
Turoctocog alfa pegol Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Turoctocog alfa pegol.
Alteplase The therapeutic efficacy of Alpha-1-proteinase inhibitor can be decreased when used in combination with Alteplase.
Urokinase The therapeutic efficacy of Alpha-1-proteinase inhibitor can be decreased when used in combination with Urokinase.
Reteplase The therapeutic efficacy of Alpha-1-proteinase inhibitor can be decreased when used in combination with Reteplase.
Anistreplase The therapeutic efficacy of Alpha-1-proteinase inhibitor can be decreased when used in combination with Anistreplase.
Tenecteplase The therapeutic efficacy of Alpha-1-proteinase inhibitor can be decreased when used in combination with Tenecteplase.
Streptokinase The therapeutic efficacy of Alpha-1-proteinase inhibitor can be decreased when used in combination with Streptokinase.
Lanoteplase The therapeutic efficacy of Alpha-1-proteinase inhibitor can be decreased when used in combination with Lanoteplase.
Amediplase The therapeutic efficacy of Alpha-1-proteinase inhibitor can be decreased when used in combination with Amediplase.
Saruplase The therapeutic efficacy of Alpha-1-proteinase inhibitor can be decreased when used in combination with Saruplase.
Protein S human Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Protein S human.
Rurioctocog alfa pegol Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Rurioctocog alfa pegol.
Etranacogene dezaparvovec Alpha-1-proteinase inhibitor may increase the thrombogenic activities of Etranacogene dezaparvovec.

Target Protein

Neutrophil elastase ELANE

Referensi & Sumber

Synthesis reference: Michael H. Coan, William J. Brockway, "Method of preparing alpha-1-proteinase inhibitor." U.S. Patent US4379087, issued December, 1968.
Artikel (PubMed)
  • PMID: 16773239
    Karnaukhova E, Ophir Y, Golding B: Recombinant human alpha-1 proteinase inhibitor: towards therapeutic use. Amino Acids. 2006 Jun;30(4):317-32. Epub 2006 May 26.

Contoh Produk & Brand

Produk: 27 • International brands: 2
Produk
  • Alpha1-proteinase Inhibitor (human)
    Powder, for solution • 500 mg / vial • Intravenous • Canada • Approved
  • Alpha1-proteinase Inhibitor (human)
    Powder, for solution • 1 g / vial • Intravenous • Canada • Approved
  • Aralast NP
    Kit • 16 mg/1mL • Intravenous • US • Approved
  • Aralast NP
    Kit • 16 mg/1mL • Intravenous • US • Approved
  • Aralast NP
    Kit • 16 mg/1mL • Intravenous • US • Approved
  • Aralast NP
    Injection, powder, lyophilized, for solution; Kit • 16 mg/1mL • Intravenous • US • Approved
  • Aralast NP
    Injection, powder, lyophilized, for solution; Kit • 16 mg/1mL • Intravenous • US • Approved
  • Glassia
    Injection, solution • 1 g/50mL • Intravenous • US • Approved
Menampilkan 8 dari 27 produk.
International Brands
  • Aralast — Baxter
  • Prolastin — Talecris Biotherapeutics C formerly Bayer

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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