Gramicidin D

DB00027

small molecule approved

Deskripsi

Gramcidin D is a heterogeneous mixture of three antibiotic compounds, gramicidins A, B and C, making up 80%, 6%, and 14% respectively all of which are obtained from the soil bacterial species Bacillus brevis and called collectively gramicidin D. Gramcidins are 15 residue peptides with alternating D and L amino acids, which assemble inside of the hydrophobic interior of the cellular lipid bilayer to form a ?-helix. Active against most Gram-positive bacteria and some Gram-negative organisms, Gramicidin D is used primarily as a topical antibiotic and is also found in Polysporin ophthalmic solution.

Struktur Molekul 2D

Berat 1811.253
Wujud liquid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

55 Data
BCG vaccine The therapeutic efficacy of BCG vaccine can be decreased when used in combination with Gramicidin D.
Dicoumarol The risk or severity of bleeding can be increased when Gramicidin D is combined with Dicoumarol.
Phenindione The risk or severity of bleeding can be increased when Gramicidin D is combined with Phenindione.
Warfarin The risk or severity of bleeding can be increased when Gramicidin D is combined with Warfarin.
Phenprocoumon The risk or severity of bleeding can be increased when Gramicidin D is combined with Phenprocoumon.
Acenocoumarol The risk or severity of bleeding can be increased when Gramicidin D is combined with Acenocoumarol.
4-hydroxycoumarin The risk or severity of bleeding can be increased when Gramicidin D is combined with 4-hydroxycoumarin.
Coumarin The risk or severity of bleeding can be increased when Gramicidin D is combined with Coumarin.
(R)-warfarin The risk or severity of bleeding can be increased when Gramicidin D is combined with (R)-warfarin.
Ethyl biscoumacetate The risk or severity of bleeding can be increased when Gramicidin D is combined with Ethyl biscoumacetate.
Fluindione The risk or severity of bleeding can be increased when Gramicidin D is combined with Fluindione.
Clorindione The risk or severity of bleeding can be increased when Gramicidin D is combined with Clorindione.
Diphenadione The risk or severity of bleeding can be increased when Gramicidin D is combined with Diphenadione.
Tioclomarol The risk or severity of bleeding can be increased when Gramicidin D is combined with Tioclomarol.
(S)-Warfarin The risk or severity of bleeding can be increased when Gramicidin D is combined with (S)-Warfarin.
Vibrio cholerae CVD 103-HgR strain live antigen The therapeutic efficacy of Vibrio cholerae CVD 103-HgR strain live antigen can be decreased when used in combination with Gramicidin D.
Estetrol The therapeutic efficacy of Estetrol can be decreased when used in combination with Gramicidin D.
Lidocaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Lidocaine.
Ropivacaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Ropivacaine.
Bupivacaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Bupivacaine.
Cinchocaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Cinchocaine.
Dyclonine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Dyclonine.
Procaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Procaine.
Prilocaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Prilocaine.
Proparacaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Proparacaine.
Meloxicam The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Meloxicam.
Oxybuprocaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Oxybuprocaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Cocaine.
Mepivacaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Mepivacaine.
Levobupivacaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Levobupivacaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Diphenhydramine.
Benzocaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Benzocaine.
Chloroprocaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Chloroprocaine.
Phenol The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Phenol.
Tetrodotoxin The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Tetrodotoxin.
Benzyl alcohol The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Benzyl alcohol.
Capsaicin The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Capsaicin.
Etidocaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Etidocaine.
Articaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Articaine.
Tetracaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Tetracaine.
Propoxycaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Propoxycaine.
Pramocaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Pramocaine.
Butamben The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Butamben.
Butacaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Butacaine.
Oxetacaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Oxetacaine.
Ethyl chloride The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Ethyl chloride.
Butanilicaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Butanilicaine.
Metabutethamine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Metabutethamine.
Quinisocaine The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Quinisocaine.
Cisatracurium Gramicidin D may increase the neuromuscular blocking activities of Cisatracurium.
Ambroxol The risk or severity of methemoglobinemia can be increased when Gramicidin D is combined with Ambroxol.
Fecal microbiota The therapeutic efficacy of Fecal microbiota can be decreased when used in combination with Gramicidin D.
Picosulfuric acid The therapeutic efficacy of Picosulfuric acid can be decreased when used in combination with Gramicidin D.
Typhoid vaccine The therapeutic efficacy of Typhoid vaccine can be decreased when used in combination with Gramicidin D.
Lactulose The therapeutic efficacy of Lactulose can be decreased when used in combination with Gramicidin D.

Target Protein

Dihydropteroate synthase folP

Referensi & Sumber

Synthesis reference: U.S.Patent 2,534,541.
Artikel (PubMed)
  • PMID: 8810522
    Ketchem RR, Lee KC, Huo S, Cross TA: Macromolecular structural elucidation with solid-state NMR-derived orientational constraints. J Biomol NMR. 1996 Jul;8(1):1-14.
  • PMID: 11570868
    Townsley LE, Tucker WA, Sham S, Hinton JF: Structures of gramicidins A, B, and C incorporated into sodium dodecyl sulfate micelles. Biochemistry. 2001 Oct 2;40(39):11676-86.
  • PMID: 10397797
    Burkhart BM, Gassman RM, Langs DA, Pangborn WA, Duax WL, Pletnev V: Gramicidin D conformation, dynamics and membrane ion transport. Biopolymers. 1999;51(2):129-44.

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Sekuens Gen/Protein (FASTA)

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