Sargramostim

DB00020

biotech approved investigational

Deskripsi

Sargramostim is a human recombinant granulocyte macrophage colony-stimulating factor (GM-CSF) expressed in yeast. It is a glycoprotein that is 127 residues. Substitution of Leu23 leads to a difference from native protein.

Struktur Molekul 2D

Struktur tidak tersedia

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) * 420 mL/min/m2 [Normal people with liquid LEUKINE (IV)] * 431 mL/min/m2 [Normal people with lyophilized LEUKINE (IV)] * 549 mL/min/m2 [Normal people with liquid LEUKINE (SC)] * 529 mL/min/m2 [Normal people with lyophilized LEUKINE (SC)]

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

9 Data
Bleomycin The risk or severity of adverse effects can be increased when Sargramostim is combined with Bleomycin.
Cyclophosphamide The risk or severity of adverse effects can be increased when Cyclophosphamide is combined with Sargramostim.
Vindesine The risk or severity of peripheral neuropathy can be increased when Sargramostim is combined with Vindesine.
Vinorelbine The risk or severity of peripheral neuropathy can be increased when Sargramostim is combined with Vinorelbine.
Vincristine The risk or severity of peripheral neuropathy can be increased when Sargramostim is combined with Vincristine.
Vinblastine The risk or severity of peripheral neuropathy can be increased when Sargramostim is combined with Vinblastine.
Vintafolide The risk or severity of peripheral neuropathy can be increased when Sargramostim is combined with Vintafolide.
Vinflunine The risk or severity of peripheral neuropathy can be increased when Sargramostim is combined with Vinflunine.
Vincamine The risk or severity of peripheral neuropathy can be increased when Sargramostim is combined with Vincamine.

Target Protein

Granulocyte-macrophage colony-stimulating factor receptor subunit alpha CSF2RA
Interleukin-3 receptor subunit alpha IL3RA
Cytokine receptor common subunit beta CSF2RB
Syndecan-2 SDC2
Bone marrow proteoglycan PRG2

Referensi & Sumber

Synthesis reference: Kaname Sugimoto, "Process for the production of human colony-stimulating factor." U.S. Patent US4621050, issued May, 1983.

Contoh Produk & Brand

Produk: 10 • International brands: 1
Produk
  • Leukine
    Liquid • 500 ug/1mL • Intravenous; Subcutaneous • US • Approved
  • Leukine
    Injection, powder, for solution • 250 ug/1mL • Intravenous; Subcutaneous • US • Approved
  • Leukine
    Liquid • 500 ug/1mL • Intravenous; Subcutaneous • US • Approved
  • Leukine
    Liquid • 500 ug/1mL • Subcutaneous • US • Approved
  • Leukine
    Injection, powder, for solution • 250 ug/1mL • Subcutaneous • US • Approved
  • Leukine
    Liquid • 500 ug/1mL • Intravenous; Subcutaneous • US • Approved
  • Leukine
    Injection, powder, for solution • 250 ug/1mL • Intravenous; Subcutaneous • US • Approved
  • Leukine
    Liquid • 500 ug/1mL • Subcutaneous • US • Approved
Menampilkan 8 dari 10 produk.
International Brands
  • Leucomax — Novartis

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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