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Total database: 17430
Struktur (SMILES)
20 (87.0%)
Target
17 (73.9%)
Genomik
0 (0%)
Referensi
23 (100.0%)

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Distribusi Wujud Zat

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Hasil Pencarian (23)

small molecule | CAS: 156316-85-7

LR-103 is a naturally occurring D-hormone that is produced by the kidneys from vitamin D. LR-103 is one of the D-hormones produced from Hectorol. It is developed for the treatment of secondary hyperparathyroidism in patients with chronic kidney disease (CKD).…

Kategori:
CholestanesCholestenesFused-Ring Compounds +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 187935-17-7

1alpha-Hydroxyvitamin D5 (CARD-024) has been used in trials studying the treatment of Drug Safety and Heart; Disease, Activity.

Kategori:
CholestanesCholestenesFused-Ring Compounds +8
Target Protein:
Renin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 40013-87-4

Deskripsi belum tersedia.

Kategori:
Bone Density Conservation AgentsCalcium-Regulating Hormones and AgentsCholestanes +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 103656-40-2

24-Homo-1,25-dihydroxyvitamin D3 is a novel [vitamin D] analogue.

Kategori:
CholestanesCholestenesFused-Ring Compounds +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alfacalcidol Approved DB01436
small molecule | CAS: 41294-56-8

Alfacalcidol, or 1-alpha-hydroxycholecalciferol or 1-alpha-hydroxyvitamin D3, is a non-endogenous analogue of [vitamin D].[A234044] It plays an essential function in calcium homeostasis and bone metabolism. Alfacaldisol is activated by the enzyme 25-hydroxyla…

Kategori:
Alimentary Tract and MetabolismBone Density Conservation AgentsCholestanes +13
Target Protein:
Vitamin D3 receptor25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrialRetinoic acid receptor RXR-alpha
Waktu ParuhThe half-life of al…
Vol. Distribusi-
Klirens-
Genetik -
Becocalcidiol DB04891
small molecule | CAS: 524067-21-8

Becocalcidiol is a vitamin D(3) analogue which has not caused hypercalcaemia or significant irritation in preclinical trials.

Kategori:
CholestanesCholestenesFused-Ring Compounds +8
Target Protein:
Mediator of RNA polymerase II transcription subunit 1Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Calcifediol Approved DB00146
small molecule | CAS: 19356-17-3

The major circulating metabolite of vitamin D3 (cholecalciferol). It is produced in the liver and is the best indicator of the body's vitamin D stores. It is effective in the treatment of rickets and osteomalacia, both in azotemic and non-azotemic patients. C…

Kategori:
Alimentary Tract and MetabolismAnti-Parathyroid AgentsBone Density Conservation Agents +17
Target Protein:
Vitamin D3 receptor
Waktu Paruh288 hours
Vol. Distribusi-
Klirens-
Genetik -
Calcipotriol Approved DB02300
small molecule | CAS: 112965-21-6

Calcipotriol (INN) or calcipotriene (USAN) is a sythetic derivative of calcitriol or Vitamin D.

Kategori:
AntipsoriaticsAntipsoriatics for Topical UseCholestanes +12
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Calcitriol Approved DB00136
small molecule | CAS: 32222-06-3

Calcitriol is an active metabolite of vitamin D with 3 hydroxyl (OH) groups and is commonly referred to as 1,25-dihydroxycholecalciferol, or 1alpha,25-dihydroxyvitamin D<sub>3</sub>, 1,25-dihydroxyvitamin D<sub>3</sub>. It is produced in the body after series…

Kategori:
Alimentary Tract and MetabolismAntipsoriaticsAntipsoriatics for Topical Use +27
Target Protein:
Vitamin D3 receptorHomeobox protein Hox-A10
Waktu ParuhAfter administratio…
Vol. DistribusiUpon intravenous ad…
KlirensThe metabolic clear…
Genetik -
Cholecalciferol Approved DB00169
small molecule | CAS: 67-97-0

Vitamin D, in general, is a secosteroid generated in the skin when 7-dehydrocholesterol located there interacts with ultraviolet irradiation - like that commonly found in sunlight [L5689]. Both the endogenous form of vitamin D (that results from 7-dehydrochol…

Kategori:
Alimentary Tract and MetabolismBone Density Conservation AgentsCalcium-Regulating Hormones and Agents +28
Target Protein:
Vitamin D3 receptor
Waktu ParuhAt this time, there…
Vol. DistribusiStudies have determ…
KlirensStudies have determ…
Genetik -
CTA018 DB05024
small molecule

CTA018 is a member of a new class of vitamin D analogues with a dual mechanism of action, called Vitamin D Signal Amplifiers. This proprietary new drug is both a potent inhibitor of CYP24 (the enzyme responsible for the breakdown of vitamin D) and a potent ac…

Target Protein:
1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrialVitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dihydrotachysterol Approved DB01070
small molecule | CAS: 67-96-9

A vitamin D that can be regarded as a reduction product of vitamin D2.

Kategori:
Alimentary Tract and MetabolismBone Density Conservation AgentsCholestanes +14
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Doxercalciferol Approved DB06410
small molecule | CAS: 54573-75-0

Doxercalciferol is a synthetic vitamin D2 analog that undergoes metabolic activation in vivo to form 1?,25-dihydroxyvitamin D2 (1?,25-(OH)2D2), a naturally occurring, biologically active form of vitamin D2. Doxercalciferol is indicated for the treatment of se…

Kategori:
Anti-Parathyroid AgentsBone Density Conservation AgentsCalcium Homeostasis +16
Target Protein:
Vitamin D3 receptor
Waktu Paruh32 to 37 hours.
Vol. Distribusi-
Klirens-
Genetik -
EF-022 DB17768
biotech

EF-022 is a modified version of vitamin D binding protein macrophage activator, with potential antineoplastic and anti-angiogenic activities.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eldecalcitol DB05295
small molecule | CAS: 104121-92-8

Eldecalcitol (ED-71), a vitamin D analog, is a more potent inhibitor of bone resorption than alfacalcidol in an estrogen-deficient rat model of osteoporosis. Eldecalcitol, effectively and safely increased lumbar and hip bone mineral density (BMD) in osteopor…

Kategori:
Bone Density Conservation AgentsFused-Ring CompoundsSecosteroids +4
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ergocalciferol Approved DB00153
small molecule | CAS: 50-14-6

Ergocalciferol is an inactivated vitamin D analog.[A177526] It is synthesized by some plants in the presence of UVB light.[T577] The production of ergocalciferol was prompted by the identification of dietary deficiency, more specifically vitamin D, as the mai…

Kategori:
Alimentary Tract and MetabolismBone Density Conservation AgentsCalcium-Regulating Hormones and Agents +11
Target Protein:
Vitamin D3 receptorVoltage-dependent calcium channel
Waktu ParuhErgocalciferol can …
Vol. DistribusiThe amount of circu…
KlirensThere are no formal…
Genetik -
Ergosterol Approved DB04038
small molecule | CAS: 57-87-4

A steroid of interest both because its biosynthesis in FUNGI is a target of ANTIFUNGAL AGENTS, notably AZOLES, and because when it is present in SKIN of animals, ULTRAVIOLET RAYS break a bond to result in ERGOCALCIFEROL.

Kategori:
CholestanesCholestenesDiet, Food, and Nutrition +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lexacalcitol DB03451
small molecule | CAS: 131875-08-6

Lexacalcitol is a solid. This compound belongs to the vitamin D and derivatives class of chemicals. These are compounds containing a secosteroid backbone, usually secoergostane or secocholestane. It is known to target the vitamin D3 receptor.

Kategori:
Antineoplastic AgentsCholestanesCholestenes +11
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Niacin Approved DB00627
small molecule | CAS: 59-67-6

Niacin is a B vitamin used to treat vitamin deficiencies as well as hyperlipidemia, dyslipidemia, hypertriglyceridemia, and to reduce the risk of myocardial infarctions.[L7550,L7553,L7556,L7559,L7562,L7565]

Kategori:
Agents Causing Muscle ToxicityCardiovascular AgentsCytochrome P-450 CYP2D6 Inhibitors +31
Target Protein:
Hydroxycarboxylic acid receptor 3Diacylglycerol O-acyltransferase 2Hydroxycarboxylic acid receptor 2 +2
Waktu ParuhThe half life of ni…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Pantothenic acid Approved DB01783
small molecule | CAS: 79-83-4

Pantothenic acid, also called pantothenate or vitamin B5 (a B vitamin), is a water-soluble vitamin discovered by Roger J. Williams in 1919. For many animals, pantothenic acid is an essential nutrient as it is required to synthesize coenzyme-A (CoA), as well a…

Kategori:
AlanineAlimentary Tract and MetabolismAmino Acids +9
Target Protein:
Pantothenate kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paricalcitol Approved DB00910
small molecule | CAS: 131918-61-1

Paricalcitol is a synthetic vitamin D analog. Paricalcitol has been used to reduce parathyroid hormone levels. Paricalcitol is indicated for the prevention and treatment of secondary hyperparathyroidism associated with chronic renal failure.

Kategori:
Anti-Parathyroid AgentsBone Density Conservation AgentsCalcium Homeostasis +16
Target Protein:
Vitamin D3 receptor
Waktu Paruh4 to 6 hours
Vol. Distribusi* 30.8 ± 7.5 L [CKD…
Klirens* 1.49 +/- 0.60 L/h…
Genetik -
Previtamin D(3) DB15614
small molecule | CAS: 1173-13-3

Deskripsi belum tersedia.

Kategori:
CholestanesCholestenesFused-Ring Compounds +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vitamin D Approved DB11094
small molecule | CAS: 1406-16-2

Vitamin D ultimately comprises a group of lipid-soluble secosteroids responsible for a variety of biological effects, some of which include increasing the intestinal absorption of calcium, magnesium, and phosphate. With reference to human use, there are 2 mai…

Kategori:
Bone Density Conservation AgentsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +12
Target Protein:
Vitamin D3 receptorVitamin D-binding protein
Waktu ParuhAlthough certain st…
Vol. Distribusi-
KlirensSome studies propos…
Genetik -