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13

Total database: 17430
Struktur (SMILES)
12 (92.3%)
Target
10 (76.9%)
Genomik
0 (0%)
Referensi
13 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (13)

small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dalbavancin Approved DB06219
small molecule | CAS: 171500-79-1

Dalbavancin is a second-generation lipoglycopeptide antibiotic that was designed to improve on the natural glycopeptides currently available, such as vancomycin and teicoplanin [A4072, A4073]. Modifications from these older glycoprotein classes facilitated a …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
D-Ala-D-Ala moiety of NAM/NAG peptide subunits of peptidoglycanPancreatic triacylglycerol lipase
Waktu ParuhTerminal half life …
Vol. DistribusiClearance and volum…
Klirens0.0513 L/h [FDA Lab…
Genetik -
Dalfopristin Approved DB01764
small molecule | CAS: 112362-50-2

Dalfopristin is a combination of two antibiotics (Dalfopristin and quinupristin) used to treat infections by staphylococci and by vancomycin-resistant Enterococcus faecium. It is not effective against Enterococcus faecalis infections. Dalfopristin inhibits th…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +8
Target Protein:
Streptogramin A acetyltransferase
Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Daptomycin Approved DB00080
small molecule | CAS: 103060-53-3

Daptomycin is a cyclic lipopeptide antibacterial agent with a broad spectrum of activity against Gram-positive bacteria, including methicillin-susceptible and -resistant _Staphylococcus aureus_ (MSSA/MRSA) and vancomycin-resistant Enterococci (VRE).[A231379, …

Kategori:
Agents Causing Muscle ToxicityAmino Acids, Peptides, and ProteinsAnti-Bacterial Agents +11
Target Protein:
Dihydropteroate synthaseCytoplasmic membrane
Waktu ParuhDaptomycin has a re…
Vol. DistribusiDaptomycin has a ve…
KlirensDaptomycin administ…
Genetik -
small molecule | CAS: 101485-50-1

Deskripsi belum tersedia.

Target Protein:
Desvancosaminyl-vancomycin vancosaminetransferasedTDP-epi-vancosaminyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fidaxomicin Approved DB08874
small molecule | CAS: 873857-62-6

Fidaxomicin is a novel macrolide antibiotic used in the treatment of diarrhea caused by _Clostridioides_ (formerly _Clostridium_) _difficile_ in adult and pediatric patients over the age of 6 months.[L11575] Fidaxomicin is a naturally-occurring 18-member macr…

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
RNA polymerase sigma factor SigA
Waktu ParuhFollowing oral admi…
Vol. DistribusiFidaxomicin is main…
KlirensThere is limited in…
Genetik -
Oritavancin Approved DB04911
small molecule | CAS: 171099-57-3

Oritavancin is a glycopeptide antibiotic used for the treatment of skin infections. It was developed by The Medicines Company (acquired by Novartis).[L12858] Oritavancin was initially approved by the FDA in 2014 and formulated to combat susceptible gram-posit…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +24
Target Protein:
Dihydropteroate synthasePeptidoglycan precursorsBacterial cell wall peptide bridging segments +1
Waktu ParuhThe average termina…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of or…
Genetik -
Quinupristin Approved DB01369
small molecule | CAS: 120138-50-3

Quinupristin/dalfopristin is a combination of two antibiotics used to treat infections by staphylococci and by vancomycin-resistant Enterococcus faecium. Dalfopristin inhibits the early phase of protein synthesis in the bacterial ribosome and quinupristin inh…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
23S ribosomal RNA50S ribosomal protein L1050S ribosomal protein L22
Waktu Paruh3.1 hours
Vol. Distribusi-
Klirens-
Genetik -
Ridinilazole DB15308
small molecule | CAS: 308362-25-6

Ridinilazole is under investigation in clinical trial NCT02092935 (A Study of SMT19969 Compared With Vancomycin for the Treatment of Clostridium Difficile-Associated Diarrhoea (CDAD)).

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Surotomycin DB12076
small molecule | CAS: 1233389-51-9

Surotomycin has been used in trials studying the treatment of Diarrhea and Clostridium Difficile Infection. It is a benzenebutanoic acid derivative patented by Cubist Pharmaceuticals, Inc. as antibacterial agents for the treatment of Gram-positive infections.…

Kategori:
Amino Acids, Peptides, and ProteinsLipidsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tedizolid Approved DB14569
small molecule | CAS: 856866-72-3

Drug-resistant bacteria, such as methicillin-resistant _Staphylococcus aureus_, vancomycin-resistant _Enterococcus faecium_, and penicillin-resistant _Streptococcus penumoniae_, represent a massive public health threat.[A199086, A199131] Tedizolid is a member…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +5
Target Protein:
23S ribosomal RNA
Waktu ParuhTedizolid has a hal…
Vol. DistribusiThe volume of distr…
KlirensTedizolid has an ap…
Genetik -
Tedizolid phosphate Approved DB09042
small molecule | CAS: 856867-55-5

Drug-resistant bacteria, such as methicillin-resistant _Staphylococcus aureus_, vancomycin-resistant _Enterococcus faecium_, and penicillin-resistant _Streptococcus penumoniae_, represent a massive public health threat.[A199086, A199131] Tedizolid is a member…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntidepressive Agents +10
Target Protein:
23S ribosomal RNA
Waktu ParuhTedizolid has a hal…
Vol. DistribusiThe volume of distr…
KlirensTedizolid has an ap…
Genetik -
Vancomycin Approved DB00512
small molecule | CAS: 1404-90-6

Antibacterial obtained from Streptomyces orientalis. It is a glycopeptide related to ristocetin that inhibits bacterial cell wall assembly and is toxic to kidneys and the inner ear. As of January 29 2018, CutisPharma's Firvanq is the only FDA approved vanc…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAmino Acids, Peptides, and Proteins +17
Target Protein:
D-Ala-D-Ala moiety of NAM/NAG peptide subunits of peptidoglycan
Waktu ParuhHalf-life in normal…
Vol. DistribusiThe volume of distr…
KlirensThe mean plasma cle…
Genetik -