Hasil Filter

12

Total database: 17430
Struktur (SMILES)
11 (91.7%)
Target
8 (66.7%)
Genomik
1 (8.3%)
Referensi
12 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (12)

Doravirine Approved DB12301
small molecule | CAS: 1338225-97-0

Doravirine is an HIV-1 non-nucleoside reverse transcriptase inhibitor (NNRTI) intended to be administered in combination with other antiretroviral medicines.[L12729,L4562] Doravirine is available by itself or as a combination product of doravirine (100 mg), l…

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +10
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu ParuhThe elimination hal…
Vol. DistribusiThe steady-state vo…
KlirensThe oral and renal …
Genetik -
Efavirenz Approved DB00625
small molecule | CAS: 154598-52-4

Efavirenz (brand names Sustiva® and Stocrin®) is a non-nucleoside reverse transcriptase inhibitor (NNRTI) and is used as part of highly active antiretroviral therapy (HAART) for the treatment of a human immunodeficiency virus (HIV) type 1. For HIV infectio…

Kategori:
Anti-Infective AgentsAnti-Retroviral AgentsAntiinfectives for Systemic Use +52
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Gen Terkait:
CYP2B6
Waktu Paruh40-55 hours
Vol. Distribusi-
Klirens-
Genetik 1 Varian
Emtricitabine Approved DB00879
small molecule | CAS: 143491-57-0

Emtricitabine is a nucleoside reverse transcriptase inhibitor (NRTI) indicated for the treatment of HIV infection in adults[L9019] or combined with [tenofovir alafenamide] for the prevention of HIV-1 infection in high risk adolescents and adults.[L9010] Emtri…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +23
Target Protein:
Reverse transcriptase/RNaseHGag-Pol polyprotein
Waktu ParuhThe half life of em…
Vol. DistribusiThe apparent centra…
KlirensEmtricitabine has a…
Genetik -
small molecule | CAS: 1951476-79-1

Fosclevudine alafenamide is under investigation in clinical trial NCT05238844 (A Study of Safety and Efficacy of ATI-2173 and Vebicorvir in Combination With Tenofovir Disoproxil Fumarate in Subjects With Chronic Hepatitis B Virus Infection).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Inarigivir DB15062
small molecule | CAS: 475650-36-3

Inarigivir is under investigation in clinical trial NCT03434353 (Study to Evaluate the Antiviral Activity of Inarigivir (GS-9992) Plus Tenofovir Alafenamide (TAF) for 12 Weeks in Adults With Chronic Hepatitis B (CHB)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 942123-43-5

Inarigivir soproxil is under investigation in clinical trial NCT03434353 (Study to Evaluate the Antiviral Activity of Inarigivir (GS-9992) Plus Tenofovir Alafenamide (TAF) for 12 Weeks in Adults With Chronic Hepatitis B (CHB)).

Target Protein:
Nucleotide-binding oligomerization domain-containing protein 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Myrcludex B DB14853
biotech | CAS: 406461-66-3

Myrcludex B is under investigation in clinical trial NCT03546621 (A Multicenter, Open-label, Randomized Clinical Study to Assess Efficacy and Safety of 3 Doses of Myrcludex B for 24 Weeks in Combination With Tenofovir Compared to Tenofovir Alone to Suppress H…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tenofovir DB14126
small molecule | CAS: 147127-20-6

Tenofovir is an acyclic nucleotide diester analog of adenosine monophosphate.[A37693] In the most strict sense and due to the fact that it presents a phosphate group bound to the nitrogenous base, it is determined as an actual nucleotide analog.[A37693] The a…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +16
Target Protein:
Reverse transcriptase/RNaseHGag-Pol polyproteinReverse transcriptase +1
Waktu ParuhThe reported half-l…
Vol. DistribusiAccumulation of ten…
KlirensThe clearance of te…
Genetik -
Tenofovir alafenamide Approved DB09299
small molecule | CAS: 379270-37-8

Tenofovir alafenamide is a novel [tenofovir] prodrug developed in order to improve renal safety when compared to the counterpart [tenofovir disoproxil].[A178060] Both of these prodrugs were first created to cover the polar phosphonic acid group on tenofovir b…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntiinfectives for Systemic Use +25
Target Protein:
Reverse transcriptase/RNaseHGag-Pol polyproteinReverse transcriptase +1
Waktu ParuhThe reported half-l…
Vol. DistribusiIn clinical trials,…
KlirensThe reported cleara…
Genetik -
small molecule | CAS: 1571076-26-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tenofovir disoproxil Approved DB00300
small molecule | CAS: 201341-05-1

Tenofovir disoproxil fumarate (a prodrug of tenofovir), marketed by Gilead Sciences under the trade name _Viread_, belongs to a class of antiretroviral drugs known as nucleotide analogue reverse transcriptase inhibitors (nRTIs). This drug is prescribed in co…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +19
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseHProtein P
Waktu ParuhWhen a single oral …
Vol. DistribusiThe volume of distr…
KlirensThe clearance of te…
Genetik -
small molecule | CAS: 911208-73-6

Tenofovir exalidex is under investigation in clinical trial NCT01080820 (A Safety, Tolerability and Pharmacokinetic Study of a Single Dose of CMX157 in Healthy Volunteers).

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +4
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -