Hasil Filter

2

Total database: 17430
Struktur (SMILES)
0 (0%)
Target
2 (100.0%)
Genomik
0 (0%)
Referensi
2 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (2)

Alteplase Approved DB00009
biotech | CAS: 105857-23-6

Alteplase is a recombinant tissue plasminogen activator (rt-PA) used as a thrombolytic agent.[L43125] It cleaves plasminogen to form plasmin, an enzyme involved in the degradation of fibrin clots. In the absence of fibrin, the alteplase-mediated conversion of…

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +19
Target Protein:
PlasminogenFibrinogen alpha chainFibrinogen gamma chain +1
Waktu ParuhAlteplase has an in…
Vol. DistribusiThe initial volume …
KlirensAlteplase has a pla…
Genetik -
Tenecteplase Approved DB00031
biotech | CAS: 191588-94-0

Tenecteplase is a tissue plasminogen activator (tPA) developed from modifications of natural human tPA complementary DNA (cDNA). It is a 527 amino acid with a substitution of threonine 103 with asparagine and substitution of asparagine 117 with glutamine with…

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +17
Target Protein:
Plasminogen
Waktu Paruh1.9 hours (mammalia…
Vol. Distribusi-
Klirens* 99 - 119 mL/min […
Genetik -