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Total database: 17430
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Hasil Pencarian (2)

Pralsetinib Approved DB15822
small molecule | CAS: 2097132-94-8

Pralsetinib, similar to the previously approved [selpercatinib], is a kinase inhibitor with enhanced specificity for RET tyrosine kinase receptors (RTKs) over other RTK classes.[A202055, A219751, L15986] Enhanced RET (Rearranged during transfection) oncogene …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +38
Target Protein:
Proto-oncogene tyrosine-protein kinase receptor RetEpithelial discoidin domain-containing receptor 1NT-3 growth factor receptor +8
Waktu ParuhPralsetinib has a p…
Vol. DistribusiPralsetinib has a m…
KlirensPralsetinib has a m…
Genetik -
Selpercatinib Approved DB15685
small molecule | CAS: 2152628-33-4

Selpercatinib is a kinase inhibitor with enhanced specificity for RET tyrosine kinase receptors (RTKs) over other RTK classes.[A202055, A202052, L13604] Enhanced RET (Rearranged during transfection) oncogene expression is a hallmark of many cancers. Although …

Kategori:
Agents that produce hypertensionAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Proto-oncogene tyrosine-protein kinase receptor RetVascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 3 +3
Waktu ParuhSelpercatinib has a…
Vol. DistribusiSelpercatinib has a…
KlirensSelpercatinib has a…
Genetik -